SCHEMBL2588069

SCHEMBL2588069

CC[C@@](CCC(=O)c1cc(F)c(F)cc1F)(NC(=O)OC(C)(C)C)C(=O)O

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 3/20 0.34
POLB P06746 1/20 0.32
APEX1 P27695 1/20 0.32
CTSS P25774 3/20 0.31
CTSK P43235 3/20 0.31
ACE P12821 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2587766 0.88 CTSS (0.35) AAK1CTSSCTSKACE
SCHEMBL2578534 0.88 ACKR3 (0.40) AAK1CTSSCTSK
SCHEMBL2581151 0.84 CHRNA1 (0.36) AAK1
SCHEMBL2584542 0.84 CES2 (0.33) AAK1CTSSCTSK
SCHEMBL2584672 0.84 AAK1 (0.34) AAK1CTSSCTSKACE
SCHEMBL2588125 0.84 AAK1 (0.36) AAK1CTSSCTSKACE
SCHEMBL2585429 0.82 CTSS (0.33) AAK1CTSSCTSKACE
SCHEMBL2586648 0.80 MEN1 (0.31) CTSSCTSK
SCHEMBL2587439 0.79 CTSS (0.41) CTSSCTSK
SCHEMBL2463123 0.76 CTSK (0.35) CTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8048878-B2 Two cyclic cinnamide compound EISAI R&D MANAGEMENT CO., LTD. (JP) 2011-11-01 US disclosed