SCHEMBL260615

SCHEMBL260615

O=C(O)c1n[nH]c2ccc(Br)cc12

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 2/20 0.61
JAK2 O60674 2/20 0.61
PRKAG1 P54619 9/20 0.55
PRKAA1 Q13131 9/20 0.55
PRKAB1 Q9Y478 9/20 0.55
DYRK1A Q13627 2/20 0.54
DCLK1 O15075 1/20 0.54
PRKD3 O94806 1/20 0.54
MAP4K4 O95819 1/20 0.54
CHEK2 O96017 1/20 0.54
CSF1R P07333 1/20 0.54
FER P16591 1/20 0.54
CDK2 P24941 1/20 0.54
MARK3 P27448 1/20 0.54
FLT4 P35916 1/20 0.54
FLT3 P36888 1/20 0.54
MAPK9 P45984 1/20 0.54
CSNK1D P48730 1/20 0.54
CLK2 P49760 1/20 0.54
CSNK2A1 P68400 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11015155 0.89 JAK2 (0.51) PDPK1JAK2PRKAG1PRKAA1PRKAB1
SCHEMBL261067 0.86 IDO1 (0.62) PDPK1JAK2PRKAG1PRKAA1PRKAB1
SCHEMBL30075258 0.86 IDO1 (0.62) PDPK1JAK2PRKAG1PRKAA1PRKAB1
SCHEMBL17039120 0.85 JAK2 (0.64) PDPK1JAK2PRKAG1PRKAA1PRKAB1
SCHEMBL9436096 0.85 PDPK1 (0.59) PDPK1JAK2PRKAG1PRKAA1PRKAB1
SCHEMBL4291226 0.81 KDM4E (0.63) PDPK1JAK2PRKAG1PRKAA1PRKAB1
SCHEMBL13386937 0.81 YTHDC1 (0.63) PDPK1JAK2DYRK1ADCLK1PRKD3
SCHEMBL21496911 0.81 PDPK1 (0.54) PDPK1JAK2PRKAG1PRKAA1PRKAB1
SCHEMBL26204518 0.81 PDPK1 (0.58) PDPK1JAK2DYRK1ADCLK1PRKD3
SCHEMBL1963463 0.81 PRKAG1 (0.56) PDPK1PRKAG1PRKAA1PRKAB1HAO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 365 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005082885-A1 IMIDAZOLE BASED KINASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2005-09-09 WO claimed
US-12558341-B2 Oral complement factor D inhibitors BIOCRYST PHARMACEUTICALS, INC. (US) 2026-02-24 US disclosed
US-12485109-B2 Pyrrolo 12.3-dipyrimidine compounds and analogues thereof BIOCRYST PHARMACEUTICALS, INC. (US) 2025-12-02 US disclosed
US-12486277-B2 CDK inhibitors and their use as pharmaceuticals Prelude Therapeutis Incorporated (US) 2025-12-02 US disclosed
US-20250243181-A2 NOVEL INDAZOLE DERIVATIVE AND USE THEREOF KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2025-07-31 US disclosed
EP-4585596-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND, PHARMACEUTICAL COMPOSITION THEREOF, AND USE THEREOF Shanghai Yingli Pharmaceutical Co., Ltd (CN) 2025-07-16 EP disclosed
WO-2025133961-A1 NITROGEN-CONTAINING HETEROARYL COMPOUNDS FOR THE TREATMENT OF CHRONIC DISEASES PFIZER INC. (US) 2025-06-26 WO disclosed
US-12338230-B2 Aryl, heteroaryl, and heterocyclic compounds for treatment of immune and inflammatory disorders ACHILLION PHARMACEUTICALS, INC. (US) 2025-06-24 US disclosed
US-20250186391-A1 ORAL COMPLEMENT FACTOR D INHIBITORS WILMINGTON TRUST, NATIONAL ASSOCIATION 2025-06-12 US disclosed
WO-2025103409-A1 NMT INHIBITOR, PREPARATION METHOD THEREFOR, AND USE THEREOF 南京同诺康医药科技有限公司 2025-05-22 WO disclosed
CN-1684962-A Indazoles, benzothiazoles, and benzisothiazoles, and preparation and use thereof MEMORY PHARM CORP (US) 2005-10-19 CN disclosed
WO-2005092890-A2 INDAZOLES, BENZOTHIAZOLES, BENZOISOTHIAZOLES, BENZISOXAZOLES, AND PREPARATION AND USES THEREOF MEMORY PHARMACEUTICALS CORPORATION (US) 2005-10-06 WO disclosed
US-20050208582-A1 Pyrazole compounds and pharmaceutical compositions comprising the compound EISAI R&D MANAGEMENT CO., LTD. (JP) 2005-09-22 US disclosed
CN-1656079-A Pyrazole compounds and pharmaceutical compositions containing the same EISAI CO LTD (JP) 2005-08-17 CN disclosed
EP-1543000-A1 INDAZOLES, BENZOTHIAZOLES, AND BENZOISOTHIAZOLES, AND PREPARATION AND USES THEREOF Memory Pharmaceuticals Corporation (US) 2005-06-22 EP disclosed
US-20050090529-A1 3,5 Disubstituted indazole compounds with nitrogen-bearing 5-membered heterocycles, pharmaceutical compositions, and methods for mediating or inhibiting cell proliferation PFIZER INC 2005-04-28 US disclosed
EP-1510516-A1 PYRAZOLE COMPOUND AND MEDICINAL COMPOSITION CONTAINING THE SAME Eisai Co., Ltd. (JP) 2005-03-02 EP disclosed
US-20040132790-A1 Indazoles, benzothiazoles, and benzoisothiazoles, and preparation and uses thereof MEMORY PHARMACEUTICALS CORPORATION 2004-07-08 US disclosed
WO-2004029050-A1 INDAZOLES, BENZOTHIAZOLES, AND BENZOISOTHIAZOLES, AND PREPARATION AND USES THEREOF MEMORY PHARMACEUTICALS CORPORATION (US) 2004-04-08 WO disclosed
WO-2004029050-A1 INDAZOLES, BENZOTHIAZOLES, AND BENZOISOTHIAZOLES, AND PREPARATION AND USES THEREOF MEMORY PHARMACEUTICALS CORPORATION (US) 2004-04-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12485109-B2 Pyrrolo 12.3-dipyrimidine compounds and analogues thereof C5, DPYD, C9 PDPK1 676/4885JAK2 1382/4885PRKAG1 2962/4885
US-20040132790-A1 Indazoles, benzothiazoles, and benzoisothiazoles, and preparation and uses thereof CHRNA5, CHRNA7, CHRNA3 PDPK1 1949/4885JAK2 2278/4885PRKAG1 2169/4885
US-12486277-B2 CDK inhibitors and their use as pharmaceuticals CDK6, CDK3, CDK9 PDPK1 179/4885JAK2 448/4885PRKAG1 346/4885
US-12338230-B2 Aryl, heteroaryl, and heterocyclic compounds for treatment of immune and inflammatory disorders CFD, TFPI, CFH PDPK1 1487/4885JAK2 1224/4885PRKAG1 4345/4885
US-20250243181-A2 NOVEL INDAZOLE DERIVATIVE AND USE THEREOF TRIB2, YAP1, IDO2 PDPK1 1076/4885JAK2 2764/4885PRKAG1 2754/4885
US-12558341-B2 Oral complement factor D inhibitors CFD, CFH, CFB PDPK1 4006/4885JAK2 4305/4885PRKAG1 4785/4885
US-20050090529-A1 3,5 Disubstituted indazole compounds with nitrogen-bearing 5-membered heterocycles, pharmaceutical compositions, and methods for mediating or inhibiting cell proliferation CDK3, CDK4, CDK9 PDPK1 110/4885JAK2 262/4885PRKAG1 750/4885
US-20250186391-A1 ORAL COMPLEMENT FACTOR D INHIBITORS CFD, CFH, CFB PDPK1 2921/4885JAK2 4719/4885PRKAG1 4698/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.