SCHEMBL2464591

SCHEMBL2464591

COc1ccccc1-c1c(C(N)=O)ccc(C(N)=O)c1N

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 2/20 0.48
PARP1 P09874 1/20 0.47
MAP2 P11137 2/20 0.45
CDC7 O00311 1/20 0.45
KEAP1 Q14145 1/20 0.45
NFE2L2 Q16236 1/20 0.45
GRK6 P43250 1/20 0.44
ALDH1A1 P00352 3/20 0.43
HPGD P15428 2/20 0.43
GAA P10253 1/20 0.43
HSD17B10 Q99714 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
APP P05067 1/20 0.42
SLC9A1 P19634 2/20 0.42
GPR35 Q9HC97 1/20 0.42
KDM4E B2RXH2 1/20 0.42
IRAK4 Q9NWZ3 1/20 0.41
CTSD P07339 1/20 0.41
HTT P42858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4117320 0.81 MYC (0.54) IKBKBPARP1MAP2CDC7KEAP1
SCHEMBL5582517 0.80 PARP1 (0.52) IKBKBPARP1MAP2CDC7KEAP1
SCHEMBL2491692 0.79 KDM4E (0.43) ALDH1A1HSD17B10L3MBTL1KDM4E
SCHEMBL3675429 0.79 EGFR (0.47) IKBKBPARP1MAP2CDC7ALDH1A1
SCHEMBL527995 0.78 PARP1 (0.56) IKBKBPARP1CDC7KEAP1NFE2L2
SCHEMBL5517143 0.78 PARP1 (0.50) IKBKBPARP1MAP2CDC7KEAP1
SCHEMBL165834 0.76 HTT (0.49) PARP1ALDH1A1KDM4EIRAK4CTSD
SCHEMBL41435 0.75 KEAP1 (0.64) PARP1KEAP1NFE2L2GRK6ALDH1A1
SCHEMBL15517040 0.75 GPR35 (0.57) ALDH1A1HPGDGAAHSD17B10APP
SCHEMBL264288 0.74 IRAK4 (0.63) ALDH1A1HPGDL3MBTL1IRAK4CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8012956-B2 Tropane compounds EXELIXIS, INC. (US) 2011-09-06 US claimed
US-20090163471-A1 Tropane compounds EXELIXIS, INC. 2009-06-25 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090163471-A1 Tropane compounds ADRA1B, ADRA2B, ADRB2 IKBKB 3815/4885PARP1 3161/4885MAP2 1148/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.