Salverine

Salverine

SCHEMBL25064

CCN(CC)CCOc1ccccc1C(=O)Nc1ccccc1

nearest known ligand 0.70

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.70
KDM4E B2RXH2 2/20 0.70
LMNA P02545 1/20 0.70
POLB P06746 1/20 0.60
NPSR1 Q6W5P4 1/20 0.60
MCHR1 Q99705 3/20 0.59
SGMS2 Q8NHU3 1/20 0.59
MEN1 O00255 3/20 0.59
KMT2A Q03164 3/20 0.59
RAB9A P51151 2/20 0.56
MCL1 Q07820 1/20 0.55
AURKA O14965 1/20 0.55
SMN1; SMN2 Q16637 2/20 0.54
CYP1A2 P05177 1/20 0.54
CYP3A4 P08684 1/20 0.54
CYP2C9 P11712 1/20 0.54
CYP2C19 P33261 1/20 0.54
KCNK3 O14649 1/20 0.53
KCNK9 Q9NPC2 1/20 0.53
BCHE P06276 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Salverine SCHEMBL29360867 1.00 ALDH1A1 (0.70) ALDH1A1KDM4ELMNAPOLBNPSR1
Salverine SCHEMBL29375616 0.99 ALDH1A1 (0.68) ALDH1A1KDM4ELMNAPOLBNPSR1
SCHEMBL10066976 0.86 RXFP1 (0.64) ALDH1A1KDM4ELMNAPOLBNPSR1
Salverine SCHEMBL5886094 0.86 KDM4E (0.54) ALDH1A1KDM4ELMNAPOLBNPSR1
SCHEMBL3500700 0.86 MCHR1 (0.59) ALDH1A1KDM4ELMNAPOLBNPSR1
SCHEMBL3500563 0.86 MCHR1 (0.59) ALDH1A1KDM4ELMNANPSR1MCHR1
SCHEMBL11338177 0.83 ALDH1A1 (0.76) ALDH1A1KDM4ELMNANPSR1MCHR1
SCHEMBL11756085 0.83 MCHR1 (0.58) ALDH1A1KDM4ELMNANPSR1MCHR1
Hydrochloric Acid SCHEMBL11751328 0.82 MCHR1 (0.57) ALDH1A1KDM4ELMNANPSR1MCHR1
Hydrochloric Acid SCHEMBL11671640 0.82 ALDH1A1 (0.74) ALDH1A1KDM4ELMNAPOLBMCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1104 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2560634-A1 NITRIC OXIDE RELEASING PRODRUGS OF THERAPEUTIC AGENTS Piramal Enterprises Limited (IN) 2013-02-27 EP claimed
US-20120063996-A1 NOVEL NIMESULIDE COMPOSITIONS ELAN PHARMA INTERNATIONAL LTD. 2012-03-15 US claimed
US-20110263526-A1 Nitric Oxide Releasing Prodrugs of Therapeutic Agents PIRAMAL LIFE SCIENCES LIMITED (IN) 2011-10-27 US claimed
WO-2011132171-A1 NITRIC OXIDE RELEASING PRODRUGS OF THERAPEUTIC AGENTS PIRAMAL LIFE SCIENCES LIMITED (IN) 2011-10-27 WO claimed
EP-1617816-B1 NANOPARTICULATE MELOXICAN FORMULATIONS ELAN PHARMA INT LTD (IE) 2009-05-13 EP claimed
EP-1938803-A2 Formulations comprising nanoparticulate meloxican Elan Pharma International Limited (IE) 2008-07-02 EP claimed
CN-100346832-C Pharmaceutical dosage form for transmucosal delivery PHARMACIA CORP (US) 2007-11-07 CN claimed
EP-1480624-B1 PHARMACEUTICAL TABLET PHARMACIA CORP (US) 2006-11-29 EP claimed
EP-1471890-B1 PHARMACEUTICAL DOSAGE FORM FOR MUCOSAL DELIVERY PHARMACIA CORP (US) 2006-09-27 EP claimed
CN-1829510-A Dispersible formulation of an anti-inflammatory agent PHARMACIA & UPJOHN CO LTD (US) 2006-09-06 CN claimed
WO-2004082719-A1 DISPERSIBLE PHARMACEUTICAL COMPOSITION FOR TREATMENT OF MASTITIS AND OTIC DISORDERS PHARMACIA CORPORATION (US) 2004-09-30 WO claimed
US-20040156872-A1 Novel nimesulide compositions ELAN PHARMA INTERNATIONAL LTD. 2004-08-12 US claimed
US-20030235617-A1 Pharmaceutical dosage form for mucosal delivery MCNEIL-PPC, INC 2003-12-25 US claimed
US-20030180357-A1 Pharmaceutical tablet MCNEIL-PPC, INC 2003-09-25 US claimed
EP-1336602-A1 Nitrate prodrugs able to release nitric oxide in a controlled and selective way and their use for prevention and treatment of inflammatory, ischemic and proliferative diseases Scaramuzzino, Giovanni (IT) 2003-08-20 EP claimed
WO-2003066029-A2 PHARMACEUTICAL DOSAGE FORM FOR MUCOSAL DELIVERY PHARMACIA CORPORATION (US) 2003-08-14 WO claimed
WO-2003066030-A2 PHARMACEUTICAL TABLET PHARMACIA CORPORATION (US) 2003-08-14 WO claimed
CN-1294519-A Pharmaceutical composition containing a compound having an activity of promoting the absorption of an active ingredient INPHARMA SA (CH) 2001-05-09 CN claimed
EP-1073470-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2001-02-07 EP claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040156872-A1 Novel nimesulide compositions NIM1K, NIT2, NCL ALDH1A1 3888/4885KDM4E 1888/4885LMNA 3668/4885
US-20030180357-A1 Pharmaceutical tablet GYPA, SORD, SRI ALDH1A1 1900/4885KDM4E 3204/4885LMNA 2379/4885
US-20120063996-A1 NOVEL NIMESULIDE COMPOSITIONS NIM1K, NIT2, NCL ALDH1A1 3888/4885KDM4E 1888/4885LMNA 3668/4885
US-20110263526-A1 Nitric Oxide Releasing Prodrugs of Therapeutic Agents NOS2, NOS1, NOS3 ALDH1A1 204/4885KDM4E 2388/4885LMNA 3648/4885
US-20030235617-A1 Pharmaceutical dosage form for mucosal delivery SI, UGGT1, GYPA ALDH1A1 1722/4885KDM4E 2862/4885LMNA 2639/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.