SCHEMBL2273187

SCHEMBL2273187

O=C(Nc1cc(-c2ccccc2)ccc1C(=O)O)C1=COC(Cc2ccccc2)O1

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ACLY P53396 16/20 0.49
DHODH Q02127 1/20 0.41
HDAC1 Q13547 1/20 0.41
MCL1 Q07820 1/20 0.41
SUCNR1 Q9BXA5 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2277761 0.95 ACLY (0.44) ACLYDHODHHDAC1MCL1SUCNR1
SCHEMBL2274220 0.92 ACLY (0.49) ACLYSUCNR1
SCHEMBL2272547 0.92 ACLY (0.40) ACLYDHODHMCL1
SCHEMBL2278113 0.87 NPC1 (0.39) ACLYMCL1
SCHEMBL2275462 0.85 HDAC2 (0.48) ACLY
SCHEMBL2276665 0.85 TTR (0.41) ACLY
SCHEMBL2267869 0.84 CYP2C9 (0.45) MCL1
SCHEMBL2274797 0.82 MEN1 (0.46) ACLYDHODHHDAC1MCL1SUCNR1
SCHEMBL2272855 0.78 HDAC2 (0.43) ACLYDHODHHDAC1
SCHEMBL7128829 0.78 PYGL (0.55)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7999132-B2 Anthranilic acid derivative or salt thereof TOYAMA CHEMICAL CO., LTD. (JP) 2011-08-16 US disclosed
US-20090240052-A1 NOVEL ANTHRANILIC ACID DERIVATIVE OR SALT THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 2009-09-24 US disclosed
EP-1820795-A1 NOVEL ANTHRANILIC ACID DERIVATIVE OR SALT THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 2007-08-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090240052-A1 NOVEL ANTHRANILIC ACID DERIVATIVE OR SALT THEREOF MMP13, MMP26, MMP11 ACLY 653/4885DHODH 1469/4885HDAC1 71/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.