SCHEMBL2587766

SCHEMBL2587766

CC[C@@](CCC(=O)c1cc(F)ccc1F)(NC(=O)OC(C)(C)C)C(=O)O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 3/20 0.35
CTSK P43235 3/20 0.35
CES2 O00748 1/20 0.35
CES1 P23141 1/20 0.35
AAK1 Q2M2I8 6/20 0.34
GPR119 Q8TDV5 1/20 0.34
DRD2 P14416 1/20 0.33
RIPK1 Q13546 1/20 0.33
ERAP1 Q9NZ08 1/20 0.32
HPGD P15428 2/20 0.32
MEN1 O00255 1/20 0.32
TSHR P16473 1/20 0.32
MAPK1 P28482 1/20 0.32
KMT2A Q03164 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
S1PR3 Q99500 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2578534 0.91 ACKR3 (0.40) CTSSCTSKCES2CES1AAK1
SCHEMBL2588069 0.88 AAK1 (0.34) CTSSCTSKAAK1ACE
SCHEMBL2584542 0.86 CES2 (0.33) CTSSCTSKCES2CES1AAK1
SCHEMBL2581151 0.83 CHRNA1 (0.36) CES2CES1AAK1HPGDMEN1
SCHEMBL2588125 0.83 AAK1 (0.36) CTSSCTSKAAK1RIPK1ACE
SCHEMBL2587439 0.83 CTSS (0.41) CTSSCTSKCES2CES1HPGD
SCHEMBL2585429 0.82 CTSS (0.33) CTSSCTSKAAK1ACE
SCHEMBL2584672 0.81 AAK1 (0.34) CTSSCTSKCES2CES1AAK1
SCHEMBL2586648 0.80 MEN1 (0.31) CTSSCTSKMEN1KMT2AGAA
SCHEMBL2575528 0.77 ALDH1A1 (0.47) DRD2HPGDMEN1TSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8048878-B2 Two cyclic cinnamide compound EISAI R&D MANAGEMENT CO., LTD. (JP) 2011-11-01 US disclosed