SCHEMBL2632415

SCHEMBL2632415

N#Cc1ccc(N(C2=NC3=NC(N(c4ccc(C#N)cc4)c4ccc(C(F)(F)F)cc4)=NC4=NC(N(c5ccc(C#N)cc5)c5ccc(C(F)(F)F)cc5)=NC(=N2)N34)c2ccc(C(F)(F)F)cc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.49
CYP3A4 P08684 3/20 0.42
CYP3A5 P20815 2/20 0.42
CYP19A1 P11511 10/20 0.40
MAOB P27338 1/20 0.38
MLYCD O95822 1/20 0.35
DGAT1 O75907 1/20 0.34
SOAT1 P35610 1/20 0.34
KCNH2 Q12809 1/20 0.34
NR1H3 Q13133 1/20 0.34
VNN1 O95497 1/20 0.34
RORC P51449 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2632322 0.88 CYP2A6 (0.34) CYP3A4CYP19A1
SCHEMBL2623748 0.86 RORC (0.37) KIF11CYP3A4CYP3A5CYP19A1MAOB
SCHEMBL2632428 0.82 CYP3A4 (0.40) KIF11CYP3A4CYP19A1
SCHEMBL2632320 0.82 TSHR (0.39) CYP19A1MAOB
SCHEMBL2623746 0.78
SCHEMBL2623742 0.77 DHFR (0.37) KIF11CYP3A4CYP19A1
SCHEMBL26044351 0.76 KIF11 (0.40) KIF11CYP3A4CYP19A1
SCHEMBL8324537 0.75 KIF11 (0.53) KIF11CYP3A4CYP3A5CYP19A1MAOB
SCHEMBL2623745 0.74 ABCG2 (0.32)
SCHEMBL524351 0.73 KIF11 (0.86) KIF11CYP3A4CYP3A5CYP19A1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120091884-A1 HEPTAAZAPHENALENE DERIVATIVES AND USE THEREOF IN ORGANIC ELECTROLUMINESCENT DEVICE COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AT) 2012-04-19 US disclosed
WO-2010132953-A1 HEPTAAZAPHENALENE DERIVATIVES AND USE THEREOF IN ORGANIC ELECTROLUMINESCENT DEVICE COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2010-11-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120091884-A1 HEPTAAZAPHENALENE DERIVATIVES AND USE THEREOF IN ORGANIC ELECTROLUMINESCENT DEVICE HSD17B2, CYP1A2, HSD17B1 KIF11 1884/4885CYP3A4 36/4885CYP3A5 35/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.