SCHEMBL22650573

SCHEMBL22650573

CC(C)(C)OC(=O)N(CCF)C1CCN(c2ccc(N)nc2)C(=O)C1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LIPE Q05469 1/20 0.35
DPP4 P27487 2/20 0.33
ALOX5AP P20292 2/20 0.33
FEN1 P39748 2/20 0.33
ROCK2 O75116 1/20 0.33
GPR119 Q8TDV5 9/20 0.33
SCN9A Q15858 1/20 0.32
SCN10A Q9Y5Y9 1/20 0.32
HSD11B1 P28845 1/20 0.32
NR1H4 Q96RI1 1/20 0.32
GCK P35557 1/20 0.32
GCKR Q14397 1/20 0.32
MCHR1 Q99705 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650571 0.89 CCR5 (0.39) LIPEROCK2GPR119SCN9ASCN10A
SCHEMBL22650570 0.87 LIPE (0.37) LIPEROCK2GPR119HSD11B1
SCHEMBL29491165 0.84 SPR (0.38) ROCK2GPR119HSD11B1
SCHEMBL22650412 0.84 SPR (0.38) ROCK2GPR119HSD11B1
SCHEMBL22650566 0.81 DPP4 (0.33) DPP4ALOX5APFEN1GCKGCKR
SCHEMBL22650368 0.74 ALOX5AP (0.37) ALOX5APFEN1GCKR
SCHEMBL29462389 0.74 ALOX5AP (0.37) ALOX5APFEN1GCKR
SCHEMBL22650562 0.74 PIK3CA (0.35)
SCHEMBL22650910 0.73 DRD3 (0.35) ROCK2
SCHEMBL22650572 0.73 CCR5 (0.38) LIPEDPP4GPR119MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed