SCHEMBL2487358

SCHEMBL2487358

CNC(=O)c1ccc(NN)nc1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NNMT P40261 1/20 0.54
BAZ2B Q9UIF8 1/20 0.53
HCAR3 P49019 5/20 0.51
GRM5 P41594 1/20 0.51
HDAC6 Q9UBN7 3/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
HDAC1 Q13547 2/20 0.43
CA2 P00918 1/20 0.43
HPGD P15428 1/20 0.43
TSHR P16473 1/20 0.43
HTT P42858 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
PLK1 P53350 4/20 0.42
MKNK1 Q9BUB5 1/20 0.41
MKNK2 Q9HBH9 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29424855 1.00 NNMT (0.54) NNMTBAZ2BHCAR3GRM5HDAC6
SCHEMBL217496 0.85 NNMT (0.49) NNMTHCAR3HDAC6HDAC1CA2
SCHEMBL18715411 0.85 HCAR3 (0.70) NNMTBAZ2BHCAR3GRM5HDAC6
SCHEMBL28117859 0.82 NNMT (0.46) NNMTHCAR3HDAC6HDAC1SMN1; SMN2
Ammonia Solution, Strong SCHEMBL28249483 0.81 HCAR3 (0.65) HCAR3
SCHEMBL11005841 0.81 NNMT (0.53) NNMTHCAR3
SCHEMBL22403855 0.81 NNMT (0.46) NNMTHCAR3HDAC6HDAC1
SCHEMBL12388325 0.81 HCAR3 (0.51) NNMTHCAR3
SCHEMBL19736133 0.81 PTK2 (0.57) NNMTBAZ2BHCAR3GRM5TSHR
SCHEMBL8722229 0.79 NNMT (0.50) NNMTHCAR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 145 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122005879-A Modified GRPR antagonist peptides for cancer imaging and treatment 慕尼黑工业大学 2026-05-12 CN claimed
US-20260021211-A1 Dual mode radiotracer and -therapeutics UNIV MUENCHEN TECH (DE) 2026-01-22 US claimed
US-12419976-B2 Hybrid tracers for targeted cancer imaging and treatment ACADEMISCH ZIEKENHUIS LEIDEN (H.O.D.N. LUMC) GMBH (NL) 2025-09-23 US claimed
US-12390540-B2 Dual mode radiotracer and -therapeutics Technische Universität München (DE) 2025-08-19 US claimed
EP-4291250-B1 DUAL MODE RADIOTRACER AND THERAPEUTICS UNIV MUENCHEN TECH (DE) 2025-01-15 EP claimed
US-20240399001-A1 RADIOTRACERS AND THERAPEUTICS BINDING TO FIBROBLAST ACTIVATION PROTEIN (FAP) Blue Earth Diagnostics Limited (GB) 2024-12-05 US claimed
US-20240366811-A1 RADIONUCLIDE LABELED POLYPEPTIDE CONJUGATES AND USES THEREOF TIANJIN CONJUSTAR BIOLOGICS CO., LTD. (CN) 2024-11-07 US claimed
WO-2024222840-A1 NOVEL RADIONUCLIDE-LABELED POLYPEPTIDE CONJUGATE AND USE THEREOF 天津星联肽生物科技有限公司 2024-10-31 WO claimed
US-20240317780-A1 RADIOPHARMACEUTICAL SOMATOSTATIN RECEPTOR LIGANDS AND PRECURSORS THEREOF Technische Universität München (DE) 2024-09-26 US claimed
EP-4424378-A2 DUAL MODE RADIOTRACER AND -THERAPEUTICS Technische Universität München (DE) 2024-09-04 EP claimed
US-20220370649-A1 DUAL MODE RADIOTRACER AND -THERAPEUTICS UNIV MUENCHEN TECH (DE) 2022-11-24 US claimed
WO-2022238553-A1 RADIOPHARMACEUTICAL SOMATOSTATIN RECEPTOR LIGANDS AND PRECURSORS THEREOF Technische Universität München (DE) 2022-11-17 WO claimed
US-20220118120-A1 CANCER DIAGNOSTIC IMAGING AGENTS Technische Universität München (DE) 2022-04-21 US claimed
WO-2022018264-A1 SILICON-CONTAINING LIGAND COMPOUNDS Technische Universität München (DE) 2022-01-27 WO claimed
EP-3917582-A1 CANCER DIAGNOSTIC IMAGING AGENTS Technische Universität München (DE) 2021-12-08 EP claimed
CN-113573743-A Diagnostic imaging agents for cancer 慕尼黑工业大学 2021-10-29 CN claimed
WO-2020157184-A1 CANCER DIAGNOSTIC IMAGING AGENTS Technische Universität München (DE) 2020-08-06 WO claimed
US-20200197545-A1 DUAL MODE RADIOTRACER AND -THERAPEUTICS TECHNISCHE UNIVERSITÄT MÜNCHEN - KLINIKUM RECHTS DER ISAR (DE) 2020-06-25 US claimed
EP-3658194-A1 DUAL MODE RADIOTRACER AND -THERAPEUTICS Technische Universität München (DE) 2020-06-03 EP claimed
WO-2019020831-A1 DUAL MODE RADIOTRACER AND -THERAPEUTICS Technische Universität München (DE) 2019-01-31 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220370649-A1 DUAL MODE RADIOTRACER AND -THERAPEUTICS PAICS, SSTR2, SSTR1 NNMT 1537/4885BAZ2B 2545/4885HCAR3 1300/4885
US-12419976-B2 Hybrid tracers for targeted cancer imaging and treatment HNRNPF, ANXA3, SLC67A1 NNMT 4701/4885BAZ2B 2574/4885HCAR3 2637/4885
US-20240366811-A1 RADIONUCLIDE LABELED POLYPEPTIDE CONJUGATES AND USES THEREOF GRPR, SSTR4, DNPEP NNMT 3985/4885BAZ2B 2603/4885HCAR3 2013/4885
US-20260021211-A1 Dual mode radiotracer and -therapeutics FOLH1, SLC19A1, KLK3 NNMT 3874/4885BAZ2B 1269/4885HCAR3 1637/4885
US-20240399001-A1 RADIOTRACERS AND THERAPEUTICS BINDING TO FIBROBLAST ACTIVATION PROTEIN (FAP) FAP, FIBP, FGFR1 NNMT 4197/4885BAZ2B 2804/4885HCAR3 1746/4885
US-20200197545-A1 DUAL MODE RADIOTRACER AND -THERAPEUTICS SSTR2, SSTR1, PAICS NNMT 1583/4885BAZ2B 2240/4885HCAR3 1208/4885
US-20240317780-A1 RADIOPHARMACEUTICAL SOMATOSTATIN RECEPTOR LIGANDS AND PRECURSORS THEREOF SSTR1, SSTR3, SSTR4 NNMT 3359/4885BAZ2B 2392/4885HCAR3 145/4885
US-12390540-B2 Dual mode radiotracer and -therapeutics PAICS, SSTR2, SSTR1 NNMT 1537/4885BAZ2B 2545/4885HCAR3 1300/4885
US-20220118120-A1 CANCER DIAGNOSTIC IMAGING AGENTS FOLH1, FOLR1, KLK3 NNMT 3845/4885BAZ2B 2786/4885HCAR3 1267/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.