SCHEMBL2344700

SCHEMBL2344700

C=Cc1ccccc1C[PH](CCCC)(CCCC)CCCC

nearest known ligand 0.34

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.33
THRA P10827 1/20 0.33
THRB P10828 1/20 0.33
LIPG Q9Y5X9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phosphine SCHEMBL8143769 0.98 ALDH1A1 (0.32) ALDH1A1THRATHRBLIPG
SCHEMBL4840342 0.94 THRA (0.37) ALDH1A1THRATHRBLIPG
SCHEMBL2346267 0.94 THRA (0.37) ALDH1A1THRATHRBLIPG
SCHEMBL4835886 0.94 THRA (0.37) ALDH1A1THRATHRBLIPG
SCHEMBL20567945 0.83 ALDH1A1 (0.33) ALDH1A1
SCHEMBL8019676 0.82 ALDH1A1 (0.38) ALDH1A1
SCHEMBL28869 0.77 CYP3A4 (0.44) ALDH1A1THRATHRBLIPG
SCHEMBL29480441 0.77 CYP3A4 (0.44) ALDH1A1THRATHRBLIPG
SCHEMBL8669532 0.77 LIPG (0.43) ALDH1A1THRATHRBLIPG
SCHEMBL5501020 0.75 ALDH1A1 (0.38) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 53 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2403843-B1 CHEMILUMINESCENT COMPOSITIONS, METHODS, ASSAYS AND KITS FOR OXIDATIVE ENZYMES LIFE TECHNOLOGIES CORP (US) 2018-11-07 EP claimed
EP-2165197-B1 REAGENTS, KITS AND METHODS FOR DETECTING BIOLOGICAL MOLECULES BY ENERGY TRANSFER FROM AN ACTIVATED CHEMILUMINESCENT SUBSTRATE TO AN ENERGY ACCEPTOR DYE LIFE TECHNOLOGIES CORP (US) 2011-08-31 EP claimed
EP-0874913-B1 MULTIPLE REPORTER GENE ASSAY APPLERA CORP (US) 2008-06-25 EP claimed
EP-1883635-A2 LIGHT-EMITTING BIOMARKER Quidd (FR) 2008-02-06 EP claimed
WO-2006129036-A2 LIGHT-EMITTING BIOMARKER QUIDD (FR) 2006-12-07 WO claimed
US-6695076-B2 Method of coring crustal core sample, and antimicrobial polymeric gel and gel material used in the method JAPAN MARINE SCIENCE & TECHNOLOGY CENTER (JP) 2004-02-24 US claimed
US-6635437-B2 Useful in methods for producing light and in assays for phosphatase enzymes and enzyme inhibitors and in assays employing enzyme-labeled specific binding pairs LUMIGEN, INC. 2003-10-21 US claimed
EP-0819119-B1 COMPOUNDS, COMPOSITIONS AND METHODS FOR GENERATING CHEMILUMINESCENCE WITH PHOSPHATASE ENZYMES LUMIGEN INC (US) 2003-04-02 EP claimed
US-20030023089-A1 Compounds, compositions and methods for generating chemiluminescence with phosphatase enzymes AKHAVAN-TAFTI HASHEM (US) 2003-01-30 US claimed
US-6296787-B1 ACRIDINE AND PHENANTHRIDINE ALKENYL PHOSPHATE DERIVATIVES LUMIGEN, INC. 2001-10-02 US claimed
US-6270695-B1 HETEROCYCLIC COMPOUNDS WITH EXOCYCLIC DOUBLE BOND HAVING PHOSPHATE GROUP ATTACHED TO DISTAL CARBON; DETECTION SENSITIVITY LUMIGEN, INC. 2001-08-07 US claimed
US-6218137-B1 SENSITIVE QUANTITATIVE ANALYSIS USING COMPOUND HAVING A HETEROCYCLIC RING SYSTEM BEARING AN EXOCYCLIC CARBON-CARBON DOUBLE BOND WHICH IS SUBSTITUTED AT DISTAL CARBON WITH PHOSPHATE GROUP AND OXYGEN OR SULFUR GROUP LUMIGEN, INC. 2001-04-17 US claimed
US-6139782-A A CHEMILUMINESCENT CONTAINING A HETEROCYCLIC RING GROUP AND AN ENOL PHOSPHATE GROUP WHICH REACT WITH OXYGEN UPON REMOVAL OF PHOSPHATE GROUP WITH A PHOSPHATASE ENZYME TO PRODUCE AN ENOLATE WHICH REACTS WITH TO PRODUCE CHEMILUMINOESCENCE LUMIGEN, INC. (US) 2000-10-31 US claimed
US-6090571-A REACTING PHOSPHATASE WITH NITROGEN-CONTAINING HETEROCYCLIC RING SYSTEM HAVING AN ENOL PHOSPHATE GROUP, DETECTING THE CHEMILUMINESCENCE, AND RELATING TO AMOUNT OF ANALYTE LUMIGEN, INC. (US) 2000-07-18 US claimed
US-6045727-A NITROGEN CONTAINING HETEROCYCLIC RING SYSTEM BEARING AN EXOCYCLIC CARBON-CARBON DOUBLE BOND. THE DOUBLE BOND IS FURTHER SUBSTITUTED AT THE DISTAL CARBON WITH A PHOSPHATE GROUP AND AN OXYGEN OR SULFUR ATOM-CONTAINING GROUP. LUMIGEN, INC. (US) 2000-04-04 US claimed
EP-0561033-B1 Polymeric phoshonium salts providing enhanced chemiluminescence from 1,2-dioxetanes, and their use. LUMIGEN INC (US) 2000-03-15 EP claimed
EP-0819119-A4 COMPOUNDS, COMPOSITIONS AND METHODS FOR GENERATING CHEMILUMINESCENCE WITH PHOSPHATASE ENZYMES LUMIGEN INC (US) 1999-04-14 EP claimed
EP-0819119-A1 COMPOUNDS, COMPOSITIONS AND METHODS FOR GENERATING CHEMILUMINESCENCE WITH PHOSPHATASE ENZYMES LUMIGEN, INC. (US) 1998-01-21 EP claimed
WO-1997026245-A1 COMPOUNDS, COMPOSITIONS AND METHODS FOR GENERATING CHEMILUMINESCENCE WITH PHOSPHATASE ENZYMES LUMIGEN, INC. (US) 1997-07-24 WO claimed
CN-113292921-A Composite insulator coating, preparation method and spraying process 广东电网有限责任公司 2021-08-24 CN disclosed
CN-111410724-B Super absorbent resin for vertical greening and preparation method thereof 东华大学 2021-01-05 CN disclosed
US-9356318-B2 Gel polymer electrolyte composition KURARAY CO., LTD. (JP) 2016-05-31 US disclosed
EP-2524932-B1 GEL POLYMER ELECTROLYTE COMPOSITION KURARAY CO (JP) 2015-11-25 EP disclosed
US-20120321963-A1 GEL POLYMER ELECTROLYTE COMPOSITION KURARAY CO., LTD. (JP) 2012-12-20 US disclosed
EP-2524932-A1 GEL POLYMER ELECTROLYTE COMPOSITION Kuraray Co., Ltd. (JP) 2012-11-21 EP disclosed
WO-2008145830-A2 NOVEL PRO-FLUORESCENT COMPOUNDS QUIDD (FR) 2008-12-04 WO disclosed
US-7343984-B2 Core sample collector equipped with sterilizing agent-applying mechanism and method of taking core sample INDEPENDENT ADMINISTRATIVE INSTITUTION, JAPAN AGENCY FOR MARINE-EARTH SCIENCE AND TECHNOLOGY (JP) 2008-03-18 US disclosed
EP-1789578-A4 CLEAVABLE SOLID PHASES FOR ISOLATING NUCLEIC ACIDS NEXGEN DIAGNOSTICS LLC (US) 2008-02-27 EP disclosed
EP-1883635-A2 LIGHT-EMITTING BIOMARKER Quidd (FR) 2008-02-06 EP disclosed
US-7308951-B2 Method of coring a crustal core sample and flow-able coating material for coring a crustal core sample INDEPENDENT ADMINISTRATIVE INSTITUTION, JAPAN AGENCY FOR MARINE-EARTH SCIENCE AND TECHNOLOGY (JP) 2007-12-18 US disclosed
EP-1781808-A4 METHODS OF USING CLEAVABLE SOLID PHASES FOR ISOLATING NUCLEIC ACIDS LUMIGEN INC (US) 2007-08-29 EP disclosed
EP-1789578-A2 CLEAVABLE SOLID PHASES FOR ISOLATING NUCLEIC ACIDS LUMIGEN, INC. (US) 2007-05-30 EP disclosed
EP-1781808-A1 METHODS OF USING CLEAVABLE SOLID PHASES FOR ISOLATING NUCLEIC ACIDS LUMIGEN, INC. (US) 2007-05-09 EP disclosed
WO-2006129036-A2 LIGHT-EMITTING BIOMARKER QUIDD (FR) 2006-12-07 WO disclosed
WO-2006019387-A1 METHODS OF USING CLEAVABLE SOLID PHASES FOR ISOLATING NUCLEIC ACIDS LUMIGEN, INC. (US) 2006-02-23 WO disclosed
WO-2006019388-A2 CLEAVABLE SOLID PHASES FOR ISOLATING NUCLEIC ACIDS LUMIGEN, INC. (US) 2006-02-23 WO disclosed
US-20050183886-A1 Method of coring a crustal core sample and flow-able coating material for coring a crustal core sample INDEPENDENT ADMINISTRATIVE INSTITUTION JAPAN AGENCY FOR MARINE-EARTH SCIENCE AND TECHNOLOGY (JP) 2005-08-25 US disclosed
US-20050106751-A1 Piston corer comprising bactericidal agents for use in isolating subsurface microorganisms JAPAN MARINE SCIENCE & TECHNOLOGY CENTER (JP) 2005-05-19 US disclosed
US-6695076-B2 Method of coring crustal core sample, and antimicrobial polymeric gel and gel material used in the method JAPAN MARINE SCIENCE & TECHNOLOGY CENTER (JP) 2004-02-24 US disclosed
EP-0988152-B1 COATING COMPOSITION AND PRINTING MEDIUM HEWLETT PACKARD CO (US) 2002-10-30 EP disclosed
US-20020139583-A1 Method of coring crustal core sample, and antimicrobial polymeric gel and gel material used in the method JAPAN MARINE SCIENCE & TECHNOLOGY CENTER (JP) 2002-10-03 US disclosed
EP-0898557-A4 WATER SOLUBLE TRI-SUBSTITUTED 1,2-DIOXETANE COMPOUNDS HAVING INCREASED STORAGE STABILITY, SYNTHETIC PROCESSES AND INTERMEDIATES LUMIGEN INC (US) 2001-01-10 EP disclosed
EP-0561033-B1 Polymeric phoshonium salts providing enhanced chemiluminescence from 1,2-dioxetanes, and their use. LUMIGEN INC (US) 2000-03-15 EP disclosed
US-5880196-A VOLATILE AQUEOUS LIQUID MEDIUM CONTAINING ONIUM-FREE AND ONIUM-CONTAINING POLYMERIC BINDERS, FINELY DIVIDED PSEUDOBOEHMITE PARTICLES; NONBLEEDING PPG INDUSTRIES, INC. (US) 1999-03-09 US disclosed
EP-0898557-A1 WATER SOLUBLE TRI-SUBSTITUTED 1,2-DIOXETANE COMPOUNDS HAVING INCREASED STORAGE STABILITY, SYNTHETIC PROCESSES AND INTERMEDIATES LUMIGEN, INC. (US) 1999-03-03 EP disclosed
WO-1998019989-A1 WATER SOLUBLE TRI-SUBSTITUTED 1,2-DIOXETANE COMPOUNDS HAVING INCREASED STORAGE STABILITY, SYNTHETIC PROCESSES AND INTERMEDIATES LUMIGEN, INC. (US) 1998-05-14 WO disclosed
US-5601977-A GENERATING CHEMILUMINESCENCE FROM OXIDATION OF CYCLIC DIACYLHYDRAZIDE DERIVATIVE BY ACTION OF PEROXIDASE ENZYME, A PEROXIDE OXIDIZER AND ENHANCER LUMIGEN, INC. (US) 1997-02-11 US disclosed
US-5582775-A WATER SOLUBLE; PREPARED BY REACTING AT LEAST TWO DIFFERENT PHOSPHINES WITH POLYVINYL POLYMER LUMIGEN, INC. (US) 1996-12-10 US disclosed
US-5474725-A Reacting polyvinylbenzyl chloride with a trialkylphosphine to form salt LUMIGEN, INC. (US) 1995-12-12 US disclosed
US-5439617-A Composition containing stable 1,2-dioxetane, polyvinyl phosphonium salt polymer LUMIGEN, INC. (US) 1995-08-08 US disclosed
US-5431845-A Polymeric phosphonium salts providing enhanced chemiluminescence from 1,2-dioxetanes LUMIGEN, INC. (US) 1995-07-11 US disclosed
US-5393469-A Triggering dioxetane with activating agents consisting of acids, bases, salts, enzymes, inorganic or organic catalysts and electron donors; used for immunoassay and nucleic acid assay LUMIGEN, INC. (US) 1995-02-28 US disclosed
EP-0561033-A1 Polymeric phoshonium salts providng enhanced chemiluminescence from 1,2-dioxetanes LUMIGEN, INC. (US) 1993-09-22 EP disclosed
EP-0561033-A1 Polymeric phoshonium salts providng enhanced chemiluminescence from 1,2-dioxetanes LUMIGEN, INC. (US) 1993-09-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030023089-A1 Compounds, compositions and methods for generating chemiluminescence with phosphatase enzymes PPP6C, PPP4C, PPP2CA ALDH1A1 2206/4885THRA 4748/4885THRB 4236/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.