SCHEMBL2659802

SCHEMBL2659802

Cc1ccsc1S(=O)(=O)Nc1cc(OC(F)(F)F)cc2cc(C(=O)NCC(CN3CCOCC3)SCc3ccccc3)[nH]c12

nearest known ligand 0.32

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTSS P25774 3/20 0.32
CTSL P07711 1/20 0.32
CTSK P43235 1/20 0.32
KDM4E B2RXH2 3/20 0.32
MAPT P10636 2/20 0.32
ALDH1A1 P00352 2/20 0.32
WNT3A P56704 3/20 0.32
NPSR1 Q6W5P4 1/20 0.32
ABL1 P00519 1/20 0.32
KCNH2 Q12809 1/20 0.32
HSD17B10 Q99714 1/20 0.31
BRD4 O60885 1/20 0.30
CASR P41180 1/20 0.30
NPC1 O15118 1/20 0.30
CRHBP P24387 1/20 0.30
CRHR2 Q13324 1/20 0.30
MCL1 Q07820 2/20 0.30
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2660075 0.88 MAPT (0.36) KDM4EMAPTALDH1A1NPSR1HSD17B10
SCHEMBL2659987 0.86 LGALS8 (0.33) KDM4EMCL1
SCHEMBL2660524 0.84 RAB9A (0.35) KDM4EMAPTALDH1A1NPSR1MCL1
SCHEMBL2661758 0.84 LGALS8 (0.32) KDM4EMAPTNPC1MCL1
SCHEMBL2659804 0.81 CTSS (0.33) CTSSCTSLCTSKKDM4EMAPT
SCHEMBL2659015 0.81 HDAC3 (0.32) MAPTLMNA
SCHEMBL2660508 0.78 SYK (0.33) KDM4EMAPTALDH1A1NPSR1HSD17B10
SCHEMBL2661595 0.78 BDKRB1 (0.32)
SCHEMBL2661312 0.77 MAPT (0.39) KDM4EMAPTALDH1A1NPSR1HSD17B10
SCHEMBL2668802 0.76 ITGB3 (0.33) KDM4EMAPTALDH1A1NPSR1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074119-A1 INDOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2009-07-01 EP disclosed
WO-2008050821-A1 INDOLE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-05-02 WO disclosed