SCHEMBL2320187

SCHEMBL2320187

[c]1nc2ccccc2cc1-c1ccccn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 10/20 0.47
TDP1 Q9NUW8 3/20 0.47
LMNA P02545 6/20 0.43
CCR1 P32246 3/20 0.43
CCR5 P51681 3/20 0.43
CCR8 P51685 3/20 0.43
METAP1 P53582 3/20 0.43
CYP1A2 P05177 2/20 0.43
POLB P06746 2/20 0.43
BLM P54132 1/20 0.43
HIF1A Q16665 1/20 0.43
DOHH Q9BU89 1/20 0.43
P4HTM Q9NXG6 1/20 0.43
SMN1; SMN2 Q16637 8/20 0.42
TP53 P04637 6/20 0.42
ALOX15 P16050 4/20 0.42
L3MBTL1 Q9Y468 4/20 0.42
HTT P42858 2/20 0.42
ALPL P05186 2/20 0.42
HSP90AA1 P07900 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2719862 0.83 CBFB (0.49) KDM4ETDP1LMNACCR1CCR5
SCHEMBL1385432 0.82 ALDH1A1 (0.42) KDM4ETDP1METAP1CYP1A2POLB
SCHEMBL11160532 0.82 PDGFRB (0.38) CYP1A2NPC1RAB9AALDH1A1HPGD
SCHEMBL724724 0.82 METAP2 (0.44) CYP1A2SMN1; SMN2HTTNPC1RAB9A
SCHEMBL15229223 0.81 ALDH1A1 (0.43) KDM4EPOLBSMN1; SMN2TP53HTT
SCHEMBL1542711 0.80 DHODH (0.39) KDM4EPOLBNPC1RAB9AALDH1A1
SCHEMBL2659111 0.78 NPC1 (0.44) KDM4ECYP1A2SMN1; SMN2ALOX15HSP90AA1
SCHEMBL523809 0.77 RAB9A (0.44) KDM4ETDP1LMNACYP1A2BLM
SCHEMBL5619122 0.76 CYP1A2 (0.35) KDM4ECYP1A2ALDH1A1HPGDMAPT
SCHEMBL938744 0.74 ALDH1A1 (0.40) KDM4ETDP1CCR1CCR8CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 69 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170162800-A1 Electrically Doped Organic Semiconducting Material and Organic Light Emitting Device Comprising It NOVALED GMBH (DE) 2017-06-08 US claimed
CN-102918037-A Carbazole compound having substituent containing electron-accepting nitrogen-containing heteroaryl group, and organic electroluminescent element JNC CORP 2013-02-06 CN claimed
US-20050288337-A1 Novel compounds MITSUBISHI TANABE PHARMA CORPORATION (JP) 2005-12-29 US claimed
EP-1539696-A2 PROCESS FOR PREPARING QUINOLIN ANTIBIOTIC INTERMEDIATES TANABE SEIYAKU CO., LTD. (JP) 2005-06-15 EP claimed
US-20050004202-A1 Indazolyl-substituted pyrroline compounds as kinase inhibitors ZHANG HAN-CHENG (US) 2005-01-06 US claimed
WO-2004014859-A2 PROCESS FOR PREPARING QUINOLIN ANTIBIOTIC INTERMEDIATES TANABE SEIYAKU CO., LTD. (JP) 2004-02-19 WO claimed
US-6225334-B1 AS PESTICIDES BAYER AKTIENGESELLSCHAFT (DE) 2001-05-01 US claimed
US-5648448-A Method of preparation of polyquinolines HITACHI CHEMICAL COMPANY, LTD. (JP) 1997-07-15 US claimed
US-5391730-A An immunsuppressantes, antiinflammatory agents, fungicides, antitumor agents AMERICAN HOME PRODUCTS CORPORATION (US) 1995-02-21 US claimed
US-20240201591-A1 PHOTORESIST UNDERLAYER COMPOSITION DUPONT SPECIALTY MATERIALS KOREA LTD (KR) 2024-06-20 US disclosed
US-11937504-B2 Organic electroluminescent device UDC IRELAND LIMITED (IE) 2024-03-19 US disclosed
CN-117384193-A Boron-containing organic compound and organic electroluminescent device prepared from same 江苏三月科技股份有限公司 2024-01-12 CN disclosed
US-11411185-B2 Organic electroluminescent device UDC IRELAND LIMITED (IE) 2022-08-09 US disclosed
EP-3305871-B1 USE OF DEUTERATED CARBAZOLE IN ORGANIC ELECTROLUMINESCENT DEVICES UDC IRELAND LTD (IE) 2020-02-26 EP disclosed
US-20040039035-A1 Modulation of CCR4 function TULARIK INC. 2004-02-26 US disclosed
US-20020173524-A1 Modulation of CCR4 function TULARIK INC. (US) 2002-11-21 US disclosed
WO-2002030358-A2 MODULATION OF CCR4 FUNCTION TULARIK INC. (US) 2002-04-18 WO disclosed
US-5766779-A Electron transporting materials for organic electroluminescent devices EASTMAN KODAK COMPANY (US) 1998-06-16 US disclosed
WO-1994014797-A1 QUINOLINE COMPOUNDS AND THE TREATMENT OF LEUCOTRIENE RELATED DISEASES THEREWITH SMITHKLINE BEECHAM CORPORATION (US) 1994-07-07 WO disclosed
US-4851547-A MALEIC ANHYDRIDE, AMINE TO MALEINAMIC ACID; CATALYST OF STRONG ACID AND/OR ITS AMINE SALT NIPPON SHOKUBAI KAGAKU KOGYO CO., LTD. (JP) 1989-07-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050288337-A1 Novel compounds ITGB4, ITGA4, ITGB5 KDM4E 810/4885TDP1 3809/4885LMNA 2016/4885
US-20020173524-A1 Modulation of CCR4 function CCR4, CCR1, CCR3 KDM4E 3826/4885TDP1 4118/4885LMNA 4708/4885
US-20170162800-A1 Electrically Doped Organic Semiconducting Material and Organic Light Emitting Device Comprising It C1S, C5, HCN2 KDM4E 3935/4885TDP1 4477/4885LMNA 399/4885
US-20050004202-A1 Indazolyl-substituted pyrroline compounds as kinase inhibitors MAP2K2, MAP3K20, MAP2K3 KDM4E 1504/4885TDP1 687/4885LMNA 3426/4885
US-20040039035-A1 Modulation of CCR4 function CCR4, CCR1, CCR3 KDM4E 3826/4885TDP1 4118/4885LMNA 4708/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.