Edetic Acid

Edetic Acid

SCHEMBL243998

O=C([O-])CN(CCN(CC(=O)[O-])CC(=O)[O-])CC(=O)[O-].[Cu+2].[Na+].[Na+]

nearest known ligand 0.73

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Edetic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACE known ✓ P12821 1/20 0.48
CA4 known ✓ P22748 8/20 0.40
CA2 known ✓ P00918 4/20 0.35
CA1 known ✓ P00915 4/20 0.35
KDM4E B2RXH2 2/20 0.73
ALOX15 P16050 2/20 0.73
MAPT P10636 1/20 0.73
SMN1; SMN2 Q16637 1/20 0.73
TDP1 Q9NUW8 2/20 0.48
EYA2 O00167 1/20 0.48
APP P05067 1/20 0.48
BLM P54132 2/20 0.46
PMP22 Q01453 2/20 0.46
LMNA P02545 1/20 0.46
CHRM2 P08172 1/20 0.46
ADRA2A P08913 1/20 0.46
TSHR P16473 1/20 0.46
DRD1 P21728 1/20 0.46
SLC6A2 P23975 1/20 0.46
SLC6A4 P31645 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Edetic Acid SCHEMBL9540648 0.97 KDM4E (0.70) KDM4EALOX15MAPTSMN1; SMN2TDP1
Edetic Acid SCHEMBL15654929 0.97 KDM4E (0.70) KDM4EALOX15MAPTSMN1; SMN2TDP1
Edetic Acid SCHEMBL28905272 0.97 KDM4E (0.70) KDM4EALOX15MAPTSMN1; SMN2TDP1
Edetic Acid SCHEMBL333822 0.97 KDM4E (0.70) KDM4EALOX15MAPTSMN1; SMN2TDP1
Edetic Acid SCHEMBL44287 0.97 KDM4E (0.76) KDM4EALOX15MAPTSMN1; SMN2TDP1
Edetic Acid SCHEMBL42427 0.97 KDM4E (0.76) KDM4EALOX15MAPTSMN1; SMN2TDP1
Edetic Acid SCHEMBL906 0.97 KDM4E (0.76) KDM4EALOX15MAPTSMN1; SMN2TDP1
Edetic Acid SCHEMBL3835316 0.97 KDM4E (0.76) KDM4EALOX15MAPTSMN1; SMN2TDP1
Edetic Acid SCHEMBL18983963 0.97 KDM4E (0.68) KDM4EALOX15MAPTSMN1; SMN2TDP1
Edetic Acid SCHEMBL144663 0.97 KDM4E (0.68) KDM4EALOX15MAPTSMN1; SMN2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 264 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240375330-A1 METHOD FOR PREPARING METAL-POLYMER RESIN COMPOSITE PLASTAL CO., LTD. (KR) 2024-11-14 US claimed
EP-4461505-A1 METHOD FOR PREPARING METAL-POLYMER RESIN COMPOSITE Plastal Co., Ltd. (KR) 2024-11-13 EP claimed
CN-118651847-A Carbon dot for zinc ion battery and preparation method thereof 郑州大学 2024-09-17 CN claimed
CN-118515974-A PPS reinforcing material with high heat conduction and preparation method thereof 国材(苏州)新材料科技有限公司 2024-08-20 CN claimed
CN-114921832-B Method for generating black ceramic film on surface of titanium alloy 常州大学 2024-02-13 CN claimed
EP-4196085-A1 SEMI-PERMANENT TATTOOS inkbox ink Inc. (CA) 2023-06-21 EP claimed
CN-115739119-A Copper particle-loaded sulfur-zinc-indium composite material and preparation method and application thereof 浙江工业大学 2023-03-07 CN claimed
CN-115521180-A Formula of matrix-cultured leek nutrient solution and culture process 宁波市蔚蓝智谷智能装备有限公司 2022-12-27 CN claimed
CN-114920602-A Preparation method of environment-friendly nutritional wettable powder 江苏剑牌农化股份有限公司 2022-08-19 CN claimed
CN-114921832-A Method for generating black ceramic film on surface of titanium alloy 常州大学 2022-08-19 CN claimed
WO-2010083318-A2 FUNGICIDAL COMPOSITIONS INCLUDING HYDRAZONE DERIVATIVES AND COPPER DOW AGROSCIENCES LLC (US) 2010-07-22 WO claimed
WO-2010083322-A2 FUNGICIDAL COMPOSITIONS INCLUDING HYDRAZONE DERIVATIVES AND COPPER DOW AGROSCIENCES LLC (US) 2010-07-22 WO claimed
WO-2010083319-A2 FUNGICIDAL COMPOSITIONS INCLUDING HYDRAZONE DERIVATIVES AND COPPER DOW AGROSCIENCES LLC (US) 2010-07-22 WO claimed
WO-2010083307-A2 SYNERGISTIC FUNGICIDAL COMPOSITIONS INCLUDING HYDRAZONE DERIVATIVES AND COPPER DOW AGROSCIENCES LLC (US) 2010-07-22 WO claimed
EP-1628655-A4 ANTISEPTIC COMPOSITIONS, METHODS AND SYSTEMS TYCO HEALTHCARE (US) 2008-10-15 EP claimed
JP-2006526664-A 2006-11-24 JP claimed
EP-1628655-A2 ANTISEPTIC COMPOSITIONS, METHODS AND SYSTEMS Tyco Healthcare Group LP (US) 2006-03-01 EP claimed
WO-2004108093-A2 ANTISEPTIC COMPOSITIONS, METHODS AND SYSTEMS TYCO HEALTHCARE GROUP LP (US) 2004-12-16 WO claimed
US-5597556-A Colored bicarbonate containing solid composition THE MENNEN COMPANY (US) 1997-01-28 US claimed
WO-1996032925-A1 COLORED BICARBONATE CONTAINING SOLID COMPOSITION COLGATE-PALMOLIVE COMPANY (US) 1996-10-24 WO claimed