SCHEMBL2584542

SCHEMBL2584542

CC[C@@](CCC(=O)c1ccc(F)c(F)c1F)(NC(=O)OC(C)(C)C)C(=O)O

nearest known ligand 0.33

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33
CTSS P25774 3/20 0.32
AAK1 Q2M2I8 3/20 0.32
CTSK P43235 2/20 0.32
ALDH1A1 P00352 2/20 0.32
MAPT P10636 2/20 0.32
KDM4E B2RXH2 1/20 0.32
GAA P10253 1/20 0.32
PKM P14618 1/20 0.32
HPGD P15428 1/20 0.32
ALOX12 P18054 1/20 0.32
RIPK1 Q13546 1/20 0.32
GPR119 Q8TDV5 1/20 0.32
AKT1 P31749 2/20 0.31
PPARG P37231 2/20 0.30
PPARA Q07869 2/20 0.30
S1PR3 Q99500 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2578534 0.86 ACKR3 (0.40) CES2CES1CTSSAAK1CTSK
SCHEMBL2587766 0.86 CTSS (0.35) CES2CES1CTSSAAK1CTSK
SCHEMBL2588069 0.84 AAK1 (0.34) CTSSAAK1CTSK
SCHEMBL2586648 0.83 MEN1 (0.31) CTSSCTSKGAA
SCHEMBL2581151 0.82 CHRNA1 (0.36) CES2CES1AAK1ALDH1A1MAPT
SCHEMBL2584672 0.82 AAK1 (0.34) CES2CES1CTSSAAK1CTSK
SCHEMBL2588125 0.80 AAK1 (0.36) CTSSAAK1CTSKRIPK1
SCHEMBL2585429 0.78 CTSS (0.33) CTSSAAK1CTSKAKT1
SCHEMBL2575528 0.78 ALDH1A1 (0.47) ALDH1A1MAPTGAAPKMHPGD
SCHEMBL2587439 0.77 CTSS (0.41) CES2CES1CTSSCTSKMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8048878-B2 Two cyclic cinnamide compound EISAI R&D MANAGEMENT CO., LTD. (JP) 2011-11-01 US disclosed