SCHEMBL2407640

SCHEMBL2407640

CNC(=O)OC(c1cc(Br)n(S(=O)(=O)c2cccc(OC)c2)c1)C(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MET P08581 1/20 0.39
HDAC1 Q13547 3/20 0.38
MEP1B Q16820 1/20 0.38
HTR6 P50406 7/20 0.37
CYP3A4 P08684 1/20 0.37
HDAC2 Q92769 2/20 0.36
HDAC8 Q9BY41 2/20 0.36
HDAC6 Q9UBN7 2/20 0.36
HDAC3 O15379 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC11 Q96DB2 1/20 0.36
ABCC9 O60706 1/20 0.35
ABCC8 Q09428 1/20 0.35
KCNJ11 Q14654 1/20 0.35
KCNJ8 Q15842 1/20 0.35
KEAP1 Q14145 1/20 0.35
NFE2L2 Q16236 1/20 0.35
MTNR1B P49286 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ALDH1A1 P00352 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2416547 0.87 HTR6 (0.35) HTR6ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL4412054 0.87 MET (0.40) METHDAC1HTR6CYP3A4NFE2L2
SCHEMBL2411499 0.83 ADAM17 (0.35) HDAC1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL2415052 0.77 MEP1B (0.43) METHDAC1MEP1BHTR6CYP3A4
SCHEMBL4418740 0.72 MET (0.41) METHDAC1HTR6HDAC2HDAC8
SCHEMBL28715560 0.71 HTR6 (0.49) METMEP1BHTR6CYP3A4KEAP1
SCHEMBL4424529 0.71 HTR6 (0.44) METHTR6CYP3A4ALDH1A1LMNA
SCHEMBL4424525 0.71 MET (0.44) METHDAC1HTR6CYP3A4HDAC2
SCHEMBL4419026 0.70 MET (0.40) METHDAC1HTR6HDAC2HDAC8
SCHEMBL2409947 0.70 HTR6 (0.35) METHTR6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364979-A1 Pyrrole compounds Takeda Pharmaceutical Company Limited (JP) 2011-09-14 EP disclosed