SCHEMBL2582785

SCHEMBL2582785

CCOc1nc2c(N)ncnc2n1[C@@H]1O[C@H](CO)C[C@H]1O

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSPA5 P11021 2/20 0.47
HSPA8 P11142 2/20 0.47
RXFP1 Q9HBX9 1/20 0.45
LMNA P02545 1/20 0.43
TP53 P04637 1/20 0.43
HBB P68871 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
ADORA3 P0DMS8 2/20 0.42
ADORA2A P29274 1/20 0.42
HSD17B10 Q99714 1/20 0.42
GAPDH P04406 1/20 0.42
POLB P06746 1/20 0.42
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
AMD1 P17707 2/20 0.41
HSP90B1 P14625 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29328694 0.91 HSPA8 (0.48) HSPA5HSPA8RXFP1LMNATP53
SCHEMBL14034324 0.86 AMD1 (0.55) HSPA5HSPA8RXFP1ADORA3ADORA2A
SCHEMBL3701954 0.83 NADK (0.57) HSPA5HSPA8RXFP1LMNAADORA3
SCHEMBL19680323 0.83 AHCY (0.55) HSPA5HSPA8RXFP1LMNATP53
SCHEMBL3704527 0.83 NADK (0.57) HSPA5HSPA8RXFP1LMNAADORA3
SCHEMBL6761931 0.81 HSPA8 (0.72) HSPA5HSPA8RXFP1LMNATP53
SCHEMBL6761939 0.81 HSPA8 (0.72) HSPA5HSPA8RXFP1LMNATP53
SCHEMBL14544481 0.77 HSPA8 (0.60) HSPA5HSPA8RXFP1LMNATP53
SCHEMBL15629276 0.76 AMD1 (0.39) HSPA5HSPA8RXFP1ADORA3AMD1
Cordycepin SCHEMBL24220702 0.74 ADORA3 (0.63) SMN1; SMN2ADORA3ADORA2AGAPDHPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10100076-B2 Modified nucleosides for the treatment of viral infections and abnormal cellular proliferation GILEAD PHARMASSET LLC (US) 2018-10-16 US disclosed
US-20140057863-A1 MODIFIED NUCLEOSIDES FOR THE TREATMENT OF VIRAL INFECTIONS AND ABNORMAL CELLULAR PROLIFERATION GILEAD SCIENCES, INC. (US) 2014-02-27 US disclosed
EP-2251015-B1 Modified nucleosides for the treatment of viral infections and abnormal cellular proliferation GILEAD PHARMASSET LLC (US) 2013-02-20 EP disclosed
US-20110269707-A1 Modified nucleosides for the treatment of viral infections and abnormal cellullar proliferation PHARMASSET, INC. 2011-11-03 US disclosed
EP-2251015-A1 Modified nucleosides for the treatment of viral infections and abnormal cellular proliferation Pharmasset, Inc. (US) 2010-11-17 EP disclosed
EP-1411954-A2 MODIFIED NUCLEOSIDES FOR TREATMENT OF VIRAL INFECTIONS AND ABNORMAL CELLULAR PROLIFERATION Pharmasset Limited (BB) 2004-04-28 EP disclosed
US-20030087873-A1 Modified nucleosides for the treatment of viral infections and abnormal cellular proliferation PHARMASSET, INC. 2003-05-08 US disclosed
WO-2002032920-A2 MODIFIED NUCLEOSIDES FOR TREATMENT OF VIRAL INFECTIONS AND ABNORMAL CELLULAR PROLIFERATION PHARMASSET LIMITED (BB) 2002-04-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140057863-A1 MODIFIED NUCLEOSIDES FOR THE TREATMENT OF VIRAL INFECTIONS AND ABNORMAL CELLULAR PROLIFERATION SLC29A1, PNP, SLC29A2 HSPA5 1617/4885HSPA8 4823/4885RXFP1 800/4885
US-20110269707-A1 Modified nucleosides for the treatment of viral infections and abnormal cellullar proliferation PNP, ALPP, XDH HSPA5 2063/4885HSPA8 4599/4885RXFP1 515/4885
US-10100076-B2 Modified nucleosides for the treatment of viral infections and abnormal cellular proliferation SLC29A1, SLC29A2, PNP HSPA5 2286/4885HSPA8 4839/4885RXFP1 768/4885
US-20030087873-A1 Modified nucleosides for the treatment of viral infections and abnormal cellular proliferation SLC29A1, PNP, SLC29A2 HSPA5 1835/4885HSPA8 4815/4885RXFP1 657/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.