SCHEMBL2741417

SCHEMBL2741417

c1ccc(-c2cc(-n3c4ccccc4c4ccc5c(c6ccccc6n5-c5cc6ccccc6c6ccccc56)c43)cc(-c3ccccc3)n2)cc1

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
KDM4E B2RXH2 2/20 0.31
L3MBTL1 Q9Y468 2/20 0.31
ATM Q13315 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2741413 0.88 ALDH1A1 (0.32) KDM4EL3MBTL1ATM
SCHEMBL2741414 0.87 KDM4E (0.33) CYP1A2KDM4EL3MBTL1ATM
SCHEMBL18086287 0.87 L3MBTL1 (0.44) CYP1A2CYP2C9CYP2C19KDM4EL3MBTL1
SCHEMBL10029935 0.86 L3MBTL1 (0.46) KDM4EL3MBTL1ATM
SCHEMBL12131960 0.86 L3MBTL1 (0.46) KDM4EL3MBTL1ATM
SCHEMBL26472290 0.85 L3MBTL1 (0.35) CYP1A2CYP2C9CYP2C19KDM4EL3MBTL1
SCHEMBL19769614 0.85 KDM4E (0.40) CYP1A2CYP2C9CYP2C19KDM4EL3MBTL1
SCHEMBL2741412 0.84 KDM4E (0.36) KDM4EL3MBTL1ATM
SCHEMBL22596583 0.84 HTR6 (0.38) KDM4EL3MBTL1ATM
SCHEMBL19342709 0.84 CYP11B1 (0.34) CYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11233201-B2 Organic electroluminescent devices and preparation methods thereof KUNSHAN GO-VISIONOX OPTO-ELECTRONICS CO., LTD. (CN) 2022-01-25 US disclosed
US-10693107-B2 Organic electroluminescence device having RGB pixel areas BEIJING VISIONOX TECHNOLOGY CO., LTD. (CN) 2020-06-23 US disclosed
US-20170373276-A1 ORGANIC ELECTROLUMINESCENCE DEVICE HAVING RGB PIXEL AREAS BEIJING VISIONOX TECHNOLOGY CO., LTD. (CN) 2017-12-28 US disclosed
US-20150166886-A1 FLUORESCENCE AND DELAYED FLUORESCENCE-TYPE ORGANIC LIGHT-EMITTING MATERIAL AND ELEMENT KYUSHU UNIVERSITY, NATIONAL UNIVERSITY CORPORATION (JP) 2015-06-18 US disclosed
US-20150166886-A1 FLUORESCENCE AND DELAYED FLUORESCENCE-TYPE ORGANIC LIGHT-EMITTING MATERIAL AND ELEMENT KYUSHU UNIVERSITY, NATIONAL UNIVERSITY CORPORATION (JP) 2015-06-18 US disclosed
US-8993129-B2 Fluorescence and delayed fluorescence-type organic light-emitting material and element NIPPON STEEL & SUMIKIN CHEMICAL CO., LTD. (JP) 2015-03-31 US disclosed
US-8993129-B2 Fluorescence and delayed fluorescence-type organic light-emitting material and element NIPPON STEEL & SUMIKIN CHEMICAL CO., LTD. (JP) 2015-03-31 US disclosed
US-8962158-B2 Material having indolocarbazole compound for phosphorescent light-emitting element and organic electroluminescent element using the same NIPPON STEEL & SUMIKIN CHEMICAL CO., LTD. (JP) 2015-02-24 US disclosed
US-8962158-B2 Material having indolocarbazole compound for phosphorescent light-emitting element and organic electroluminescent element using the same NIPPON STEEL & SUMIKIN CHEMICAL CO., LTD. (JP) 2015-02-24 US disclosed
EP-2416397-B1 MATERIAL FOR PHOSPHORESCENT LIGHT-EMITTING ELEMENT AND ORGANIC ELECTROLUMINESCENT ELEMENT USING SAME NIPPON STEEL & SUMIKIN CHEM CO (JP) 2014-08-20 EP disclosed
US-20120241732-A1 ORGANIC LIGHT-EMITTING MATERIAL AND ORGANIC LIGHT-EMITTING ELEMENT NIPPON STEEL CHEMICAL & MATERIAL CO., LTD. (JP) 2012-09-27 US disclosed
US-20120241732-A1 ORGANIC LIGHT-EMITTING MATERIAL AND ORGANIC LIGHT-EMITTING ELEMENT NIPPON STEEL CHEMICAL & MATERIAL CO., LTD. (JP) 2012-09-27 US disclosed
US-20120001165-A1 MATERIAL FOR PHOSPHORESCENT LIGHT-EMITTING ELEMENT AND ORGANIC ELECTROLUMINESCENT ELEMENT USING SAME NIPPON STEEL CHEMICAL & MATERIAL CO., LTD. (JP) 2012-01-05 US disclosed
US-20120001165-A1 MATERIAL FOR PHOSPHORESCENT LIGHT-EMITTING ELEMENT AND ORGANIC ELECTROLUMINESCENT ELEMENT USING SAME NIPPON STEEL CHEMICAL & MATERIAL CO., LTD. (JP) 2012-01-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150166886-A1 FLUORESCENCE AND DELAYED FLUORESCENCE-TYPE ORGANIC LIGHT-EMITTING MATERIAL AND ELEMENT LEF1, EML4, TEAD1 CYP1A2 764/4885CYP2C9 1306/4885CYP2C19 751/4885
US-10693107-B2 Organic electroluminescence device having RGB pixel areas RHEB, CYBA, RUVBL2 CYP1A2 2306/4885CYP2C9 986/4885CYP2C19 1395/4885
US-20120001165-A1 MATERIAL FOR PHOSPHORESCENT LIGHT-EMITTING ELEMENT AND ORGANIC ELECTROLUMINESCENT ELEMENT USING SAME LEF1, ELOC, ELP1 CYP1A2 1445/4885CYP2C9 1938/4885CYP2C19 1045/4885
US-20170373276-A1 ORGANIC ELECTROLUMINESCENCE DEVICE HAVING RGB PIXEL AREAS RUVBL2, RHEB, RUVBL1 CYP1A2 2668/4885CYP2C9 1272/4885CYP2C19 1884/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.