SCHEMBL244963

SCHEMBL244963

Clc1nc(Cl)c2ncn(C3CCCCO3)c2n1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
YTHDC1 Q96MU7 1/20 0.72
CYP2C19 P33261 1/20 0.53
TP53 P04637 2/20 0.50
MEN1 O00255 2/20 0.50
ALDH1A1 P00352 2/20 0.50
KMT2A Q03164 2/20 0.50
CYP2C9 P11712 1/20 0.50
NFKB1 P19838 1/20 0.50
MAPK1 P28482 1/20 0.50
HSD17B10 Q99714 1/20 0.50
APEX1 P27695 1/20 0.50
PI4KA P42356 1/20 0.50
BLM P54132 1/20 0.50
ADCY1 Q08828 1/20 0.50
PI4K2B Q8TCG2 1/20 0.50
PI4K2A Q9BTU6 1/20 0.50
PI4KB Q9UBF8 1/20 0.50
CYP1A2 P05177 1/20 0.48
TSHR P16473 1/20 0.48
LMNA P02545 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20275400 1.00 YTHDC1 (0.72) YTHDC1CYP2C19TP53MEN1ALDH1A1
SCHEMBL29353722 1.00 YTHDC1 (0.72) YTHDC1CYP2C19TP53MEN1ALDH1A1
SCHEMBL4151824 0.96 YTHDC1 (0.66) YTHDC1CYP2C19TP53MEN1ALDH1A1
SCHEMBL2489808 0.93 YTHDC1 (0.64) YTHDC1CYP2C19TP53MEN1ALDH1A1
SCHEMBL7265843 0.89 YTHDC1 (0.62) YTHDC1CYP2C19TP53MEN1ALDH1A1
SCHEMBL9885109 0.88 YTHDC1 (0.74) YTHDC1CYP2C19TP53MEN1ALDH1A1
SCHEMBL7265845 0.87 YTHDC1 (0.57) YTHDC1CYP2C19TP53MEN1ALDH1A1
SCHEMBL179599 0.87 YTHDC1 (0.59) YTHDC1CYP2C19TP53MEN1ALDH1A1
SCHEMBL4133669 0.87 YTHDC1 (0.59) YTHDC1CYP2C19TP53MEN1ALDH1A1
SCHEMBL20275350 0.87 YTHDC1 (0.69) YTHDC1CYP2C19TP53MEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 702 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260125395-A1 PROCESS FOR THE PREPARATION OF TRICYCLIC PI3K INHIBITOR COMPOUNDS AND METHODS FOR USING THE SAME FOR THE TREATMENT OF CANCER GENENTECH INC (US) 2026-05-07 US disclosed
US-12569566-B2 Compositions containing, methods and uses of antibody-TLR agonist conjugates AMBRX, INC. (US) 2026-03-10 US disclosed
EP-4694893-A1 NOVEL INHIBITORS OF PIKFYVE AND METHODS USING SAME TME Therapeutics LLC (US) 2026-02-18 EP disclosed
US-20250388599-A1 TRICYCLIC PI3K INHIBITOR COMPOUNDS AND METHODS OF USE GENENTECH INC (US) 2025-12-25 US disclosed
US-20250388582-A1 NOVEL BICYCLIC HETEROARYL COMPOUND AND USE THEREOF ILDONG PHARMACEUTICAL CO LTD (KR) 2025-12-25 US disclosed
US-20250353851-A1 PURINES AND METHODS OF THEIR USE KINETA INC (US) 2025-11-20 US disclosed
US-20250346601-A1 HETEROCYCLIC COMPOUNDS FOR THE PREVENTION AND THERAPY OF CIRCADIAN RHYTHM DISORDERS UNIV PALACKEHO (CZ) 2025-11-13 US disclosed
EP-4532498-B1 HETEROCYCLIC COMPOUNDS FOR THE PREVENTION AND THERAPY OF CIRCADIAN RHYTHM DISORDERS UNIV PALACKEHO (CZ) 2025-10-29 EP disclosed
US-12421273-B2 Ectonucleotidase inhibitors and methods of use thereof ANTENGENE THERAPEUTICS LIMITED (CN) 2025-09-23 US disclosed
EP-4178959-B1 NITROGEN HETEROCYCLIC CYTOKININ DERIVATIVES, COMPOSITIONS CONTAINING THESE DERIVATIVES AND USE THEREOF UNIV PALACKEHO (CZ) 2025-09-10 EP disclosed
WO-2001094368-A1 2-AMINOCARBONYL-9H-PURINE DERIVATIVES PFIZER LIMITED (GB) 2001-12-13 WO disclosed
US-6326359-B1 PURINE DERIVATIVES PFIZER INC 2001-12-04 US disclosed
US-20010020089-A1 Purine derivatives PFIZER INC. 2001-09-06 US disclosed
WO-2001060835-A1 PURINE DERIVATIVES PFIZER LIMITED (GB) 2001-08-23 WO disclosed
EP-1121372-A1 ADENINE DERIVATIVES Pfizer Limited (GB) 2001-08-08 EP disclosed
WO-2001027131-A1 PURINE DERIVATIVES PFIZER LIMITED (GB) 2001-04-19 WO disclosed
WO-2001027130-A1 PURINE DERIVATIVES PFIZER LIMITED (GB) 2001-04-19 WO disclosed
WO-2000077018-A2 PURINE DERIVATIVES PFIZER LIMITED (GB) 2000-12-21 WO disclosed
WO-2000023457-A1 ADENINE DERIVATIVES PFIZER LIMITED (GB) 2000-04-27 WO disclosed
US-4241063-A Purine derivatives and their use as bronchodilators BRISTOL-MYERS COMPANY (US) 1980-12-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250346601-A1 HETEROCYCLIC COMPOUNDS FOR THE PREVENTION AND THERAPY OF CIRCADIAN RHYTHM DISORDERS CRY1, PER2, CRY2 YTHDC1 812/4885CYP2C19 256/4885TP53 4795/4885
US-20010020089-A1 Purine derivatives ADORA2A, ADORA1, ADORA3 YTHDC1 1043/4885CYP2C19 295/4885TP53 3378/4885
US-20260125395-A1 PROCESS FOR THE PREPARATION OF TRICYCLIC PI3K INHIBITOR COMPOUNDS AND METHODS FOR USING THE SAME FOR THE TREATMENT OF CANCER PIK3C2B, PIK3C2A, PIK3CA YTHDC1 4104/4885CYP2C19 584/4885TP53 374/4885
US-12421273-B2 Ectonucleotidase inhibitors and methods of use thereof NT5E, ENTPD5, NT5C2 YTHDC1 3612/4885CYP2C19 977/4885TP53 2516/4885
US-20250388582-A1 NOVEL BICYCLIC HETEROARYL COMPOUND AND USE THEREOF GBA1, PIKFYVE, MAN2B1 YTHDC1 3248/4885CYP2C19 4174/4885TP53 1437/4885
US-12569566-B2 Compositions containing, methods and uses of antibody-TLR agonist conjugates TLR3, TLR2, TLR1 YTHDC1 3411/4885CYP2C19 1699/4885TP53 1089/4885
US-20250353851-A1 PURINES AND METHODS OF THEIR USE TDP1, TDP2, PIKFYVE YTHDC1 2276/4885CYP2C19 4257/4885TP53 1604/4885
US-20250388599-A1 TRICYCLIC PI3K INHIBITOR COMPOUNDS AND METHODS OF USE PIK3C2B, PIK3C2A, PIK3R1 YTHDC1 3570/4885CYP2C19 2219/4885TP53 751/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.