Chromone

Chromone

SCHEMBL27856502

O.O=c1ccoc2ccccc12

nearest known ligand 0.95

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Chromone. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE known ✓ P22303 1/20 0.51
MEN1 known ✓ O00255 1/20 0.43
PARP1 known ✓ P09874 1/20 0.41
ADORA3 known ✓ P0DMS8 1/20 0.41
DPP4 known ✓ P27487 1/20 0.41
MAOA P21397 6/20 0.95
MAOB P27338 6/20 0.95
FTO Q9C0B1 2/20 0.95
GRM5 P41594 1/20 0.51
KDM4E B2RXH2 2/20 0.47
DAO P14920 1/20 0.43
HPGD P15428 3/20 0.43
ALDH1A1 P00352 2/20 0.43
CYP3A4 P08684 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
LMNA P02545 1/20 0.43
KMT2A Q03164 1/20 0.43
GLA P06280 1/20 0.43
MAPT P10636 1/20 0.43
PGAM1 P18669 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Chromone SCHEMBL26661260 1.00 MAOA (0.95) MAOAMAOBFTOACHEGRM5
Chromone SCHEMBL30075941 0.98 MAOA (1.00) MAOAMAOBFTOACHEGRM5
Chromone SCHEMBL29369932 0.98 MAOA (1.00) MAOAMAOBFTOACHEGRM5
Chromone SCHEMBL6347379 0.98 MAOA (1.00) MAOAMAOBFTOACHEGRM5
Chromone SCHEMBL28268880 0.98 MAOA (1.00) MAOAMAOBFTOACHEGRM5
Chromone SCHEMBL37994 0.98 MAOA (1.00) MAOAMAOBFTOACHEGRM5
Chromone SCHEMBL1034108 0.95 MAOA (0.95) MAOAMAOBFTOACHEGRM5
Chromone SCHEMBL31277121 0.95 MAOA (0.95) MAOAMAOBFTOACHEGRM5
Chromone SCHEMBL31622445 0.95 MAOA (0.95) MAOAMAOBFTOACHEGRM5
Chromone SCHEMBL3203755 0.95 MAOA (0.95) MAOAMAOBFTOACHEGRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 56 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115385884-A Extraction and separation method of new chromone alcohols in purslane and application thereof 辽宁中医药大学 2022-11-25 CN claimed
CN-106397445-A Pyrazoles N-p-bromophenyl maleimide derivative containing chromone structure as well as preparation method and application thereof 绍兴文理学院 2017-02-15 CN claimed
CN-105924445-A Pyrazole-type N-p-nitrophenyl maleimide derivative containing chromone structure, and preparation method and application thereof 绍兴文理学院 2016-09-07 CN claimed
CN-105906634-A 3-(6-bromine-4-oxygen-4H-chromone)-1-phenyl-5-p-methoxyphenyl-1, 6a-pyrroline (3, 4-c) pyrazole-4, 6(3aH, 5H)-diketone and preparation method and application thereof 绍兴文理学院 2016-08-31 CN claimed
CN-105906632-A Pyrazole-type N-p-methylphenyl maleimide derivative with chromone structure, and preparation method and application thereof 绍兴文理学院 2016-08-31 CN claimed
CN-105859724-A 3-(6-bromo-4-oxy-4H-chromone)-1-phenyl-5-p-chlorphenyl-1,6a-dihydro pyrroline[3,4-c] pyrazole-4,6(3aH,5H)-diketone and preparation method and application thereof 绍兴文理学院 2016-08-17 CN claimed
CN-115385884-B Extraction and separation method of neochronol in purslane and application thereof 辽宁中医药大学 2023-04-25 CN disclosed
CN-115716790-A Extraction and separation method and application of amide ester alkaloid in purslane 辽宁中医药大学 2023-02-28 CN disclosed
CN-115385884-A Extraction and separation method of new chromone alcohols in purslane and application thereof 辽宁中医药大学 2022-11-25 CN disclosed
CN-115385884-A Extraction and separation method of new chromone alcohols in purslane and application thereof 辽宁中医药大学 2022-11-25 CN disclosed
CN-112535282-A Food for regulating diabetes 深圳市华韵生物科技产业有限公司 2021-03-23 CN disclosed
CN-109700997-A A kind of External-applicationtraditional traditional Chinese medicinal and preparation method thereof for set a broken bone section disease 贵州苗老吉药业有限公司 2019-05-03 CN disclosed
CN-107955013-B A kind of method of the preparation method of Benzofurantone compound hamaudol and detection wherein optical isomer 南京美新诺医药科技有限公司 2019-02-15 CN disclosed
CN-104147147-A Traditional Chinese medicinal composition for treating skin diseases and preparation method thereof HENAN MINGXUAN FOOD TECHNOLOGY CO LTD 2014-11-19 CN disclosed
CN-104127558-A Heat-clearing and detoxifying traditional Chinese medicine composition for livestock, and preparation method and application thereof HENAN JINERKANG ANIMAL PHARMACEUTICAL CO LTD 2014-11-05 CN disclosed
CN-104107215-A Medicinal composition for treating allergic rhinitis PANG HAILING 2014-10-22 CN disclosed
CN-103989763-A Compound arthritis capsules for treating hemophilia joint diseases, and preparation method thereof SHAANXI UNIVERSITY S INST OF HEMOPHILIA 2014-08-20 CN disclosed
CN-103585452-A Traditional Chinese medicinal composition for treating xerophthalmia XIE LIKE 2014-02-19 CN disclosed
CN-102488096-B Natural plant feedstuff additive, preparation method thereof, and feedstuff INST AGRI RESOURCES CAAS 2013-04-10 CN disclosed
CN-102488096-A Natural plant feedstuff additive, preparation method thereof, and feedstuff INST AGRI RESOURCES CAAS 2012-06-13 CN disclosed