SCHEMBL22309474

SCHEMBL22309474

Cc1cc(-c2ccccc2)cc(C)c1N1C=CN(c2c(C)cc(-c3ccccc3)cc2C)C1C(C)C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.37
TSHR P16473 2/20 0.33
ALDH1A1 P00352 2/20 0.33
ALOX15 P16050 1/20 0.33
PDE1A P54750 1/20 0.33
PDE1B Q01064 1/20 0.33
PDE1C Q14123 1/20 0.33
PPARG P37231 1/20 0.33
PPARA Q07869 1/20 0.33
KDM4E B2RXH2 1/20 0.31
HTT P42858 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CHRM1 P11229 2/20 0.31
SLC22A2 O15244 1/20 0.31
SLC22A1 O15245 1/20 0.31
SLC22A3 O75751 1/20 0.31
SLC6A4 P31645 1/20 0.31
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
ESR1 P03372 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22825416 0.78 KDM4E (0.31) ALDH1A1KDM4E
SCHEMBL22309483 0.78 ALDH1A1 (0.34) TSHRALDH1A1ALOX15ESR1
SCHEMBL22309482 0.75 SCN4A (0.32)
SCHEMBL22309523 0.72 ALDH1A1 (0.34) ALDH1A1
SCHEMBL22309524 0.72 TSHR (0.31) TSHR
SCHEMBL22309471 0.67 LMNA (0.36) TSHRALDH1A1KDM4EHTTSMN1; SMN2
SCHEMBL22309527 0.67 KDM4E (0.42) TSHRALDH1A1PPARAKDM4E
SCHEMBL19431477 0.65 ALDH1A1 (0.50) BRD4TSHRALDH1A1PPARGPPARA
SCHEMBL22309517 0.63
SCHEMBL27898746 0.62 BRD4 (0.46) BRD4ALDH1A1PPARGPPARAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220009854-A1 A SERIES OF CATALYSTS FOR THE HYPERPOLARISATION OF SUBSTRATES UNIVERSITY OF YORK (GB) 2022-01-13 US disclosed
US-20210154333-A1 POLARISATION TRANSFER VIA A SECOND METAL COMPLEX UNIVERSITY OF YORK (GB) 2021-05-27 US disclosed
US-20200397923-A1 HYPERPOLARISATION IN AQUEOUS MEDIA VIA SABRE UNIVERSITY OF YORK (GB) 2020-12-24 US disclosed
US-20200246491-A1 HyperPolarising Substrates Through Relayed Transfer Via Systems Containing Exchangeable Protons UNIVERSITY OF YORK (GB) 2020-08-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220009854-A1 A SERIES OF CATALYSTS FOR THE HYPERPOLARISATION OF SUBSTRATES SPR, YAP1, KRAS BRD4 537/4885TSHR 1139/4885ALDH1A1 1891/4885
US-20200246491-A1 HyperPolarising Substrates Through Relayed Transfer Via Systems Containing Exchangeable Protons TSPO, RHOT2, KRAS BRD4 1764/4885TSHR 952/4885ALDH1A1 2261/4885
US-20210154333-A1 POLARISATION TRANSFER VIA A SECOND METAL COMPLEX TSPO, SPR, TIMM50 BRD4 2465/4885TSHR 2931/4885ALDH1A1 3970/4885
US-20200397923-A1 HYPERPOLARISATION IN AQUEOUS MEDIA VIA SABRE KRAS, FH, HYOU1 BRD4 1646/4885TSHR 1217/4885ALDH1A1 2889/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.