SCHEMBL2715618

SCHEMBL2715618

CC(N)c1cccc(OC(F)(F)F)c1

nearest known ligand 0.46

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 7/20 0.43
SLC6A4 P31645 2/20 0.43
GPR139 Q6DWJ6 1/20 0.42
SLC6A3 Q01959 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1728892 1.00 SLC6A2 (0.43) SLC6A2SLC6A4GPR139SLC6A3
SCHEMBL1727565 1.00 SLC6A2 (0.43) SLC6A2SLC6A4GPR139SLC6A3
Hydrochloric Acid SCHEMBL2719228 0.98 SLC6A2 (0.44) SLC6A2SLC6A4GPR139SLC6A3
Hydrochloric Acid SCHEMBL14737983 0.98 SLC6A2 (0.44) SLC6A2SLC6A4GPR139SLC6A3
Hydrochloric Acid SCHEMBL16989095 0.98 SLC6A2 (0.44) SLC6A2SLC6A4GPR139SLC6A3
SCHEMBL21801025 0.90 SLC6A2 (0.42) SLC6A2
SCHEMBL4550413 0.86 CETP (0.44)
SCHEMBL16233093 0.86 DUT (0.40) SLC6A2SLC6A4
SCHEMBL24588079 0.85 TRPM8 (0.41) SLC6A2
SCHEMBL760742 0.85 TRPM8 (0.41) SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 60 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250002452-A1 BICYCLOPENTANE DERIVATIVES ANGELINI PHARMA S.P.A. (IT) 2025-01-02 US disclosed
EP-4479377-A1 NEW BICYCLOPENTANE DERIVATIVES Icagen, LLC (US) 2024-12-25 EP disclosed
CN-118829626-A Novel dicyclopentane derivatives 伊卡根有限责任公司 2024-10-22 CN disclosed
US-20230303486-A1 CYCLOBUTYL-UREA DERIVATIVES IDORSIA PHARMACEUTICALS LTD (CH) 2023-09-28 US disclosed
EP-4241843-A2 ALCOHOL DERIVATIVES AS KV7 POTASSIUM CHANNEL OPENERS H. Lundbeck A/S (DK) 2023-09-13 EP disclosed
WO-2023158584-A1 NEW BICYCLOPENTANE DERIVATIVES ICAGEN, LLC (US) 2023-08-24 WO disclosed
EP-3755684-B1 ALCOHOL DERIVATIVES AS KV7 POTASSIUM CHANNEL OPENERS H LUNDBECK AS (DK) 2023-07-12 EP disclosed
EP-4172140-A1 CYCLOBUTYL-UREA DERIVATIVES Idorsia Pharmaceuticals Ltd (CH) 2023-05-03 EP disclosed
CN-115702141-A Cyclobutyl-urea derivatives 爱杜西亚药品有限公司 2023-02-14 CN disclosed
CN-113508109-B Substituted heterocyclic amide compound, preparation method and medical application thereof 劲方医药科技(上海)有限公司 2023-02-10 CN disclosed
US-20080139640-A1 Hydroxamates, Their Manufacture And Use As Pharmaceutical Agents HOFFMANN-LA ROCHE, INC. 2008-06-12 US disclosed
US-7273866-B2 2-aryl thiazole derivatives as KCNQ modulators BRISTOL-MYERS SQUIBB COMPANY (US) 2007-09-25 US disclosed
CN-1964963-A Hydroxamates, their manufacture and use as pharmaceutical agents HOFFMANN LA ROCHE (CH) 2007-05-16 CN disclosed
CN-1646493-A 5HT2cReceptor modulators ARENA PHARM INC (US) 2005-07-27 CN disclosed
US-6831080-B2 E.g., 3-(2-fluorophenyl)-N-(1-(3-morpholin-4-yl)phenyl)-propyl)acrylamide; disorders responsive to opening of KCNQ potassium channels; analgesics; migraine, bipolar disorders, anticonvulsants, antiepileptic, anxiolytic agents BRISTOL-MYERS SQUIBB COMPANY 2004-12-14 US disclosed
US-20040147401-A1 2-aryl thiazole derivatives as KCNQ modulators BRISTOL-MYERS SQUIBB COMPANY 2004-07-29 US disclosed
WO-2004060281-A2 2-ARYL THIAZOLE DERIVATIVES AS KCNQ MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-07-22 WO disclosed
US-20030166650-A1 Cinnamide derivatives as KCNQ potassium channel modulators BRISTOL-MYERS SQUIBB COMPANY 2003-09-04 US disclosed
US-5028256-A Metolachlor and an acylamide compound, for maize or sorghum CIBA-GEIGY CORPORATION (US) 1991-07-02 US disclosed
US-4897109-A ACYLAMINE DERIVATIVE CIBA-GEIGY CORPORATION (US) 1990-01-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250002452-A1 BICYCLOPENTANE DERIVATIVES BICRA, C1R, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16 SLC6A2 4227/4885SLC6A4 4133/4885GPR139 772/4885
US-20230303486-A1 CYCLOBUTYL-UREA DERIVATIVES KCNA4, KCNMB4, KCNA7 SLC6A2 3599/4885SLC6A4 2283/4885GPR139 2801/4885
US-20030166650-A1 Cinnamide derivatives as KCNQ potassium channel modulators KCNH2, KCNH3, KCNQ1 SLC6A2 1495/4885SLC6A4 1115/4885GPR139 315/4885
US-20080139640-A1 Hydroxamates, Their Manufacture And Use As Pharmaceutical Agents HCAR3, HCAR1, HCAR2 SLC6A2 1252/4885SLC6A4 530/4885GPR139 1912/4885
US-20040147401-A1 2-aryl thiazole derivatives as KCNQ modulators KCNJ2, KCNT1, KCNQ1 SLC6A2 1127/4885SLC6A4 766/4885GPR139 281/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.