SCHEMBL22458325

SCHEMBL22458325

CC(=O)On1cnc2c(Cl)ncnc21

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 9/20 0.45
FGFR4 P22455 9/20 0.45
P2RX7 Q99572 2/20 0.44
FDPS P14324 1/20 0.43
HDAC6 Q9UBN7 2/20 0.41
DGAT1 O75907 1/20 0.34
GSK3B P49841 1/20 0.33
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
TP53 P04637 1/20 0.32
MAPT P10636 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
TYMP P19971 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14125909 0.81 ADORA2A (0.51) GSK3BALDH1A1TDP1
SCHEMBL28406876 0.80 ADORA2A (0.50) GSK3BALDH1A1TDP1
SCHEMBL11168017 0.78 FDPS (0.40) FGFR1FGFR4P2RX7FDPSHDAC6
SCHEMBL28003435 0.78 FDPS (0.43) FGFR1FGFR4P2RX7FDPSHDAC6
SCHEMBL10974937 0.75 P2RX7 (0.40) FGFR1FGFR4P2RX7FDPSHDAC6
SCHEMBL7594629 0.73 ACHE (0.41) FGFR1FGFR4HDAC6ALDH1A1LMNA
SCHEMBL28020916 0.72 P2RX7 (0.64) FGFR1FGFR4P2RX7FDPSHDAC6
SCHEMBL24021919 0.71 HPRT1 (0.47)
SCHEMBL7448126 0.70 MEN1 (0.53) FGFR1FGFR4P2RX7FDPSHDAC6
SCHEMBL7626872 0.70 FDPS (0.41) FDPSHDAC6ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11339188-B2 Compounds for the treatment of cancer EISAI R&D MANAGEMENT CO., LTD. (JP) 2022-05-24 US disclosed
US-20200299321-A1 COMPOUNDS FOR THE TREATMENT OF CANCER EISAI R&D MANAGEMENT CO., LTD. (JP) 2020-09-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200299321-A1 COMPOUNDS FOR THE TREATMENT OF CANCER TP53, MYC, CDC73 FGFR1 1838/4885FGFR4 1342/4885P2RX7 4661/4885
US-11339188-B2 Compounds for the treatment of cancer TP53, MYC, CDC73 FGFR1 1838/4885FGFR4 1342/4885P2RX7 4661/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.