SCHEMBL2147241

SCHEMBL2147241

CCOC(=O)c1c[nH]nc1O

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.50
MEN1 O00255 3/20 0.50
TSHR P16473 1/20 0.50
ALDH1A1 P00352 5/20 0.47
CA12 O43570 5/20 0.46
CA1 P00915 5/20 0.46
CA2 P00918 5/20 0.46
CA7 P43166 5/20 0.46
CA9 Q16790 5/20 0.46
CA14 Q9ULX7 5/20 0.46
MAPT P10636 2/20 0.45
LMNA P02545 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
PDE4D Q08499 1/20 0.44
KDM4E B2RXH2 3/20 0.44
HSD17B10 Q99714 1/20 0.43
ESR1 P03372 1/20 0.43
ESR2 Q92731 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL263628 0.83 TSHR (0.52) KMT2AMEN1TSHRALDH1A1CA12
SCHEMBL161443 0.81 KMT2A (0.50) KMT2AMEN1TSHRALDH1A1CA12
SCHEMBL3376695 0.81 KDM4E (0.51) KMT2AMEN1TSHRALDH1A1CA12
SCHEMBL3356162 0.80 KMT2A (0.49) KMT2AMEN1TSHRALDH1A1CA12
SCHEMBL370881 0.80 KMT2A (0.49) KMT2AMEN1TSHRALDH1A1CA12
SCHEMBL23824155 0.80 KMT2A (0.49) KMT2AMEN1TSHRALDH1A1MAPT
SCHEMBL416936 0.80 KMT2A (0.49) KMT2AMEN1TSHRALDH1A1CA12
SCHEMBL309808 0.80 ALDH1A1 (0.54) KMT2AMEN1TSHRALDH1A1MAPT
SCHEMBL3261638 0.79 TSHR (0.52) KMT2AMEN1TSHRALDH1A1MAPT
SCHEMBL3721899 0.79 TSHR (0.52) KMT2AMEN1TSHRALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 141 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116283778-A Pyrazolecarboxylic acid compound as well as preparation method and application thereof 江苏理工学院 2023-06-23 CN claimed
CN-111057006-B Preparation method of 1- (4-chlorphenyl) -3-pyrazole alcohol 浙江工业大学 2021-08-03 CN claimed
CN-111057006-A Preparation method of 1- (4-chlorphenyl) -3-pyrazole alcohol 浙江工业大学 2020-04-24 CN claimed
US-12624024-B2 EP2 antagonist compounds RESERVOIR NEUROSCIENCE, INC. (US) 2026-05-12 US disclosed
US-20260125363-A1 PROCESSES FOR MAKING MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMA (US) 2026-05-07 US disclosed
EP-3697774-B1 CRYSTALLINE FORMS AND COMPOSITIONS OF CFTR MODULATORS VERTEX PHARMA (US) 2025-09-24 EP disclosed
US-12415798-B2 Processes for making modulators of cystic fibrosis transmembrane conductance regulator VERTEX PHARMACEUTICALS INCORPORATED (US) 2025-09-16 US disclosed
CN-116283778-B Pyrazolecarboxylic acid compound as well as preparation method and application thereof 江苏理工学院 2025-08-29 CN disclosed
EP-4499630-A1 BCL-XL INHIBITORS BeiGene, Ltd. (KY) 2025-02-05 EP disclosed
US-20250034128-A1 BCL-XL INHIBITORS BEIGENE, LTD. (KY) 2025-01-30 US disclosed
US-12122788-B2 Process of making CFTR modulators VERTEX PHARMACEUTICALS INCORPORATED (US) 2024-10-22 US disclosed
EP-1457490-A1 5-membered N-heterocyclic compounds with hypoglycemic and hypolipidemic activity Takeda Chemical Industries, Ltd. (JP) 2004-09-15 EP disclosed
EP-1445254-A1 PROCESS FOR PRODUCTION OF PYRAZOLE COMPOUNDS Takeda Chemical Industries, Ltd. (JP) 2004-08-11 EP disclosed
EP-1228067-B1 5-MEMBERED N-HETEROCYCLIC COMPOUNDS WITH HYPOGLYCEMIC AND HYPOLIPIDEMIC ACTIVITY TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2004-07-14 EP disclosed
US-20040063775-A1 Five-membered heterocyclic alkanoic acid derivative TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2004-04-01 US disclosed
EP-1394154-A1 FIVE-MEMBERED HETEROCYCLIC ALKANOIC ACID DERIVATIVE Takeda Chemical Industries, Ltd. (JP) 2004-03-03 EP disclosed
US-20030149006-A1 New vitamin D derivatives with cyclic substructures in the side chains, process and intermediate products for their production, and the use for the production of pharmaceutical agents STEINMEYER ANDREAS (US) 2003-08-07 US disclosed
US-6603031-B1 Active metabolites of vitamin D2 and vitamin D3 and their synthetic derivatives have a proliferation- inhibiting and differentiation-stimulating action on tumor cells and normal cells, SCHERING AKTIENGESELLSCHAFT (DE) 2003-08-05 US disclosed
EP-1228067-A1 5-MEMBERED N-HETEROCYCLIC COMPOUNDS WITH HYPOGYLCEMIC AND HYPOLIPIDEMIC ACTIVITY Takeda Chemical Industries, Ltd. (JP) 2002-08-07 EP disclosed
WO-2001038325-A1 5-MEMBERED N-HETEROCYCLIC COMPOUNDS WITH HYPOGLYCEMIC AND HYPOLIPIDEMIC ACTIVITY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030149006-A1 New vitamin D derivatives with cyclic substructures in the side chains, process and intermediate products for their production, and the use for the production of pharmaceutical agents CYP24A1, CYP2R1, VDR KMT2A 4855/4885MEN1 1811/4885TSHR 634/4885
US-20260125363-A1 PROCESSES FOR MAKING MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR CFTR, SLC26A4, SLC26A3 KMT2A 3014/4885MEN1 1794/4885TSHR 1602/4885
US-20040063775-A1 Five-membered heterocyclic alkanoic acid derivative SLC5A1, AHR, ALOX5 KMT2A 1788/4885MEN1 1753/4885TSHR 2362/4885
US-12624024-B2 EP2 antagonist compounds PTGER1, PTGER2, PTGER4 KMT2A 2217/4885MEN1 3479/4885TSHR 657/4885
US-20250034128-A1 BCL-XL INHIBITORS BCL2, BCL2L1, BCL2L10 KMT2A 3308/4885MEN1 4213/4885TSHR 3890/4885
US-12122788-B2 Process of making CFTR modulators CFTR, SLC26A4, TMEM109 KMT2A 4522/4885MEN1 2440/4885TSHR 2184/4885
US-12415798-B2 Processes for making modulators of cystic fibrosis transmembrane conductance regulator CFTR, SCNN1B, SCNN1G KMT2A 4813/4885MEN1 4316/4885TSHR 2866/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.