SCHEMBL212810

SCHEMBL212810

O=C1NN=C(c2ccccc2)C(c2ccccc2)O1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.50
PDE3B Q13370 6/20 0.45
PDE3A Q14432 6/20 0.45
ALDH1A1 P00352 3/20 0.42
KMT2A Q03164 3/20 0.42
KDM4E B2RXH2 2/20 0.42
MAPT P10636 2/20 0.42
GAA P10253 1/20 0.42
HPGD P15428 1/20 0.42
GFER P55789 1/20 0.42
HSD17B10 Q99714 1/20 0.42
GPR119 Q8TDV5 4/20 0.42
RAB9A P51151 1/20 0.40
SLC6A3 Q01959 1/20 0.40
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
POLB P06746 2/20 0.36
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7112822 0.87 PDE3B (0.50) PDE3BPDE3A
SCHEMBL4649359 0.78 PDE3B (0.71) PDE3BPDE3AGPR119PDE4APDE4B
SCHEMBL4650466 0.77 KDM4E (0.49) CA2PDE3BPDE3AALDH1A1KMT2A
SCHEMBL41171 0.74 RAB9A (0.47) CA2ALDH1A1KMT2AKDM4EMAPT
SCHEMBL11248792 0.71 PDE3B (0.38) PDE3BPDE3AALDH1A1KMT2AKDM4E
SCHEMBL9188792 0.70 CA2 (0.65) CA2ALDH1A1KMT2AKDM4EMAPT
SCHEMBL6766023 0.70 CA2 (0.50) CA2ALDH1A1KMT2AKDM4EMAPT
SCHEMBL3290342 0.69 RAB9A (0.42) CA2ALDH1A1KMT2AKDM4EMAPT
Carbamic Acid SCHEMBL6809303 0.68 RAB9A (0.45) CA2ALDH1A1KMT2AKDM4EMAPT
Pemoline Dione SCHEMBL7864463 0.67 CA2 (1.00) CA2ALDH1A1KMT2AKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 57 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4683247-A Foamable thermoplastic compositions, foamed articles and foaming method based on pre-compounded nucleating agent-resin concentrate GENERAL ELECTRIC COMPANY (US) 1987-07-28 US claimed
US-4163037-A USING A DIHYDROOXADIAZINONE BLOWING AGENT, INJECTION MOLDING GENERAL ELECTRIC COMPANY (US) 1979-07-31 US claimed
US-4097425-A POLYCARBONATES, POLYESTERS, SUBSTITUTED 3,6-DIHYDRO-1,3,4-OXDIAZIN-2-ONE GENERAL ELECTRIC COMPANY (US) 1978-06-27 US claimed
US-20240093512-A1 PHOTO-CURABLE INSULATION FOAM, DISPENSER FOR INJECTION THEREOF, AND METHODS OF USING SAME IN THE INSULATION CERTAINTEED LLC 2024-03-21 US disclosed
US-10119004-B2 Foam, composition, and method CERTAINTEED CORPORATION (US) 2018-11-06 US disclosed
EP-3381975-A1 FOAM, COMPOSITION, AND METHOD CertainTeed Corporation (US) 2018-10-03 EP disclosed
EP-2797995-B1 FOAM, COMPOSITION, AND METHOD CERTAIN TEED CORP (US) 2018-05-23 EP disclosed
US-20170190863-A1 FOAM, COMPOSITION, AND METHOD CERTAINTEED LLC 2017-07-06 US disclosed
US-9617412-B2 Foam, composition, and method CERTAINTEED CORPORATION (US) 2017-04-11 US disclosed
US-20160340909-A1 WALL PANEL SYSTEMS AND METHODS OF ASSEMBLING AND REFINISHING WALL PANEL SYSTEMS Green Bay Decking, LLC (US) 2016-11-24 US disclosed
US-9487654-B2 Foam, composition, and method CERTAINTEED CORPORATION (US) 2016-11-08 US disclosed
US-4587272-A Foamable polycarbonate compositions, articles and methods GENERAL ELECTRIC COMPANY (US) 1986-05-06 US disclosed
US-4544677-A IMPACT STRENGTH GENERAL ELECTRIC COMPANY (US) 1985-10-01 US disclosed
US-4543368-A DIHYDRODIAZINONE BLOWING AGENT GENERAL ELECTRIC COMPANY (US) 1985-09-24 US disclosed
US-4334030-A INJECTION MOLDABLE CONCENTRATES CONTAINING AMIDE DERIVATIVES OF AZODICARBOXYLIC ACID AND A DIHYDROOXADIAZINONE AS BLOWING AGENTS GENERAL ELECTRIC COMPANY (US) 1982-06-08 US disclosed
US-4163037-A USING A DIHYDROOXADIAZINONE BLOWING AGENT, INJECTION MOLDING GENERAL ELECTRIC COMPANY (US) 1979-07-31 US disclosed
US-4160088-A HALOGENATION OF KETONE, ALKANOL, HYDROLYSIS GENERAL ELECTRIC COMPANY (US) 1979-07-03 US disclosed
US-4158094-A BLOWING AGENTS GENERAL ELECTRIC COMPANY (US) 1979-06-12 US disclosed
US-4097671-A 5-PHENYL-3,6-DIHYDRO-1,3,4-OXADIAZIN-2-ONE, THERMOPLASTIC POLYMER BLOWING AGENT GENERAL ELECTRIC COMPANY (US) 1978-06-27 US disclosed
US-4097425-A POLYCARBONATES, POLYESTERS, SUBSTITUTED 3,6-DIHYDRO-1,3,4-OXDIAZIN-2-ONE GENERAL ELECTRIC COMPANY (US) 1978-06-27 US disclosed