SCHEMBL28046665

SCHEMBL28046665

NC(=O)c1cc2ccc(-c3cccc(F)c3)nc2[nH]1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 1/20 0.51
KMO O15229 2/20 0.45
CDC7 O00311 1/20 0.43
NUDT1 P36639 1/20 0.42
FYN P06241 1/20 0.41
MAP4K4 O95819 4/20 0.41
PIN1 Q13526 1/20 0.41
SLC9A1 P19634 1/20 0.41
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
MAPT P10636 1/20 0.40
KMT2A Q03164 1/20 0.40
ATR Q13535 1/20 0.40
CCNT1 O60563 1/20 0.40
CCND1 P24385 1/20 0.40
CCNC P24863 1/20 0.40
CDK8 P49336 1/20 0.40
CDK7 P50613 1/20 0.40
CDK9 P50750 1/20 0.40
CCNH P51946 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28046616 0.85 PARP1 (0.47) CDC7KDM4EPARP1ROCK2ROCK1
SCHEMBL28046612 0.84 DHODH (0.46) KMOCDC7NUDT1PIN1SLC9A1
SCHEMBL28046684 0.83 KMO (0.44) KMONUDT1MEN1MAPTKMT2A
SCHEMBL28046666 0.81 ROCK2 (0.56) CDC7MAPTPARP1ROCK2ROCK1
SCHEMBL28046677 0.77 ALPL (0.45) MAPTCCNCCDK8ROCK2ROCK1
SCHEMBL28046615 0.77 PARP1 (0.49) CDC7NUDT1SLC9A1ATRPARP1
SCHEMBL28046667 0.77 KMO (0.42) KMONUDT1KDM4EMEN1MAPT
SCHEMBL28046609 0.77 CASP1 (0.43) CDC7NUDT1ROCK2ROCK1CHEK2
SCHEMBL28046664 0.77 MAP4K4 (0.46) KMONUDT1MAP4K4MAPTCCNC
SCHEMBL28046611 0.75 MAPT (0.54) SLC9A1KDM4EMEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105294688-A 6-chlorine-N-(substituted benzyl)-1H-pyrrolo[2,3-b]pyridine-2-amide compound and preparation method as well as application thereof UNIV BEIJING TECHNOLOGY 2016-02-03 CN disclosed