SCHEMBL265489

SCHEMBL265489

CN(CC=O)Cc1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.52
TSHR P16473 2/20 0.52
CARM1 Q86X55 1/20 0.52
PRMT6 Q96LA8 1/20 0.52
PRMT8 Q9NR22 1/20 0.52
LMNA P02545 2/20 0.50
USP2 O75604 1/20 0.50
CYP3A4 P08684 1/20 0.50
MAOA P21397 1/20 0.50
MAOB P27338 1/20 0.50
PYCR1 P32322 1/20 0.50
SMN1; SMN2 Q16637 2/20 0.48
BLM P54132 1/20 0.48
AOC3 Q16853 1/20 0.48
SIGMAR1 Q99720 1/20 0.47
KDM4E B2RXH2 1/20 0.47
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
CA12 O43570 1/20 0.46
CA9 Q16790 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7324033 0.81 ALDH1A1 (0.54) ALDH1A1TSHRCARM1PRMT6PRMT8
SCHEMBL7937668 0.80 CARM1 (0.58) ALDH1A1TSHRCARM1PRMT6PRMT8
SCHEMBL29956348 0.80 KDM4E (0.42) ALDH1A1TSHRUSP2CYP3A4PYCR1
SCHEMBL19910402 0.80 CYP2D6 (0.48) MAOAMAOB
Dibemethine SCHEMBL10542007 0.79 ALDH1A1 (0.70) ALDH1A1TSHRCARM1PRMT6PRMT8
Dibemethine SCHEMBL276863 0.79 ALDH1A1 (0.70) ALDH1A1TSHRCARM1PRMT6PRMT8
SCHEMBL185582 0.79 PYCR1 (0.67) ALDH1A1TSHRCARM1PRMT6PRMT8
SCHEMBL1650495 0.78 CA2 (0.47) ALDH1A1TSHRAOC3KDM4ENPC1
SCHEMBL16924691 0.78 CHRNB2 (0.67) ALDH1A1LMNAKDM4E
SCHEMBL9687347 0.78 ALDH1A1 (0.50) ALDH1A1TSHRCARM1PRMT6PRMT8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 198 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12258316-B2 Biphenyl compounds useful as muscarinic receptor antagonists THERAVANCE BIOPHARMA R&D IP, LLC (US) 2025-03-25 US claimed
US-20220306579-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE BIOPHARMA R&D IP, LLC (US) 2022-09-29 US claimed
EP-2044083-A1 ANTIVIRAL AGENTS GENELABS TECHNOLOGIES, INC. (US) 2009-04-08 EP claimed
US-20080051384-A1 ANTIVIRAL AGENTS GENELABS TECHNOLOGIES, INC. 2008-02-28 US claimed
WO-2008008912-A1 ANTIVIRAL AGENTS GENELABS TECHNOLOGIES, INC. (US) 2008-01-17 WO claimed
WO-2008008907-A2 ANTIVIRAL AGENTS GENELABS TECHNOLOGIES, INC. (US) 2008-01-17 WO claimed
US-20060211698-A1 Bicyclic heteroaryl derivatives for treating viruses GENELABS, INC. 2006-09-21 US claimed
US-20060058553-A1 Novel bicyclic hydroxamates as inhibitors of histone deacetylase AXYS PHARMACEUTICALS, INC. (US) 2006-03-16 US claimed
EP-1472216-A2 NOVEL BICYCLIC HYDROXAMATES AS INHIBITORS OF HISTONE DEACETYLASE Axys Pharmaceuticals (US) 2004-11-03 EP claimed
WO-2003066579-A2 NOVEL BICYCLIC HYDROXAMATES AS INHIBITORS OF HISTONE DEACETYLASE AXYS PHARMACEUTICALS (US) 2003-08-14 WO claimed
US-12258316-B2 Biphenyl compounds useful as muscarinic receptor antagonists THERAVANCE BIOPHARMA R&D IP, LLC (US) 2025-03-25 US disclosed
US-20240327352-A1 NOVEL PROCESS FOR THE PREPARATION OF 1-(2-{4-[(4-CARBAMOYLPIPERIDIN-1-YL)METHYL]- N-METHYLBENZAMIDO}ETHYL)PIPERIDIN-4-YL N-({1,1'-BIPHENYL}-2-YL)CARBAMATE MSN LABORATORIES PRIVATE LTD, R&D CENTER (IN) 2024-10-03 US disclosed
CN-117263850-A Synthesis method of raffinacine 华中药业股份有限公司 2023-12-22 CN disclosed
US-20220388981-A1 CRYSTALLINE FORMS OF A BIPHENYL COMPOUND THERAVANCE BIOPHARMA R&D IP LLC (US) 2022-12-08 US disclosed
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
WO-2005087736-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2005-09-22 WO disclosed
US-20050203133-A1 Biphenyl compounds useful as muscarinic receptor antagonists THERAVANCE, INC. 2005-09-15 US disclosed
US-20050203131-A1 Biphenyl compounds useful as muscarinic receptor antagonists THERAVANCE, INC. (US) 2005-09-15 US disclosed
US-20050203137-A1 Biphenyl compounds useful as muscarinic receptor antagonists THERAVANCE, INC. 2005-09-15 US disclosed
US-20050203138-A1 Biphenylylaminocarbonyl-amino- or -oxypiperidine derivatives, e.g., biphenyl-2-ylcarbamic acid 1-[2-((4-[(4-hydroxybenzylamino)methyl]benzoyl)methylamino)ethyl]piperidin-4-yl ester; treating bronchodilation, asthma and chronic obstructive pulmonary disease (COPD) THERAVANCE, INC. 2005-09-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (11 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220306579-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS CHRM2, CHRM1, CHRM3 ALDH1A1 1082/4885TSHR 68/4885CARM1 587/4885
US-20050203131-A1 Biphenyl compounds useful as muscarinic receptor antagonists CHRM2, CHRM3, CHRM1 ALDH1A1 1207/4885TSHR 92/4885CARM1 793/4885
US-20220388981-A1 CRYSTALLINE FORMS OF A BIPHENYL COMPOUND FFAR1, FFAR4, FFAR3 ALDH1A1 2252/4885TSHR 3505/4885CARM1 3175/4885
US-20050203133-A1 Biphenyl compounds useful as muscarinic receptor antagonists CHRM2, CHRM1, CHRM3 ALDH1A1 1082/4885TSHR 68/4885CARM1 587/4885
US-20050203138-A1 Biphenylylaminocarbonyl-amino- or -oxypiperidine derivatives, e.g., biphenyl-2-ylcarbamic acid 1-[2-((4-[(4-hydroxybenzylamino)methyl]benzoyl)methylamino)ethyl]piperidin-4-yl ester; treating bronchodilation, asthma and chronic obstructive pulmonary disease (COPD) CHRM1, CHRM2, CHRM3 ALDH1A1 828/4885TSHR 426/4885CARM1 260/4885
US-20060211698-A1 Bicyclic heteroaryl derivatives for treating viruses HAVCR2, ZC3HAV1, SARS1 ALDH1A1 1627/4885TSHR 4537/4885CARM1 1625/4885
US-12258316-B2 Biphenyl compounds useful as muscarinic receptor antagonists CHRM2, CHRM1, CHRM3 ALDH1A1 1082/4885TSHR 68/4885CARM1 587/4885
US-20240327352-A1 NOVEL PROCESS FOR THE PREPARATION OF 1-(2-{4-[(4-CARBAMOYLPIPERIDIN-1-YL)METHYL]- N-METHYLBENZAMIDO}ETHYL)PIPERIDIN-4-YL N-({1,1'-BIPHENYL}-2-YL)CARBAMATE CYP4B1, CYP1B1, KDM4B ALDH1A1 250/4885TSHR 2899/4885CARM1 87/4885
US-20080051384-A1 ANTIVIRAL AGENTS EIF2AK2, MAVS, ZC3HAV1 ALDH1A1 1357/4885TSHR 4492/4885CARM1 4190/4885
US-20050203137-A1 Biphenyl compounds useful as muscarinic receptor antagonists CHRM2, CHRM1, CHRM3 ALDH1A1 1670/4885TSHR 76/4885CARM1 800/4885
US-20060058553-A1 Novel bicyclic hydroxamates as inhibitors of histone deacetylase HDAC1, HDAC2, HDAC11 ALDH1A1 1478/4885TSHR 3583/4885CARM1 145/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.