Fentonium

Fentonium

SCHEMBL24584

C[N+]1(CC(=O)c2ccc(-c3ccccc3)cc2)C2CCC1CC(OC(=O)C(CO)c1ccccc1)C2.[Br-]

nearest known ligand 0.69

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHKACHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGHRH2OPRM1

The experimentally established mechanism targets of Fentonium. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 known ✓ P08172 8/20 0.67
CHRM5 known ✓ P08912 6/20 0.64
CHRM1 known ✓ P11229 6/20 0.64
CHRM3 known ✓ P20309 5/20 0.64
CHRM4 known ✓ P08173 4/20 0.64
BLM P54132 4/20 0.69
PABPC1 P11940 1/20 0.66
CYP2C19 P33261 1/20 0.64
MEN1 O00255 3/20 0.64
KMT2A Q03164 3/20 0.64
SMN1; SMN2 Q16637 2/20 0.64
TSHR P16473 2/20 0.63
CYP3A4 P08684 1/20 0.55
CYP2C9 P11712 1/20 0.55
HIF1A Q16665 1/20 0.55
HSD17B10 Q99714 1/20 0.55
KDM4E B2RXH2 1/20 0.53
LMNA P02545 1/20 0.53
POLB P06746 1/20 0.53
ADRA2C P18825 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fentonium SCHEMBL30186606 1.00 BLM (0.69) BLMCHRM2PABPC1CYP2C19CHRM5
Fentonium SCHEMBL24583 1.00 BLM (0.69) BLMCHRM2PABPC1CYP2C19CHRM5
Fentonium SCHEMBL251444 0.99 CHRM2 (0.68) BLMCHRM2PABPC1CYP2C19CHRM5
Fentonium SCHEMBL13724144 0.88 CHRM1 (0.58) BLMCHRM2PABPC1CYP2C19CHRM5
Xenytropium SCHEMBL29371652 0.86 BLM (0.71) BLMCHRM2PABPC1CYP2C19CHRM5
Xenytropium SCHEMBL24707 0.86 BLM (0.71) BLMCHRM2PABPC1CYP2C19CHRM5
Xenytropium SCHEMBL30428452 0.85 CHRM2 (0.71) BLMCHRM2PABPC1CYP2C19CHRM5
Xenytropium SCHEMBL29361010 0.85 CHRM2 (0.71) BLMCHRM2PABPC1CYP2C19CHRM5
SCHEMBL14507225 0.82 CHRM2 (0.80) BLMCHRM2PABPC1CYP2C19CHRM5
Methylatropine SCHEMBL30647266 0.82 BLM (1.00) BLMCHRM2PABPC1CYP2C19CHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 476 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108430482-A Control of cellular redox levels 伊丽莎白·麦克纳 2018-08-21 CN claimed
US-20140171645-A1 ELECTROPHILIC ALKYLATING REAGENTS, THEIR PREPARATION AND USE HOVIONE INTER LTD. (CH) 2014-06-19 US claimed
EP-2691367-A1 ELECTROPHILIC ALKYLATING REAGENTS, THEIR PREPARATION AND USE Hovione Inter Ltd. (CH) 2014-02-05 EP claimed
CN-103502211-A Electrophilic alkylating reagents, preparation and use thereof HOVIONE FARMACIENCIA S A 2014-01-08 CN claimed
WO-2012131286-A1 ELECTROPHILIC ALKYLATING REAGENTS, THEIR PREPARATION AND USE HOVIONE INTER. LTD (CH) 2012-10-04 WO claimed
US-20100144657-A1 PHENYLPIPERIDINE MODULATORS OF mu-OPIOID RECEPTORS AUSPEX PHARMACEUTICALS, INC. (US) 2010-06-10 US claimed
EP-1879578-A4 METHODS AND COMPOSITIONS FOR THE TREATMENT OF URINARY INCONTINENCE DOV PHARMACEUTICAL INC (US) 2009-05-13 EP claimed
EP-1879578-A2 METHODS AND COMPOSITIONS FOR THE TREATMENT OF URINARY INCONTINENCE DOV Pharmaceutical Inc. (US) 2008-01-23 EP claimed
WO-2006102029-A9 METHODS AND COMPOSITIONS FOR THE TREATMENT OF URINARY INCONTINENCE DOV PHARMACEUTICAL INC (US) 2006-12-07 WO claimed
WO-2006102029-A2 METHODS AND COMPOSITIONS FOR THE TREATMENT OF URINARY INCONTINENCE DOV PHARMACEUTICAL, INC. (US) 2006-09-28 WO claimed
EP-1273301-B1 Pharmaceutical preparations based on active ingredients susceptible to illicit administration ALTERGON SA (CH) 2006-09-06 EP claimed
EP-1273301-A2 Pharmaceutical preparations based on active ingredients susceptible to illicit administration ALTERGON S.A. (CH) 2003-01-08 EP claimed
CN-1294519-A Pharmaceutical composition containing a compound having an activity of promoting the absorption of an active ingredient INPHARMA SA (CH) 2001-05-09 CN claimed
EP-1073470-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2001-02-07 EP claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed
EP-4168092-B1 BALLOON CATHETER WITH PRECISION DRUG-ELUTING CAPABILITY BARD INC C R (US) 2026-05-27 EP disclosed
US-20260097102-A1 Treatment Of Respiratory Disorders With Arachidonate 15-Lipoxygenase (ALOX15) Inhibitors REGENERON PHARMA (US) 2026-04-09 US disclosed
WO-1996040084-A1 COMPOSITIONS AND METHODS FOR USE OF PRESSURE SENSITIVE ADHESIVE TRANSDERMAL DEVICES CONTAINING A BIOADHESIVE HUMECTANT NOVEN PHARMACEUTICALS, INC. (US) 1996-12-19 WO disclosed
EP-0737066-A1 TRANSDERMAL DEVICE CONTAINING POLYVINYLPYRROLIDONE AS SOLUBILITY ENHANCER NOVEN PHARMACEUTICALS, INC. (US) 1996-10-16 EP disclosed
WO-1995018603-A1 TRANSDERMAL DEVICE CONTAINING POLYVINYLPYRROLIDONE AS SOLUBILITY ENHANCER NOVEN PHARMACEUTICALS, INC. (US) 1995-07-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100144657-A1 PHENYLPIPERIDINE MODULATORS OF mu-OPIOID RECEPTORS OPRM1, OPRK1, OPRD1 CHRM2 116/4885CHRM5 23/4885CHRM1 71/4885
US-20260097102-A1 Treatment Of Respiratory Disorders With Arachidonate 15-Lipoxygenase (ALOX15) Inhibitors ALOX15, ALOX15B, ALOX5 CHRM2 4475/4885CHRM5 3509/4885CHRM1 4534/4885
US-20140171645-A1 ELECTROPHILIC ALKYLATING REAGENTS, THEIR PREPARATION AND USE MGMT, MCL1, TOP2B CHRM2 2607/4885CHRM5 3007/4885CHRM1 3157/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.