SCHEMBL2476178

SCHEMBL2476178

CCOC(OCC)c1ccccc1Cc1cnccc1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 5/20 0.34
SLC6A4 P31645 5/20 0.34
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
SLC6A3 Q01959 2/20 0.32
MAPK8 P45983 1/20 0.32
ALDH1A1 P00352 3/20 0.32
ALOX15 P16050 1/20 0.32
MAPK1 P28482 1/20 0.32
CYP51A1 Q16850 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
KDM4E B2RXH2 1/20 0.31
CHUK O15111 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
HPGD P15428 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2474309 0.89 ALDH1A1 (0.33) SLC6A2SLC6A4SLC6A3ALDH1A1ALOX15
SCHEMBL2475970 0.81 LOXL2 (0.41) ADORA2AADORA1ALDH1A1KDM4E
SCHEMBL27547933 0.81 SGMS2 (0.35) SLC6A2SLC6A4ALDH1A1MAPK1NPC1
SCHEMBL2475915 0.76 CASP1 (0.36) SLC6A2SLC6A4SLC6A3HPGDHSD17B10
SCHEMBL8550005 0.72 NPC1 (0.34) ADORA2AADORA1NPC1CYP3A4
SCHEMBL6155730 0.70 CASP1 (0.45) SLC6A2SLC6A4SLC6A3MAPK1KDM4E
SCHEMBL8017632 0.70 HSPA5 (0.55) ADORA2AADORA1ALDH1A1ALOX15NPC1
SCHEMBL28446557 0.70 ALDH1A1 (0.38) ADORA2AADORA1ALDH1A1CYP51A1NPC1
SCHEMBL21806628 0.68 CYP4F2 (0.41) ALDH1A1NPC1RAB9AL3MBTL1
SCHEMBL27046064 0.67 CA12 (0.37) SLC6A2SLC6A4NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2159216-B1 3-BUTENYL-1-AMINE DERIVATIVES AND THEIR USE AS Ih MODULORS FOR THE TREATMENT OF PSYCHIATIRC DISORDERS ORGANON NV (NL) 2011-10-12 EP disclosed
EP-2159216-A1 Ih - Modulators N.V. Organon (NL) 2010-03-03 EP disclosed
US-20040229910-A1 Therapeutic compounds N.V. ORGANON (NL) 2004-11-18 US disclosed
US-20020037885-A1 Therapeutic compounds DIJCKS FREDERICUS ANTONIUS (NL) 2002-03-28 US disclosed
US-6313139-B1 ADMINISTERING BENZYLAMINE DERIVATIVE FOR THERAPY OF PSYCHIATRIC DISORDER IN MAMMALS AKZO NOBEL N. V. (NL) 2001-11-06 US disclosed
CN-1275909-A In-modulators AKZO NOBEL NV (NL) 2000-12-06 CN disclosed
EP-1035843-A2 I h?-MODULATORS Akzo Nobel N.V. (NL) 2000-09-20 EP disclosed
US-6080773-A USEFUL FOR TREATMENT OF DEPRESSION, ANXIETY OR PSYCHOSIS AKZO NOBEL, N.V. (NL) 2000-06-27 US disclosed
WO-1999018941-A2 Ih-MODULATORS AKZO NOBEL N.V. (NL) 1999-04-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040229910-A1 Therapeutic compounds BDNF, PNMT, SLC18A2 SLC6A2 15/4885SLC6A4 20/4885ADORA2A 71/4885
US-20020037885-A1 Therapeutic compounds BDNF, PNMT, SLC18A2 SLC6A2 15/4885SLC6A4 20/4885ADORA2A 71/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.