SCHEMBL2145850

SCHEMBL2145850

O=CC(c1ccncc1)c1cccc(Br)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.39
SLC6A2 P23975 2/20 0.37
SLC6A4 P31645 2/20 0.37
SLC6A3 Q01959 2/20 0.37
KMT2A Q03164 1/20 0.36
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
MAPT P10636 1/20 0.35
MAPK1 P28482 1/20 0.35
GRK2 P25098 1/20 0.33
CDC7 O00311 1/20 0.33
HSD11B1 P28845 1/20 0.33
CTSA P10619 1/20 0.32
CYP1A1 P04798 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP1B1 Q16678 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2756356 0.88 ALDH1A1 (0.48) ALDH1A1IDO1TDO2MAPK1HSD11B1
SCHEMBL931178 0.86 IDO1 (0.47) ALDH1A1KMT2AIDO1TDO2MAPT
Bromide SCHEMBL11274115 0.83 KCNA5 (0.41) ALDH1A1SLC6A2SLC6A4SLC6A3KMT2A
SCHEMBL8309987 0.80 LMNA (0.42) ALDH1A1SLC6A2SLC6A4SLC6A3KMT2A
SCHEMBL3907301 0.80 CYP19A1 (0.41) SLC6A2SLC6A4SLC6A3KMT2AIDO1
SCHEMBL3403146 0.80 CYP11B1 (0.41) SLC6A2SLC6A4SLC6A3IDO1TDO2
SCHEMBL6510105 0.80 MAPKAPK2 (0.44) SLC6A2SLC6A4SLC6A3KMT2ANPC1
SCHEMBL1515763 0.80 SLC6A3 (0.58) ALDH1A1SLC6A2SLC6A4SLC6A3KMT2A
SCHEMBL6501433 0.76 SLC6A2 (0.40) ALDH1A1SLC6A2SLC6A4SLC6A3MAPT
SCHEMBL7555691 0.76 CES2 (0.46) IDO1TDO2NPC1RAB9AGRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011085269-A1 RAF KINASE INHIBITORS SELEXAGEN THERAPEUTICS, INC. (US) 2011-07-14 WO disclosed