SCHEMBL237859

SCHEMBL237859

Cn1c(=O)c2[nH]c(Cl)nc2n(C(=O)O)c1=O

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.60
ALDH1A1 P00352 4/20 0.43
CYP1A2 P05177 3/20 0.43
HSD17B10 Q99714 3/20 0.43
LMNA P02545 1/20 0.43
CHRM2 P08172 1/20 0.43
CHRM4 P08173 1/20 0.43
CHRM5 P08912 1/20 0.43
ADRA2A P08913 1/20 0.43
CYP2D6 P10635 1/20 0.43
CHRM1 P11229 1/20 0.43
ADRA2B P18089 1/20 0.43
CHRM3 P20309 1/20 0.43
SLC6A2 P23975 1/20 0.43
ADRA1D P25100 1/20 0.43
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
HRH1 P35367 1/20 0.43
HTR2B P41595 1/20 0.43
SLC6A3 Q01959 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrazine SCHEMBL9281750 0.97 SMN1; SMN2 (0.58) SMN1; SMN2ALDH1A1CYP1A2HSD17B10LMNA
8-Chlorotheophylline SCHEMBL411139 0.80 POLB (0.57) SMN1; SMN2ALDH1A1CYP1A2HSD17B10LMNA
8-Chlorotheophylline SCHEMBL5719335 0.79 POLB (0.55) SMN1; SMN2ALDH1A1CYP1A2HSD17B10LMNA
Diphenhydramine SCHEMBL4193326 0.78 SMN1; SMN2 (1.00) SMN1; SMN2ALDH1A1CYP1A2HSD17B10LMNA
Diphenylpyraline SCHEMBL1274388 0.77 SMN1; SMN2 (0.63) SMN1; SMN2ALDH1A1CYP1A2HSD17B10LMNA
SCHEMBL3181178 0.74 ADORA2A (0.54) CYP1A2ADORA2BADORA2AADORA1CYP2C19
SCHEMBL29430494 0.72 ADORA2B (0.49) ALDH1A1CYP1A2HSD17B10LMNACHRM2
SCHEMBL11239048 0.71 ATAD2 (0.66) CYP1A2LMNAADORA2BADORA2AADORA1
SCHEMBL3175131 0.71 PDE4A (0.57) CYP1A2ADORA2ACYP2C19
SCHEMBL18833875 0.71 HPGD (0.55) SMN1; SMN2ALDH1A1CYP1A2HSD17B10LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1178 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11459341-B1 Organic anion lithium ionic cocrystal compounds and compositions UNIVERSITY OF SOUTH FLORIDA (US) 2022-10-04 US claimed
US-20220226205-A1 Coated Particles and Their Uses KENVUE BRANDS LLC 2022-07-21 US claimed
EP-3527192-B9 AMINO ACID DERIVATIVES AND THEIR USES JOHNSON & JOHNSON CONSUMER INC (US) 2022-04-27 EP claimed
EP-2986618-B1 ORGANIC ANION LITHIUM IONIC COCRYSTAL COMPOUNDS AND COMPOSITIONS UNIV SOUTH FLORIDA (US) 2021-12-01 EP claimed
US-20210284604-A1 Amino Acid Derivatives and Their Uses KENVUE BRANDS LLC 2021-09-16 US claimed
EP-3527192-B1 AMINO ACID DERIVATIVES AND THEIR USES JOHNSON & JOHNSON CONSUMER INC (US) 2021-09-08 EP claimed
EP-3753562-A1 COMPOSITIONS COMPRISING THE TROMETHAMINE SALT OF L-AMPICILLIN. Alpha-1 Biologics LLC (US) 2020-12-23 EP claimed
US-10870665-B1 Organic anion lithium ionic cocrystal compounds and compositions UNIVERSITY OF SOUTH FLORIDA (US) 2020-12-22 US claimed
US-20200115331-A1 Amino Acid Derivatives and Their Uses KENVUE BRANDS LLC 2020-04-16 US claimed
EP-3634372-A1 COATED PARTICLES AND THEIR USES Johnson & Johnson Consumer Inc. (US) 2020-04-15 EP claimed
US-20060241295-A1 Preparation of pharmaceutical salts of piperazine compounds SCHERING CORPORATION 2006-10-26 US claimed
WO-2006074269-A2 PREPARATION OF PHARMACEUTICAL SALTS OF PIPERAZINE COMPOUNDS SCHERING CORPORATION (US) 2006-07-13 WO claimed
US-6936718-B2 Preparation of rotamer mixtures of pharmaceutical salts SCHERING CORPORATION (US) 2005-08-30 US claimed
US-20050171117-A1 Preparation of pharmaceutical salts GALA DINESH (US) 2005-08-04 US claimed
EP-1451174-A2 PROCESS FOR THE PREPARATION OF COMPOSITIONS HAVING AN INCREASED AMOUNT OF PHARMACEUTICALLY ACTIVE SALTS OF ROTAMERS SCHERING CORPORATION (US) 2004-09-01 EP claimed
EP-1448528-A2 PREPARATION OF PHARMACEUTICAL SALTS OF 4((Z)-(4-BROMOPHENYL)(ETHOXYIMINO)METHYL)-1'-((2,4-DIMETHYL-1-OXIDO-3-PYRIDINYL)CARBONYL)-4'-METHYL-1,4'BIPIPERIDINE AS CCR5-ANTAGONISTS FOR THE TREATMENT OF AIDS AND RELATED HIV INFECTIONS SCHERING CORPORATION (US) 2004-08-25 EP claimed
WO-2003066593-A2 PREPARATION OF PHARMACEUTICAL SALTS OF 4 ( (Z) - (4-BROMOPHENYL) (ETHOXYIMINO) METHYL )-1'-( (2,4-DIMETHYL-1-OXIDO-3-PYRIDINYL) CARBONYL) -4'-METHYL-1,4' BIPIPERIDINE AS CCR5-ANTAGONISTS FOR THE TREATMENT OF AIDS AND RELATED HIV INFECTIONS SCHERING CORPORATION (US) 2003-08-14 WO claimed
US-20030144510-A1 receptor which are useful for the treatment of AIDS and related HIV infections, including the compound of Formula I. CCR-5 receptors have also been reported to mediate cell transfer in inflammatory diseases such as arthritis, SCHERING CORPORATION 2003-07-31 US claimed
US-20030139446-A1 Preparation of pharmaceutical salts SCHERING CORPORATION 2003-07-24 US claimed
WO-2003048153-A1 PROCESS FOR THE PREPARATION OF COMPOSITIONS HAVING AN INCREASED AMOUNT OF PHARMACEUTICALLY ACTIVE SALTS OF ROTAMERS SCHERING CORPORATION (US) 2003-06-12 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210284604-A1 Amino Acid Derivatives and Their Uses BCAT2, BCAT1, SLC1A5 SMN1; SMN2 3546/4885ALDH1A1 809/4885CYP1A2 852/4885
US-20030139446-A1 Preparation of pharmaceutical salts PKD1, REN, ADCYAP1R1 SMN1; SMN2 1486/4885ALDH1A1 1255/4885CYP1A2 871/4885
US-11459341-B1 Organic anion lithium ionic cocrystal compounds and compositions SLC10A6, MLX, LPXN SMN1; SMN2 3280/4885ALDH1A1 1450/4885CYP1A2 870/4885
US-20200115331-A1 Amino Acid Derivatives and Their Uses BCAT1, BCAT2, SLC1A5 SMN1; SMN2 4366/4885ALDH1A1 997/4885CYP1A2 1271/4885
US-20220226205-A1 Coated Particles and Their Uses CD63, EPCAM, CD44 SMN1; SMN2 2837/4885ALDH1A1 4610/4885CYP1A2 4762/4885
US-20060241295-A1 Preparation of pharmaceutical salts of piperazine compounds ADCYAP1R1, CYP3A5, RAP2C SMN1; SMN2 3848/4885ALDH1A1 847/4885CYP1A2 235/4885
US-20030144510-A1 receptor which are useful for the treatment of AIDS and related HIV infections, including the compound of Formula I. CCR-5 receptors have also been reported to mediate cell transfer in inflammatory diseases such as arthritis, CCR1, CCR5, CCR6 SMN1; SMN2 2575/4885ALDH1A1 845/4885CYP1A2 2914/4885
US-10870665-B1 Organic anion lithium ionic cocrystal compounds and compositions SLC10A6, MLX, LPXN SMN1; SMN2 3280/4885ALDH1A1 1450/4885CYP1A2 870/4885
US-20050171117-A1 Preparation of pharmaceutical salts PKD1, REN, ADCYAP1R1 SMN1; SMN2 2045/4885ALDH1A1 1141/4885CYP1A2 877/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.