SCHEMBL2737282

SCHEMBL2737282

CC(C)c1ccc(-c2cccnc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 4/20 0.60
CYP3A4 P08684 2/20 0.60
ALDH1A1 P00352 1/20 0.60
CYP1A2 P05177 1/20 0.60
KIF11 P52732 1/20 0.56
MKNK1 Q9BUB5 4/20 0.52
MKNK2 Q9HBH9 4/20 0.52
CYP11B2 P19099 2/20 0.52
CYP19A1 P11511 2/20 0.52
CYP17A1 P05093 1/20 0.52
CYP11B1 P15538 1/20 0.52
GPR55 Q9Y2T6 3/20 0.50
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
CA12 O43570 1/20 0.49
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
CA9 Q16790 1/20 0.49
NPC1 O15118 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29631885 0.85 CYP2A6 (0.56) CYP2A6CYP3A4ALDH1A1CYP1A2KIF11
SCHEMBL29337469 0.85 CYP2A6 (0.56) CYP2A6CYP3A4ALDH1A1CYP1A2KIF11
SCHEMBL10035332 0.83 UCHL3 (0.47) CYP2A6CYP3A4ALDH1A1CYP1A2KIF11
SCHEMBL24534338 0.82 CYP2A6 (0.88) CYP2A6CYP3A4ALDH1A1CYP1A2KIF11
SCHEMBL29360677 0.82 CYP2A6 (0.88) CYP2A6CYP3A4ALDH1A1CYP1A2KIF11
SCHEMBL13907273 0.82 CYP2A6 (0.88) CYP2A6CYP3A4ALDH1A1CYP1A2KIF11
SCHEMBL11996116 0.82 CYP2A6 (0.58) CYP2A6CYP3A4ALDH1A1CYP1A2KIF11
SCHEMBL12360035 0.82 NPC1 (0.54) CYP2A6CYP3A4ALDH1A1CYP1A2KIF11
SCHEMBL21003619 0.82 CYP2A6 (0.52) CYP2A6CYP3A4ALDH1A1CYP1A2KIF11
SCHEMBL11996114 0.82 CYP19A1 (0.54) CYP2A6CYP3A4ALDH1A1CYP1A2KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 98 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240018115-A1 ALLOSTERIC CHROMENONE INHIBITORS OF PHOSPHOINOSITIDE 3-KINASE (PI3K) FOR THE TREATMENT OF DISEASE LOXO ONCOLOGY, INC. 2024-01-18 US disclosed
WO-2023227734-A1 FLAVIVIRUS INHIBITORS IRBM S.P.A. (IT) 2023-11-30 WO disclosed
US-20230365556-A1 N-ACYL AMINO ACID COMPOUNDS AND METHODS OF USE PLIANT THERAPEUTICS, INC. (US) 2023-11-16 US disclosed
US-11806335-B2 Heterocyclic carboxylate compounds as glycolate oxidase inhibitors Lilac Therapeutics, Inc. (US) 2023-11-07 US disclosed
US-11806335-B2 Heterocyclic carboxylate compounds as glycolate oxidase inhibitors Lilac Therapeutics, Inc. (US) 2023-11-07 US disclosed
US-11795159-B2 Compounds for the treatment of SARS PURDUE RESEARCH FOUNDATION (US) 2023-10-24 US disclosed
US-11795159-B2 Compounds for the treatment of SARS PURDUE RESEARCH FOUNDATION (US) 2023-10-24 US disclosed
US-11718583-B2 Nitrogen-containing compound, electronic component using same and electronic device SHAANXI LIGHTE OPTOELECTRONICS MATERIAL CO., LTD. (CN) 2023-08-08 US disclosed
US-20230192671-A1 COMPOUNDS FOR THE TREATMENT OF SARS PURDUE RESEARCH FOUNDATION 2023-06-22 US disclosed
US-20230192671-A1 COMPOUNDS FOR THE TREATMENT OF SARS PURDUE RESEARCH FOUNDATION 2023-06-22 US disclosed
US-20090105279-A1 Antiviral protease inhibitors GILEAD SCIENCES, INC. 2009-04-23 US disclosed
US-20090099096-A1 AZA-peptide protease inhibitors GILEAD SCIENCES, INC. 2009-04-16 US disclosed
US-20090087409-A1 Viral Polymerase Inhibitors BOEHRINGER INGELHEIM (CANADA) LTD. (CA) 2009-04-02 US disclosed
US-20080200475-A1 4-Piperazinothieno[2,3-D] Pyrimidine Compounds As Platelet Aggregation Inhibitors PFIZER INC. 2008-08-21 US disclosed
US-20080200475-A1 4-Piperazinothieno[2,3-D] Pyrimidine Compounds As Platelet Aggregation Inhibitors PFIZER INC. 2008-08-21 US disclosed
US-20080194590-A1 4-Piperazinylthieno [2,3-D] Pyrimidine Compounds as Platelet Aggregation Inhibitors PFIZER INC 2008-08-14 US disclosed
US-20080176857-A1 4-Piperazinnylthieno[2,3-d]Pyrimidine Compounds as Platelet Aggregation Inhibitors PFIZER INC. 2008-07-24 US disclosed
US-20080176857-A1 4-Piperazinnylthieno[2,3-d]Pyrimidine Compounds as Platelet Aggregation Inhibitors PFIZER INC. 2008-07-24 US disclosed
US-7361654-B2 Substituted heteroaryl amide modulators of glucocorticoid receptor, AP-1, and/or NF-κB activity and use thereof BRISTOL-MYERS SQUIBB CO. (US) 2008-04-22 US disclosed
US-20070232610-A1 Novel compounds that are ERK inhibitors SCHERING CORPORATION 2007-10-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (13 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090087409-A1 Viral Polymerase Inhibitors NR2C2, NR4A1, MED25 CYP2A6 98/4885CYP3A4 322/4885ALDH1A1 3616/4885
US-11806335-B2 Heterocyclic carboxylate compounds as glycolate oxidase inhibitors UGDH, PGD, PNPO CYP2A6 599/4885CYP3A4 555/4885ALDH1A1 184/4885
US-20240018115-A1 ALLOSTERIC CHROMENONE INHIBITORS OF PHOSPHOINOSITIDE 3-KINASE (PI3K) FOR THE TREATMENT OF DISEASE PIK3CA, PIK3R4, PIK3R5 CYP2A6 833/4885CYP3A4 610/4885ALDH1A1 3412/4885
US-20080176857-A1 4-Piperazinnylthieno[2,3-d]Pyrimidine Compounds as Platelet Aggregation Inhibitors TBXA2R, P2RY4, PF4 CYP2A6 171/4885CYP3A4 152/4885ALDH1A1 622/4885
US-20080194590-A1 4-Piperazinylthieno [2,3-D] Pyrimidine Compounds as Platelet Aggregation Inhibitors PFKP, PF4, P2RY4 CYP2A6 267/4885CYP3A4 294/4885ALDH1A1 1204/4885
US-20090105279-A1 Antiviral protease inhibitors ACE, TMPRSS15, MME CYP2A6 2088/4885CYP3A4 1420/4885ALDH1A1 3629/4885
US-11795159-B2 Compounds for the treatment of SARS ACE2, ACE, SARS1 CYP2A6 1672/4885CYP3A4 344/4885ALDH1A1 3093/4885
US-11718583-B2 Nitrogen-containing compound, electronic component using same and electronic device EXOC1, NOS1, EXOSC10 CYP2A6 4002/4885CYP3A4 2434/4885ALDH1A1 2244/4885
US-20070232610-A1 Novel compounds that are ERK inhibitors MAPK1, MAPK4, MAPKAPK2 CYP2A6 2394/4885CYP3A4 2048/4885ALDH1A1 342/4885
US-20230192671-A1 COMPOUNDS FOR THE TREATMENT OF SARS ACE2, ACE, SARS1 CYP2A6 1672/4885CYP3A4 344/4885ALDH1A1 3093/4885
US-20080200475-A1 4-Piperazinothieno[2,3-D] Pyrimidine Compounds As Platelet Aggregation Inhibitors PF4, TBXA2R, P2RY4 CYP2A6 140/4885CYP3A4 325/4885ALDH1A1 849/4885
US-20230365556-A1 N-ACYL AMINO ACID COMPOUNDS AND METHODS OF USE ITGA1, ITGB1, ITGAL CYP2A6 4288/4885CYP3A4 4404/4885ALDH1A1 524/4885
US-20090099096-A1 AZA-peptide protease inhibitors DNPEP, ANPEP, PEPD CYP2A6 3049/4885CYP3A4 2794/4885ALDH1A1 4015/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.