SCHEMBL21392320

SCHEMBL21392320

COCCC(C)(C(=O)OC)c1ccnc(N(Cc2ccc(OC)cc2)SC)n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.35
TSHR P16473 1/20 0.35
AR P10275 1/20 0.34
ALDH1A1 P00352 5/20 0.34
KDM4E B2RXH2 1/20 0.34
ASPH Q12797 1/20 0.34
KDM8 Q8N371 1/20 0.34
SMN1; SMN2 Q16637 4/20 0.33
NR1H4 Q96RI1 2/20 0.33
KMT2A Q03164 3/20 0.33
GAA P10253 1/20 0.33
RAB9A P51151 2/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
L3MBTL1 Q9Y468 3/20 0.32
MEN1 O00255 2/20 0.32
HTT P42858 2/20 0.32
ALOX12 P18054 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
TDP1 Q9NUW8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21392150 0.86 RAB9A (0.32) USP2TSHRARALDH1A1KDM4E
SCHEMBL21384620 0.84 PTPN1 (0.39) USP2TSHRALDH1A1LMNAMAPT
SCHEMBL30725707 0.84 PTPN1 (0.39) USP2TSHRALDH1A1LMNAMAPT
SCHEMBL21392075 0.82 ALDH1A1 (0.35) USP2TSHRALDH1A1SMN1; SMN2KMT2A
SCHEMBL21392292 0.78 ALDH1A1 (0.35) USP2TSHRARALDH1A1KDM4E
SCHEMBL21392074 0.74 USP2 (0.35) USP2TSHRALDH1A1KDM4EASPH
SCHEMBL21384619 0.74 CASP6 (0.44) ARSMN1; SMN2KMT2AGAARAB9A
SCHEMBL21392152 0.71 PTPN1 (0.36) ALDH1A1LMNAMAPTPTGER2
SCHEMBL30415860 0.71 PTPN1 (0.36) ALDH1A1LMNAMAPTPTGER2
SCHEMBL21392147 0.69 CXCR3 (0.35) ALDH1A1KDM4ESMN1; SMN2GAAPTGER2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019179652-A1 AMINOPYRIMIDINE DERIVATIVES AS CTPS1 INHIBITORS STEP PHARMA S.A.S. (FR) 2019-09-26 WO disclosed