SCHEMBL21392292

SCHEMBL21392292

CCC(C)(C(=O)OC)c1ccnc(N(Cc2ccc(OC)cc2)SC2CC2)n1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 2/20 0.35
AR P10275 1/20 0.34
PTGER2 P43116 2/20 0.33
CACNA1B Q00975 1/20 0.33
ASPH Q12797 1/20 0.33
KDM8 Q8N371 1/20 0.33
LMNA P02545 2/20 0.33
CXCR3 P49682 1/20 0.33
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33
POLB P06746 1/20 0.33
KMT2A Q03164 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
USP2 O75604 1/20 0.32
TSHR P16473 1/20 0.32
MAPT P10636 1/20 0.32
EPHX2 P34913 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21392335 0.83 MLYCD (0.35) ALDH1A1KDM4ECACNA1BLMNAPOLB
SCHEMBL21392038 0.83 MAPT (0.35) KDM4EASPHKDM8LMNAUSP2
SCHEMBL21392148 0.83 LMNA (0.33) ALDH1A1PTGER2CACNA1BLMNACXCR3
SCHEMBL30416683 0.81 CXCR3 (0.35) ALDH1A1KDM4EPTGER2CXCR3
SCHEMBL21392147 0.81 CXCR3 (0.35) ALDH1A1KDM4EPTGER2CXCR3
SCHEMBL22762439 0.80 LMNA (0.33) ALDH1A1LMNAL3MBTL1USP2TSHR
SCHEMBL21392320 0.78 USP2 (0.35) ALDH1A1KDM4EARPTGER2ASPH
SCHEMBL21392246 0.76 APLNR (0.35) ALDH1A1KDM4EASPHKDM8LMNA
SCHEMBL21392076 0.76 MLYCD (0.33) ALDH1A1KDM4ELMNAPOLBKMT2A
SCHEMBL21392159 0.73 SLC2A1 (0.32) ALDH1A1KDM4ECACNA1BLMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019179652-A1 AMINOPYRIMIDINE DERIVATIVES AS CTPS1 INHIBITORS STEP PHARMA S.A.S. (FR) 2019-09-26 WO disclosed