SCHEMBL21392051

SCHEMBL21392051

CCOC(=O)C(C(=O)OC(C)(C)C)c1nccc(N(Cc2ccc(OC)cc2)SC2CC2)n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 2/20 0.36
BRD4 O60885 1/20 0.33
APLNR P35414 4/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
ALDH1A1 P00352 2/20 0.33
HTT P42858 1/20 0.33
SLC2A1 P11166 1/20 0.33
TRPM8 Q7Z2W7 1/20 0.33
LMNA P02545 2/20 0.32
TDP1 Q9NUW8 1/20 0.32
RPLP1 P05386 1/20 0.32
RPLP0 P05388 1/20 0.32
RPS17 P08708 1/20 0.32
RPSA P08865 1/20 0.32
RPS2 P15880 1/20 0.32
RPL35A P18077 1/20 0.32
RPL7 P18124 1/20 0.32
RPL17 P18621 1/20 0.32
RPS4Y1 P22090 1/20 0.32
RPS3 P23396 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21392050 0.83 CACNA1B (0.35) CACNA1BBRD4APLNRSMN1; SMN2ALDH1A1
SCHEMBL21392159 0.81 SLC2A1 (0.32) CACNA1BBRD4SMN1; SMN2ALDH1A1HTT
SCHEMBL21392168 0.78 APLNR (0.33) APLNRSMN1; SMN2ALDH1A1HTTTRPM8
SCHEMBL21391987 0.73 CLK4 (0.36) SMN1; SMN2ALDH1A1HTTLMNAKCNH2
SCHEMBL21392246 0.70 APLNR (0.35) APLNRSMN1; SMN2ALDH1A1HTTLMNA
SCHEMBL21392292 0.70 ALDH1A1 (0.35) CACNA1BALDH1A1LMNAKDM4EUSP2
SCHEMBL21392335 0.69 MLYCD (0.35) CACNA1BAPLNRSMN1; SMN2ALDH1A1HTT
SCHEMBL21392038 0.68 MAPT (0.35) SMN1; SMN2TRPM8LMNAKDM4EUSP2
SCHEMBL21392162 0.68 APLNR (0.36) BRD4APLNRSMN1; SMN2ALDH1A1HTT
SCHEMBL21392148 0.68 LMNA (0.33) CACNA1BAPLNRALDH1A1SLC2A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019180244-A1 AMINOPYRIMIDINE DERIVATIVES AS CTPS1 INHIBITORS STEP PHARMA S.A.S. (FR) 2019-09-26 WO disclosed
WO-2019179652-A1 AMINOPYRIMIDINE DERIVATIVES AS CTPS1 INHIBITORS STEP PHARMA S.A.S. (FR) 2019-09-26 WO disclosed