SCHEMBL2393938

SCHEMBL2393938

NC(=O)Cc1ccccc1-c1cc(F)cc(F)c1F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 2/20 0.37
CES2 O00748 1/20 0.36
CES1 P23141 1/20 0.36
ICMT O60725 4/20 0.36
ATR Q13535 1/20 0.36
ALDH1A1 P00352 1/20 0.36
PKM P14618 1/20 0.34
LMNA P02545 1/20 0.34
RAB9A P51151 1/20 0.34
KCNN4 O15554 1/20 0.33
CFD P00746 1/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
LOX P28300 1/20 0.33
KCNK3 O14649 1/20 0.33
KCNK5 O95279 1/20 0.33
KCNK17 Q96T54 1/20 0.33
KCNK9 Q9NPC2 1/20 0.33
RORC P51449 1/20 0.33
TRPM8 Q7Z2W7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9890790 0.83 PKM (0.40) KCNA5ICMTALDH1A1PKMLMNA
SCHEMBL2393136 0.83 SLC9A1 (0.42) KCNA5CES2CES1ICMTPKM
SCHEMBL2395880 0.83 ALDH1A1 (0.41) CES2CES1ATRALDH1A1LMNA
SCHEMBL2395669 0.81 ATR (0.39) ICMTATRALDH1A1LMNARAB9A
SCHEMBL2391854 0.80 ALDH1A1 (0.45) ATRALDH1A1LMNARAB9AMAOB
SCHEMBL9890738 0.80 ALDH1A1 (0.41) ICMTATRALDH1A1LMNARAB9A
SCHEMBL2392135 0.80 ICMT (0.44) ICMTATRCFD
SCHEMBL2397530 0.78 CTSL (0.43) CES2CES1ICMTATRALDH1A1
SCHEMBL2394997 0.78 DPP4 (0.40) ICMTALDH1A1PKM
SCHEMBL9890744 0.78 SLC9A1 (0.41) ICMTPKMLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120142771-A1 BIPHENYLACETAMIDE DERIVATIVE DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2012-06-07 US claimed
CN-102282124-A Biphenylacetamide derivative 2011-12-14 CN claimed
EP-2374790-A1 BIPHENYLACETAMIDE DERIVATIVE Dainippon Sumitomo Pharma Co., Ltd. (JP) 2011-10-12 EP claimed
US-20110224304-A1 BIPHENYLACETAMIDE DERIVATIVE DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2011-09-15 US claimed
US-20120142771-A1 BIPHENYLACETAMIDE DERIVATIVE DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2012-06-07 US disclosed
US-20120142771-A1 BIPHENYLACETAMIDE DERIVATIVE DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2012-06-07 US disclosed
US-20120142771-A1 BIPHENYLACETAMIDE DERIVATIVE DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2012-06-07 US disclosed
CN-102282124-A Biphenylacetamide derivative 2011-12-14 CN disclosed
EP-2374790-A1 BIPHENYLACETAMIDE DERIVATIVE Dainippon Sumitomo Pharma Co., Ltd. (JP) 2011-10-12 EP disclosed
EP-2374790-A1 BIPHENYLACETAMIDE DERIVATIVE Dainippon Sumitomo Pharma Co., Ltd. (JP) 2011-10-12 EP disclosed
US-20110224304-A1 BIPHENYLACETAMIDE DERIVATIVE DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2011-09-15 US disclosed
US-20110224304-A1 BIPHENYLACETAMIDE DERIVATIVE DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2011-09-15 US disclosed
US-20110224304-A1 BIPHENYLACETAMIDE DERIVATIVE DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2011-09-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120142771-A1 BIPHENYLACETAMIDE DERIVATIVE HRH3, KCNH3, BRPF3 KCNA5 41/4885CES2 1468/4885CES1 610/4885
US-20110224304-A1 BIPHENYLACETAMIDE DERIVATIVE HRH3, KCNH3, BRPF3 KCNA5 41/4885CES2 1468/4885CES1 610/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.