SCHEMBL2585429

SCHEMBL2585429

CC[C@@](CCC(=O)c1cc(F)cc(F)c1)(NC(=O)OC(C)(C)C)C(=O)O

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSS P25774 3/20 0.33
CTSK P43235 2/20 0.33
AAK1 Q2M2I8 4/20 0.32
SLC6A3 Q01959 1/20 0.32
LMNA P02545 1/20 0.32
ACE P12821 1/20 0.31
GABRB1 P18505 1/20 0.30
GABRB2 P47870 1/20 0.30
AKT1 P31749 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2584672 0.89 AAK1 (0.34) CTSSCTSKAAK1ACE
SCHEMBL2587439 0.89 CTSS (0.41) CTSSCTSKLMNA
SCHEMBL2588125 0.87 AAK1 (0.36) CTSSCTSKAAK1ACE
SCHEMBL2581151 0.85 CHRNA1 (0.36) AAK1SLC6A3GABRB1GABRB2
SCHEMBL2588069 0.82 AAK1 (0.34) CTSSCTSKAAK1ACE
SCHEMBL2578534 0.82 ACKR3 (0.40) CTSSCTSKAAK1
SCHEMBL2587766 0.82 CTSS (0.35) CTSSCTSKAAK1ACE
SCHEMBL2575528 0.81 ALDH1A1 (0.47) LMNA
SCHEMBL2583802 0.80 ERCC5 (0.42) SLC6A3LMNA
SCHEMBL2584542 0.78 CES2 (0.33) CTSSCTSKAAK1AKT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8048878-B2 Two cyclic cinnamide compound EISAI R&D MANAGEMENT CO., LTD. (JP) 2011-11-01 US disclosed