SCHEMBL23770731

SCHEMBL23770731

Cc1c(F)cccc1-c1nc(NSc2cccc(N3CCNCC3)n2)ccc1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 2/20 0.40
HTR3E A5X5Y0 1/20 0.40
HTR3B O95264 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HTR3D Q70Z44 1/20 0.40
HTR3C Q8WXA8 1/20 0.40
PTPN11 Q06124 1/20 0.36
CHEK1 O14757 3/20 0.33
BPTF Q12830 2/20 0.33
HTR1A P08908 2/20 0.33
HTR7 P34969 1/20 0.33
HTR2B P41595 1/20 0.33
HTR6 P50406 1/20 0.33
CDK7 P50613 2/20 0.33
PIM1 P11309 1/20 0.33
PIM3 Q86V86 1/20 0.33
PIM2 Q9P1W9 1/20 0.33
NPC1 O15118 1/20 0.33
KCNH2 Q12809 1/20 0.32
CACNA1C Q13936 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23770819 0.91 HTR3A (0.41) HTR3AHTR3EHTR3BALDH1A1HTR3D
SCHEMBL23770862 0.88 HTR3E (0.42) HTR3AHTR3EHTR3BALDH1A1HTR3D
SCHEMBL23770453 0.87 CYP1A2 (0.40) HTR3AHTR3EHTR3BALDH1A1HTR3D
SCHEMBL23770808 0.85 HTR3E (0.38) HTR3AHTR3EHTR3BALDH1A1HTR3D
SCHEMBL23770850 0.85 LRRK2 (0.33)
SCHEMBL23770669 0.84 HTR3A (0.40) HTR3AHTR3EHTR3BALDH1A1HTR3D
SCHEMBL23770884 0.84 RORC (0.36) PTPN11
SCHEMBL23770450 0.84 HTR3E (0.43) HTR3AHTR3EHTR3BALDH1A1HTR3D
SCHEMBL23770650 0.82 PTPN11 (0.32) PTPN11NPC1
SCHEMBL19925107 0.80 HTR3E (0.38) HTR3AHTR3EHTR3BALDH1A1HTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3504194-B1 N-(PYRIDIN-2-YL)PYRIDINE-SULFONAMIDE DERIVATIVES AND THEIR USE IN THE TREATMENT OF DISEASE NOVARTIS AG (CH) 2021-08-18 EP disclosed