SCHEMBL21384569

SCHEMBL21384569

O=C(O)c1cc(Br)c(F)cc1NS(=O)(=O)C1CC1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ACLY P53396 2/20 0.48
KCNK2 O95069 1/20 0.42
KCNK10 P57789 1/20 0.42
MRGPRX1 Q96LB2 7/20 0.39
TSPO P30536 2/20 0.38
HDAC4 P56524 1/20 0.37
SIRT6 Q8N6T7 1/20 0.35
HRH1 P35367 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
BRAF P15056 1/20 0.35
KDM4E B2RXH2 1/20 0.34
GPR27 Q9NS67 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21384577 0.85 MRGPRX1 (0.42) ACLYMRGPRX1TSPOSIRT6HRH1
SCHEMBL21384590 0.83 ACLY (0.48) ACLYMRGPRX1
SCHEMBL15847893 0.77 ACLY (0.60) ACLYMRGPRX1TSPOHRH1KDM4E
SCHEMBL21384564 0.77 METAP2 (0.56) ACLYMRGPRX1TSPOTDP1KDM4E
SCHEMBL31433781 0.77 ROCK2 (0.48) KCNK2KCNK10TDP1KDM4E
SCHEMBL21381491 0.72 ACLY (0.61) ACLYMRGPRX1KDM4E
SCHEMBL16004173 0.72 KCNK2 (0.49) KCNK2KCNK10TDP1KDM4E
SCHEMBL15847815 0.71 ACLY (0.51) ACLYMRGPRX1TSPOBRAFKDM4E
Hydrochloric Acid SCHEMBL21988903 0.71 KCNK2 (0.48) KCNK2KCNK10SIRT6TDP1KDM4E
Hydrochloric Acid SCHEMBL15994581 0.71 KCNK2 (0.48) KCNK2KCNK10SIRT6TDP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019179436-A1 ACID AMIDE COMPOUND AND USE THEREOF IN TREATMENT OF CANCERS 成都海创药业有限公司 2019-09-26 WO disclosed