SCHEMBL224550

SCHEMBL224550

COc1cc(CCCO)cc(OC)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNKS2 Q9H2K2 1/20 0.56
PTGS2 P35354 1/20 0.55
AKR1B1 P15121 1/20 0.52
CYP19A1 P11511 1/20 0.50
ALDH1A1 P00352 1/20 0.48
CALM1 P0DP23 6/20 0.47
CNR1 P21554 2/20 0.45
CNR2 P34972 2/20 0.45
GABRA1 P14867 1/20 0.44
GABRG2 P18507 1/20 0.44
GABRB3 P28472 1/20 0.44
GABRA3 P34903 1/20 0.44
GABRA2 P47869 1/20 0.44
GABRB2 P47870 1/20 0.44
CYP4A11 Q02928 1/20 0.43
DAO P14920 1/20 0.42
IGF1R P08069 1/20 0.42
ALOX15 P16050 1/20 0.42
PTGES O14684 1/20 0.41
ALOX5 P09917 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23266717 0.94 PTGS2 (0.58) TNKS2PTGS2AKR1B1CYP19A1ALDH1A1
SCHEMBL5275704 0.92 PTGS2 (0.56) TNKS2PTGS2AKR1B1CYP19A1ALDH1A1
SCHEMBL1050377 0.92 PTGS2 (0.56) TNKS2PTGS2AKR1B1CYP19A1ALDH1A1
SCHEMBL22598538 0.87 CYP19A1 (0.51) TNKS2PTGS2AKR1B1CYP19A1ALDH1A1
SCHEMBL919408 0.86 AKR1B1 (0.55) TNKS2PTGS2AKR1B1CYP19A1ALDH1A1
SCHEMBL6568817 0.84 PTGS2 (0.49) TNKS2PTGS2AKR1B1CYP19A1CALM1
SCHEMBL920546 0.83 AKR1B1 (0.52) PTGS2AKR1B1CYP19A1ALDH1A1CALM1
SCHEMBL10296730 0.81 PTGS2 (0.50) TNKS2PTGS2AKR1B1CYP19A1CALM1
SCHEMBL9491787 0.81 CYP19A1 (0.68) PTGS2AKR1B1CYP19A1ALDH1A1CALM1
SCHEMBL81474 0.80 CHRM2 (0.63)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 47 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115385782-A Mechanochemical synthesis method of benzoyl compound 兰州大学 2022-11-25 CN claimed
CN-115385782-A Mechanochemical synthesis method of benzoyl compound 兰州大学 2022-11-25 CN disclosed
WO-2022133544-A1 CBD CANNABINOIDS AND CBD CANNABINOID ANALOGUES Botanix Pharmaceuticals Limited (AU) 2022-06-30 WO disclosed
CN-110720456-B Application of 3, 5-dimethoxytoluene 西南林业大学 2021-11-16 CN disclosed
US-9321045-B2 Catalyst and process for synthesising the same THE UNIVERSITY OF WARWICK (GB) 2016-04-26 US disclosed
US-9321045-B2 Catalyst and process for synthesising the same THE UNIVERSITY OF WARWICK (GB) 2016-04-26 US disclosed
US-20150290634-A1 Catalyst and Process for Synthesising the Same THE UNIVERSITY OF WARWICK (GB) 2015-10-15 US disclosed
US-20150290634-A1 Catalyst and Process for Synthesising the Same THE UNIVERSITY OF WARWICK (GB) 2015-10-15 US disclosed
EP-2914609-A1 CATALYST AND PROCESS FOR SYNTHESISING THE SAME THE UNIVERSITY OF WARWICK (GB) 2015-09-09 EP disclosed
EP-1577288-B1 Selective estrogen receptor modulators EISAI R&D MAN CO LTD (JP) 2014-07-23 EP disclosed
WO-2008079382-A1 SPHINGOSINE-1 -PHOSPHATE RECEPTOR AGONIST AND ANTAGONIST COMPOUNDS ABBOTT LABORATORIES (US) 2008-07-03 WO disclosed
WO-2008079382-A1 SPHINGOSINE-1 -PHOSPHATE RECEPTOR AGONIST AND ANTAGONIST COMPOUNDS ABBOTT LABORATORIES (US) 2008-07-03 WO disclosed
CN-101081853-A 4- (hydroxymethyl) -2, 6-dimethoxyphenylboronic acid compound EISAI CO LTD (JP) 2007-12-05 CN disclosed
CN-101081850-A 7-phenylpyrazolopyridine compounds EISAI CO LTD (JP) 2007-12-05 CN disclosed
CN-100338063-C 7-phenylpyrazolopyridine compounds EISAI CO LTD (JP) 2007-09-19 CN disclosed
US-20060116364-A1 Such as (R)-6-{2-{ethyl[4-(2-ethylaminoethyl)benzyl]amino }-4-methoxyphenyl }-5,6,7,8-tetrahydronaphthalen-2-ol; osteoporosis; breast cancer EISAI CO., LTD. (JP) 2006-06-01 US disclosed
WO-2006013399-A1 PHARMACEUTICAL INTERMEDIATES AND A PROCESS FOR THE PREPARATION THEREOF EGIS Gyógyszergyár Rt. (HU) 2006-02-09 WO disclosed
CN-1705665-A 7-phenylpyrazolopyridine compounds EISAI CO LTD (JP) 2005-12-07 CN disclosed
EP-1577288-A1 SELECTIVE ESTROGEN RECEPTOR MODULATORS Eisai Co., Ltd. (JP) 2005-09-21 EP disclosed
WO-1998008837-A1 PHENYLBUTANOL DERIVATIVES, METHODS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS THEREOF FARMACON, INC. (US) 1998-03-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150290634-A1 Catalyst and Process for Synthesising the Same CBR3, SPR, RNF5 TNKS2 161/4885PTGS2 1318/4885AKR1B1 604/4885
US-20060116364-A1 Such as (R)-6-{2-{ethyl[4-(2-ethylaminoethyl)benzyl]amino }-4-methoxyphenyl }-5,6,7,8-tetrahydronaphthalen-2-ol; osteoporosis; breast cancer BRCA1, BCR, RCC1 TNKS2 2475/4885PTGS2 3624/4885AKR1B1 369/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.