SCHEMBL24252407

SCHEMBL24252407

O=C1C=C(c2ccncn2)C(N2CCCCC2)O1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 9/20 0.40
ROCK2 O75116 1/20 0.34
ROCK1 Q13464 1/20 0.34
CDC42BPB Q9Y5S2 1/20 0.34
SCD O00767 1/20 0.32
SCD5 Q86SK9 1/20 0.32
OPRK1 P41145 1/20 0.31
CAMKK2 Q96RR4 1/20 0.30
UCHL1 P09936 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2D6 P10635 1/20 0.30
CSNK1A1 P48729 1/20 0.30
GSK3A P49840 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24252414 0.99 GSK3B (0.38) GSK3BROCK2ROCK1CDC42BPBSCD
SCHEMBL24252413 0.88 GSK3B (0.43) GSK3BCYP1A2CYP2D6CSNK1A1GSK3A
SCHEMBL24252377 0.79 HRH3 (0.35)
SCHEMBL24252378 0.77 LMNA (0.35)
SCHEMBL24252370 0.76 ROCK2 (0.34) ROCK2ROCK1CDC42BPBOPRK1
SCHEMBL24252374 0.75 ROCK2 (0.32) ROCK2ROCK1CDC42BPB
SCHEMBL24252410 0.74 CCNT1 (0.33) GSK3BSCDSCD5CAMKK2CYP2D6
SCHEMBL24252409 0.73 CCNT1 (0.33) GSK3BSCDSCD5CAMKK2
SCHEMBL24252408 0.70 GSK3B (0.33) GSK3BCYP2D6
SCHEMBL24252411 0.70 CYP2D6 (0.33) GSK3BCYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022034203-A1 PROCESS FOR THE PREPARATION OF PYRIDAZINONE DERIVATIVES SYNGENTA CROP PROTECTION AG (CH) 2022-02-17 WO disclosed