SCHEMBL24316438

SCHEMBL24316438

Cc1cnc2ccc(Oc3ccc(OCc4ccc(F)c(Cl)c4)nc3)cn2c1=O

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 2/20 0.43
P2RX7 Q99572 12/20 0.36
FFAR1 O14842 1/20 0.34
AXL P30530 1/20 0.34
PIK3CA P42336 1/20 0.34
MTOR P42345 1/20 0.34
PLA2G7 Q13093 1/20 0.34
P2RX3 P56373 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24316432 0.86 ACACB (0.37) GRM5PIK3CAMTOR
SCHEMBL24316428 0.83 ALKBH1 (0.39) GRM5
SCHEMBL24316623 0.77 P2RX3 (0.39) GRM5P2RX3
SCHEMBL24316814 0.76 CSF1R (0.47) GRM5P2RX7PIK3CAMTORP2RX3
SCHEMBL24316565 0.76 CSF1R (0.44) GRM5PIK3CAMTOR
SCHEMBL24316436 0.73 KDM4E (0.37) GRM5PIK3CAMTOR
SCHEMBL24316434 0.72 CSF1R (0.53) GRM5PIK3CAMTOR
SCHEMBL24316659 0.72 ALKBH1 (0.40) GRM5
SCHEMBL24316545 0.72 CSF1R (0.43) GRM5PIK3CAMTOR
SCHEMBL24316624 0.71 KDM4E (0.36) GRM5PIK3CAMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022057895-A1 HETEROAROMATIC COMPOUNDS AND USES THEREOF HUTCHISON MEDIPHARMA LIMITED (CN) 2022-03-24 WO disclosed
US-9585884-B2 Pyrimidinone inhibitors of lipoprotein-associated phospholipase A2 AUSPEX PHARMACEUTICALS, INC. (US) 2017-03-07 US disclosed