SCHEMBL23770837

SCHEMBL23770837

Cc1cccc(C)c1-c1nc(NSc2cccc(N3CCC3)n2)ccc1Cl

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMO Q99835 1/20 0.34
KDM4E B2RXH2 2/20 0.33
GAA P10253 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
KMT2A Q03164 2/20 0.33
HTR3E A5X5Y0 4/20 0.33
HTR3B O95264 4/20 0.33
HTR3A P46098 4/20 0.33
HTR3D Q70Z44 4/20 0.33
HTR3C Q8WXA8 4/20 0.33
TDP1 Q9NUW8 1/20 0.32
CNR1 P21554 4/20 0.32
CNR2 P34972 1/20 0.32
MEN1 O00255 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
ALOX15 P16050 1/20 0.32
TSHR P16473 1/20 0.32
NFKB1 P19838 1/20 0.32
PDE10A Q9Y233 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23770450 0.91 HTR3E (0.43) SMOKDM4EHTR3EHTR3BHTR3A
SCHEMBL23770800 0.85 RORC (0.32) SMOKMT2ACNR1CNR2MEN1
SCHEMBL23770659 0.85 PTPN11 (0.36) SMOCNR1CNR2
SCHEMBL23770844 0.85 PTPN11 (0.33) SMOCNR1CNR2
SCHEMBL23770648 0.84 GPBAR1 (0.41) KDM4EKMT2AMEN1TSHRALDH1A1
SCHEMBL23770785 0.84 LMNA (0.43) SMOKDM4EL3MBTL1KMT2ATDP1
SCHEMBL19970116 0.84 DGAT1 (0.35) CNR1CNR2
SCHEMBL23770475 0.83 L3MBTL1 (0.39) KDM4EL3MBTL1KMT2ACNR1CNR2
SCHEMBL23770843 0.83 SMO (0.33) SMO
SCHEMBL23770874 0.83 SMO (0.31) SMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3504194-B1 N-(PYRIDIN-2-YL)PYRIDINE-SULFONAMIDE DERIVATIVES AND THEIR USE IN THE TREATMENT OF DISEASE NOVARTIS AG (CH) 2021-08-18 EP disclosed