Water

Water

SCHEMBL2359149

O.O=C(O)c1ccc2ccccc2c1C(=O)O

nearest known ligand 0.66

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Water. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 known ✓ O00255 2/20 0.59
FDPS known ✓ P14324 1/20 0.44
WDR5 P61964 1/20 0.66
LDHA P00338 1/20 0.63
ALDH1A1 P00352 6/20 0.59
HPGD P15428 5/20 0.59
KDM4E B2RXH2 3/20 0.59
GLA P06280 2/20 0.59
KMT2A Q03164 2/20 0.59
HSD17B10 Q99714 2/20 0.59
NR4A1 P22736 1/20 0.59
NR4A2 P43354 1/20 0.59
NR4A3 Q92570 1/20 0.59
CYP1A2 P05177 1/20 0.59
CYP2C19 P33261 1/20 0.59
CDC25B P30305 2/20 0.56
METAP2 P50579 1/20 0.49
METAP1 P53582 1/20 0.49
LMNA P02545 1/20 0.47
CSNK2A2 P19784 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29376013 0.98 WDR5 (0.68) WDR5LDHAALDH1A1HPGDKDM4E
SCHEMBL27804512 0.98 WDR5 (0.68) WDR5LDHAALDH1A1HPGDKDM4E
SCHEMBL33850 0.98 WDR5 (0.68) WDR5LDHAALDH1A1HPGDKDM4E
Benzene SCHEMBL27549874 0.98 WDR5 (0.68) WDR5LDHAALDH1A1HPGDKDM4E
Naphthalene SCHEMBL1831655 0.96 WDR5 (0.66) WDR5LDHAALDH1A1HPGDKDM4E
Ammonia Solution, Strong SCHEMBL8803959 0.96 WDR5 (0.66) WDR5LDHAALDH1A1HPGDKDM4E
SCHEMBL964273 0.96 WDR5 (0.66) WDR5LDHAALDH1A1HPGDKDM4E
Hydrochloric Acid SCHEMBL608188 0.96 LDHA (0.69) WDR5LDHAALDH1A1HPGDKDM4E
SCHEMBL19307798 0.96 WDR5 (0.66) WDR5LDHAALDH1A1HPGDKDM4E
SCHEMBL4577224 0.96 WDR5 (0.66) WDR5LDHAALDH1A1HPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230295398-A1 THERMALLY CONDUCTIVE SHEET AND DEVICE PROVIDED WITH THERMALLY CONDUCTIVE SHEET RESONAC CORPORATION (JP) 2023-09-21 US disclosed
WO-2020234937-A1 METHOD FOR PRODUCING HEAT STORAGE SHEET 昭和電工マテリアルズ株式会社 (JP) 2020-11-26 WO disclosed
US-10807830-B2 Winding core and roll HITACHI CHEMICAL COMPANY, LTD. (JP) 2020-10-20 US disclosed
US-10144383-B2 Steering wheel with video screen and airbag STEERING SOLUTIONS IP HOLDING CORPORATION (US) 2018-12-04 US disclosed
CN-107878386-A Steering wheel with display screen and air bag 操纵技术IP控股公司 2018-04-06 CN disclosed
US-20180086297-A1 STEERING WHEEL WITH VIDEO SCREEN AND AIRBAG STEERING SOLUTIONS IP HOLDING CORPORATION 2018-03-29 US disclosed
US-20150129706-A1 WINDING CORE AND ROLL RESONAC CORPORATION (JP) 2015-05-14 US disclosed
US-20120114934-A1 BONDING SHEET HITACHI CHEMICAL COMPANY, LTD. (JP) 2012-05-10 US disclosed
US-20110193244-A1 ADHESIVE FILM AND PROCESS FOR PREPARING THE SAME AS WELL AS ADHESIVE SHEET AND SEMICONDUCTOR DEVICE MASUKO TAKASHI 2011-08-11 US disclosed
US-7696441-B2 Flexible wired circuit board NITTO DENKO CORPORATION (JP) 2010-04-13 US disclosed
US-20070141864-A1 Flexible wired circuit board NITTO DENKO CORPORATION (JP) 2007-06-21 US disclosed
US-20070098995-A1 Adhesive film and process for preparing the same as well as adhesive sheet and semiconductor device HITACHI CHEMICAL CO., LTD. (JP) 2007-05-03 US disclosed