SCHEMBL21708879

SCHEMBL21708879

C#CCNCC(O)c1cc(O)c(O)c(C#C)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 7/20 0.43
ADRB1 P08588 6/20 0.43
ADRB3 P13945 5/20 0.43
ADRA2A P08913 2/20 0.37
ADRA2B P18089 2/20 0.37
ADRA2C P18825 2/20 0.37
MAPT P10636 5/20 0.36
TDP1 Q9NUW8 4/20 0.36
KDM4E B2RXH2 4/20 0.36
TSHR P16473 4/20 0.36
HIF1A Q16665 4/20 0.36
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
MTOR P42345 3/20 0.36
ADRA1A P35348 3/20 0.36
MAPK1 P28482 3/20 0.36
HSD17B10 Q99714 3/20 0.36
ALDH1A1 P00352 2/20 0.36
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21709164 0.81 KDM1A (0.35) ADRB2ADRB1ADRB3TSHRHIF1A
SCHEMBL21708881 0.80 MAOA (0.33)
SCHEMBL21708856 0.77 ADRB2 (0.63) ADRB2ADRB1ADRB3ADRA2AADRA2B
SCHEMBL21709152 0.76 ADRA1A (0.41) ADRB2ADRB1ADRB3ADRA2AADRA2B
SCHEMBL21708927 0.73 ADRB2 (0.34) ADRB2ADRB1ADRB3
SCHEMBL21709145 0.73 KDM1A (0.35) LMNA
SCHEMBL21708926 0.72 ALDH1A1 (0.31) ALDH1A1CYP1A2CYP2C19
SCHEMBL21708917 0.70 ACHE (0.39) ADRB2ADRA2BADRA2CMAPTKDM4E
SCHEMBL21709054 0.67 SLC22A3 (0.48) ADRB2ADRB1ADRB3ADRA2AADRA2B
SCHEMBL21709262 0.67 P2RX3 (0.38) ADRB2ADRB1ADRB3TSHRHIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020032080-A1 COMPOUND, SALT OF COMPOUND, NEUROMODULATION AGENT, METHOD FOR EVALUATING NEUROMODULATION AGENT, METHOD FOR PRODUCING COMPOUND, AND METHOD FOR PRODUCING SALT OF COMPOUND 学校法人慶應義塾 2020-02-13 WO disclosed