SCHEMBL2397951

SCHEMBL2397951

CSc1ccc(OC(F)(F)[C@H](OS(=O)(=O)C(F)(F)F)c2ccc(F)cc2)cc1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.36
MAPK1 P28482 1/20 0.36
NR3C1 P04150 2/20 0.33
PGR P06401 1/20 0.33
CXCR2 P25025 2/20 0.33
ALOX5 P09917 1/20 0.33
CXCR1 P25024 1/20 0.32
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31
LMNA P02545 1/20 0.30
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2397948 1.00 ALDH1A1 (0.36) ALDH1A1MAPK1NR3C1PGRCXCR2
SCHEMBL2399535 0.75 ALOX5 (0.42) ALDH1A1MAPK1NR3C1ALOX5SLC6A2
SCHEMBL2399533 0.75 ALOX5 (0.42) ALDH1A1MAPK1NR3C1ALOX5SLC6A2
SCHEMBL1272882 0.74 IDO1 (0.34) CXCR2CXCR1
SCHEMBL12800457 0.74 IDO1 (0.34) CXCR2CXCR1
SCHEMBL2100565 0.74 IDO1 (0.34) CXCR2CXCR1
SCHEMBL1272889 0.71 POLB (0.36) CXCR2CXCR1
SCHEMBL11699965 0.70 CXCR2 (0.44) ALDH1A1MAPK1CXCR2CXCR1LMNA
SCHEMBL2396614 0.68 CTSL (0.42) ALDH1A1NR3C1LMNAGAA
SCHEMBL2396618 0.68 CTSL (0.42) ALDH1A1NR3C1LMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8013186-B2 Haloalkyl containing compounds as cysteine protease inhibitors VIROBAY, INC. (US) 2011-09-06 US disclosed
US-20090023781-A1 Haloalkyl Containing Compounds as Cysteine Protease Inhibitors VIROBAY, INC. (US) 2009-01-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090023781-A1 Haloalkyl Containing Compounds as Cysteine Protease Inhibitors CTSF, CTSS, CTSE ALDH1A1 1944/4885MAPK1 4492/4885NR3C1 4864/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.