SCHEMBL2463879

SCHEMBL2463879

NC(=O)c1ccc(C(N)=O)c(NCCN2CCOCC2)c1

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.58
ALDH1A1 P00352 2/20 0.49
AR P10275 1/20 0.48
CD274 Q9NZQ7 4/20 0.47
POLB P06746 1/20 0.47
HTR1A P08908 1/20 0.47
MAOA P21397 1/20 0.47
MAOB P27338 1/20 0.47
KCNH2 Q12809 1/20 0.47
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C19 P33261 1/20 0.46
HPGD P15428 1/20 0.45
PARP1 P09874 1/20 0.45
HSP90AA1 P07900 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11465420 0.83 ALDH1A1 (0.66) KDM4EALDH1A1CD274POLBHPGD
SCHEMBL3222256 0.80 EPHX2 (0.54) KDM4EALDH1A1CD274POLBHTR1A
SCHEMBL11465072 0.80 KDM4E (0.50) KDM4EALDH1A1ARCD274POLB
SCHEMBL3230823 0.79 HTR7 (0.63) KDM4EALDH1A1CYP1A2CYP2D6CYP2C19
SCHEMBL27516593 0.78 KDM4E (0.46) KDM4EALDH1A1ARCD274POLB
SCHEMBL4524250 0.76 KDM4E (0.63) KDM4EALDH1A1POLBPARP1
SCHEMBL23286940 0.75 ALDH1A1 (0.54) KDM4EALDH1A1CD274POLBCYP2C19
SCHEMBL3770520 0.75 LMNA (0.74) KDM4EALDH1A1CD274POLBCYP1A2
SCHEMBL12513990 0.74 SMN1; SMN2 (0.55) KDM4EALDH1A1CD274HTR1AMAOA
SCHEMBL30216224 0.74 KDM4E (1.00) KDM4EALDH1A1ARPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8012956-B2 Tropane compounds EXELIXIS, INC. (US) 2011-09-06 US claimed
US-20090163471-A1 Tropane compounds EXELIXIS, INC. 2009-06-25 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090163471-A1 Tropane compounds ADRA1B, ADRA2B, ADRB2 KDM4E 4402/4885ALDH1A1 323/4885AR 361/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.