SCHEMBL2399535

SCHEMBL2399535

CSc1ccc(OC(F)(F)[C@H](O)c2ccc(F)cc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.42
NR3C1 P04150 1/20 0.37
SLC6A4 P31645 2/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A3 Q01959 1/20 0.35
ALDH1A1 P00352 2/20 0.33
MAPK1 P28482 1/20 0.33
PTGS1 P23219 1/20 0.33
CASR P41180 1/20 0.33
GAA P10253 2/20 0.33
GABBR2 O75899 1/20 0.33
GABBR1 Q9UBS5 1/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
LMNA P02545 1/20 0.32
MAOB P27338 1/20 0.32
AOC3 Q16853 1/20 0.32
CYP1A1 P04798 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP1B1 Q16678 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2399533 1.00 ALOX5 (0.42) ALOX5NR3C1SLC6A4SLC6A2SLC6A3
SCHEMBL2397951 0.75 ALDH1A1 (0.36) ALOX5NR3C1SLC6A4SLC6A2SLC6A3
SCHEMBL2397948 0.75 ALDH1A1 (0.36) ALOX5NR3C1SLC6A4SLC6A2SLC6A3
SCHEMBL2396618 0.72 CTSL (0.42) NR3C1ALDH1A1GAAMEN1KMT2A
SCHEMBL2396614 0.72 CTSL (0.42) NR3C1ALDH1A1GAAMEN1KMT2A
SCHEMBL7917238 0.72 ALOX5 (0.33) ALOX5SLC6A4ALDH1A1LMNAMAOB
SCHEMBL2337214 0.72 ALOX5 (0.33) ALOX5SLC6A4ALDH1A1LMNAMAOB
SCHEMBL2401014 0.71 GAA (0.44) NR3C1SLC6A4SLC6A2SLC6A3ALDH1A1
SCHEMBL514680 0.69 CYP1A1 (0.44) SLC6A4SLC6A2SLC6A3ALDH1A1LMNA
SCHEMBL315215 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8013186-B2 Haloalkyl containing compounds as cysteine protease inhibitors VIROBAY, INC. (US) 2011-09-06 US disclosed
US-20090023781-A1 Haloalkyl Containing Compounds as Cysteine Protease Inhibitors VIROBAY, INC. (US) 2009-01-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090023781-A1 Haloalkyl Containing Compounds as Cysteine Protease Inhibitors CTSF, CTSS, CTSE ALOX5 1384/4885NR3C1 4864/4885SLC6A4 2592/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.