Gamma-Cyclodextrin

Gamma-Cyclodextrin

SCHEMBL2780992

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nearest known ligand 0.95

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Gamma-Cyclodextrin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 known ✓ O15379 1/20 0.50
HDAC1 known ✓ Q13547 1/20 0.50
HDAC2 known ✓ Q92769 1/20 0.50
HDAC8 known ✓ Q9BY41 1/20 0.50
HDAC6 known ✓ Q9UBN7 1/20 0.50
SLC6A2 known ✓ P23975 1/20 0.46
HTR2C known ✓ P28335 1/20 0.46
HTR2B known ✓ P41595 1/20 0.46
SLC6A3 known ✓ Q01959 1/20 0.46
ALDH1A1 P00352 2/20 0.95
TSHR P16473 2/20 0.95
LMNA P02545 1/20 0.95
TDP1 Q9NUW8 1/20 0.95
TXNRD1 Q16881 6/20 0.74
TXNRD3 Q86VQ6 6/20 0.74
TXNRD2 Q9NNW7 6/20 0.74
FYN P06241 1/20 0.46
MAOA P21397 1/20 0.46
LGALS1 P09382 2/20 0.35
LGALS3 P17931 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Betadex SCHEMBL692932 1.00 ALDH1A1 (0.95) ALDH1A1TSHRLMNATDP1TXNRD1
Alfadex SCHEMBL11030738 1.00 ALDH1A1 (0.95) ALDH1A1TSHRLMNATDP1TXNRD1
Alfadex SCHEMBL28176234 1.00 ALDH1A1 (0.95) ALDH1A1TSHRLMNATDP1TXNRD1
Alfadex SCHEMBL2432145 1.00 ALDH1A1 (0.95) ALDH1A1TSHRLMNATDP1TXNRD1
Betadex SCHEMBL7195429 0.98 ALDH1A1 (0.91) ALDH1A1TSHRLMNATDP1TXNRD1
Gamma-Cyclodextrin SCHEMBL25455463 0.98 ALDH1A1 (1.00) ALDH1A1TSHRLMNATDP1TXNRD1
Alfadex SCHEMBL23188277 0.98 ALDH1A1 (1.00) ALDH1A1TSHRLMNATDP1TXNRD1
Gamma-Cyclodextrin SCHEMBL25455531 0.98 ALDH1A1 (1.00) ALDH1A1TSHRLMNATDP1TXNRD1
Betadex SCHEMBL23188251 0.98 ALDH1A1 (1.00) ALDH1A1TSHRLMNATDP1TXNRD1
Gamma-Cyclodextrin SCHEMBL20533920 0.98 ALDH1A1 (1.00) ALDH1A1TSHRLMNATDP1TXNRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119452101-A Compositions and methods for nucleic acid sequencing 因美纳公司 2025-02-14 CN claimed
CN-119095982-A Palladium catalyst compositions and methods for sequencing-by-synthesis 伊路米纳有限公司 2024-12-06 CN claimed
US-8435966-B2 Associations of xanthogenates and cyclodextrins, and their use BIOSPHINGS AG (DE) 2013-05-07 US claimed
US-20100240606-A1 ASSOCIATIONS OF XANTHOGENATES AND CYCLODEXTRINS, AND THEIR USE BIOSPHINGS AG (DE) 2010-09-23 US claimed
US-6284269-B1 Pharmaceutical compositions of meloxicam with improved solubility and bioavailability HEXAL AG (DE) 2001-09-04 US claimed
EP-1007049-A1 NEW PHARMACEUTICAL COMPOSITIONS OF MELOXICAM WITH IMPROVED SOLUBILITY AND BIOAVAILABILITY Hexal AG (DE) 2000-06-14 EP claimed
WO-1999009988-A1 NEW PHARMACEUTICAL COMPOSITIONS OF MELOXICAM WITH IMPROVED SOLUBILITY AND BIOAVAILABILITY HEXAL AG (DE) 1999-03-04 WO claimed
CN-119095982-A Palladium catalyst compositions and methods for sequencing-by-synthesis 伊路米纳有限公司 2024-12-06 CN disclosed
CN-112961124-B Method for treating sewage by using microbial preparation 杭州楠大环保科技有限公司 2022-06-21 CN disclosed
CN-112961124-A Method for treating sewage by using microbial preparation 杭州楠大环保科技有限公司 2021-06-15 CN disclosed
CN-112585457-A Systems, devices, and methods for gas sensing 麻省理工学院 2021-03-30 CN disclosed
CN-107626337-A A kind of loaded Ag/g C3N4The preparation method of aerogel microball 东北林业大学 2018-01-26 CN disclosed
US-8435966-B2 Associations of xanthogenates and cyclodextrins, and their use BIOSPHINGS AG (DE) 2013-05-07 US disclosed
US-20100240606-A1 ASSOCIATIONS OF XANTHOGENATES AND CYCLODEXTRINS, AND THEIR USE BIOSPHINGS AG (DE) 2010-09-23 US disclosed
WO-2010086129-A1 INCLUSION COMPLEX COMPRISING CINACALCET AND CYCLODEXTRIN RATHIOPHARM GMBH (DE) 2010-08-05 WO disclosed
CN-1671421-A Inclusion complexes of rosiglitazone GLAXO GROUP LTD (GB) 2005-09-21 CN disclosed
US-6284269-B1 Pharmaceutical compositions of meloxicam with improved solubility and bioavailability HEXAL AG (DE) 2001-09-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100240606-A1 ASSOCIATIONS OF XANTHOGENATES AND CYCLODEXTRINS, AND THEIR USE HLA-DRB1, CXCR3, ANTXR2 HDAC3 2096/4885HDAC1 1496/4885HDAC2 2435/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.