SCHEMBL265015

SCHEMBL265015

COC(=O)c1ccc2ncccc2c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 1.00
HTT P42858 1/20 1.00
PLK1 P53350 1/20 0.68
NPC1 O15118 4/20 0.58
RAB9A P51151 4/20 0.58
TAS1R3 Q7RTX0 1/20 0.56
TAS1R1 Q7RTX1 1/20 0.56
DOT1L Q8TEK3 1/20 0.56
ALDH1A1 P00352 5/20 0.55
POLB P06746 2/20 0.55
MAPT P10636 2/20 0.54
MEN1 O00255 1/20 0.54
KMT2A Q03164 1/20 0.54
HDAC1 Q13547 1/20 0.53
HDAC2 Q92769 1/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
GAA P10253 2/20 0.53
CYP19A1 P11511 1/20 0.52
CYP11B1 P15538 1/20 0.52
CYP11B2 P19099 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30718649 1.00 ALOX15 (1.00) ALOX15HTTPLK1NPC1RAB9A
SCHEMBL27928930 0.98 ALOX15 (0.97) ALOX15HTTPLK1NPC1RAB9A
Quinoline SCHEMBL28071393 0.95 ALOX15 (0.91) ALOX15HTTPLK1NPC1RAB9A
Sulfuric Acid SCHEMBL28071302 0.92 ALOX15 (0.84) ALOX15HTTPLK1NPC1RAB9A
SCHEMBL18371293 0.88 ALOX15 (0.78) ALOX15HTTPLK1NPC1RAB9A
SCHEMBL29893321 0.87 ALOX15 (0.77) ALOX15HTTPLK1NPC1RAB9A
SCHEMBL2671065 0.87 ALOX15 (0.77) ALOX15HTTPLK1NPC1RAB9A
Quinoline SCHEMBL28161564 0.86 ALOX15 (0.76) ALOX15HTTPLK1NPC1RAB9A
SCHEMBL25294487 0.85 HTT (0.74) ALOX15HTTPLK1NPC1RAB9A
SCHEMBL2492569 0.84 ALOX15 (0.73) ALOX15HTTPLK1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 501 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117205211-B Application of quinoline compound in preparation of fish parasitic protozoan resisting medicine 西北农林科技大学深圳研究院 2024-04-05 CN claimed
CN-117205211-A Application of quinoline compound in preparation of fish parasitic protozoan resisting medicine 西北农林科技大学深圳研究院 2023-12-12 CN claimed
CN-110229102-B 2-alkylated quinoline, derivative and synthetic method thereof 湘潭大学 2022-05-17 CN claimed
CN-110229102-A 2- is alkylated quinoline, derivative and its synthetic method 湘潭大学 2019-09-13 CN claimed
US-10224485-B2 Process for preparing a crystalline organic semiconductor material BASF SE (DE) 2019-03-05 US claimed
US-20170012208-A1 ORGANIC SEMICONDUCTOR FORMULATIONS USINVEST LLC 2017-01-12 US claimed
EP-4745134-A1 PROTEIN ARGINASE METHYLTRANSFERASE-5 INHIBITOR AND MEDICAL USE THEREOF Jiangsu Yahong Meditech Co., Ltd. (CN) 2026-05-20 EP disclosed
US-12577243-B2 Monoacylglycerol lipase modulators JANSSEN PHARMACEUTICA NV (BE) 2026-03-17 US disclosed
EP-3856178-B1 MONOACYLGLYCEROL LIPASE MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2026-03-11 EP disclosed
WO-2025087033-A1 COMPOUND CONTAINING (1,3,4-THIADIAZOLE)BENZENE-1,2-ETHYLENEDIAMINE, PREPARATION METHOD THEREFOR AND USE THEREOF 中国海洋大学 2025-05-01 WO disclosed
US-12227524-B2 Anti-infective compounds INSTITUT PASTEUR KOREA (KR) 2025-02-18 US disclosed
CN-119325469-A WEE1 degrading compounds and uses thereof 百时美施贵宝公司 2025-01-17 CN disclosed
CN-119285426-A Synthesis method of diaryl acetylene 南京工业大学 2025-01-10 CN disclosed
US-6284796-B1 NAPHTHAMIDINE COMPOUNDS ABBOTT LABORATORIES 2001-09-04 US disclosed
CN-1268942-A Sulfonamide compounds and medicinal use thereof FUJISAWA PHARMACEUTICAL CO (JP) 2000-10-04 CN disclosed
US-6093729-A TREATING ARRHYTHMIAS, PROPHYLAXIS OF CARDIAC INFARCTION, ANGINA PECTORIS AND ISCHEMIC CONDITIONS OF THE HEART, SHOCK CONDITIONS, USING IN SURGICAL OPERATIONS AND ORGAN TRANSPLANTATIONS, CELL PROLIFERATION, HYPERTENSION HOECHST AKTIENGESELLSCHAFT (DE) 2000-07-25 US disclosed
CN-1117045-A Substituted bicyclic heteroaroylguanidines, a process for their preparation, their use as a medicament or a diagnostic agent, and a medicament containing them HOECHST AG (DE) 1996-02-21 CN disclosed
EP-0240859-B1 LIPOXYGENASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 1993-04-28 EP disclosed
US-4968803-A FLUORINE AS OXIDANT ALLIED-SIGNAL INC. (US) 1990-11-06 US disclosed
CN-85100796-A The preparation method of qualone derivative 1986-10-01 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12577243-B2 Monoacylglycerol lipase modulators MGLL, LPL, FAAH ALOX15 356/4885HTT 3651/4885PLK1 3246/4885
US-12227524-B2 Anti-infective compounds RABGGTB, ELANE, SERPINB1 ALOX15 1708/4885HTT 3860/4885PLK1 893/4885
US-10224485-B2 Process for preparing a crystalline organic semiconductor material STOM, SPOP, TTR ALOX15 4022/4885HTT 2419/4885PLK1 273/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.