SCHEMBL28047249

SCHEMBL28047249

O=COC(Cc1ccc(Cn2ccccc2=O)cc1)Cc1cn[nH]c1

nearest known ligand 0.37

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 18/20 0.37
POLB P06746 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
KLK1 P06870 2/20 0.34
ROCK2 O75116 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28869739 0.81 KLKB1 (0.36) KLKB1POLBNPSR1KLK1
SCHEMBL29437752 0.80 POLB (0.45) KLKB1POLBNPSR1KLK1ROCK2
SCHEMBL28825963 0.79 KLKB1 (0.38) KLKB1KLK1
SCHEMBL28047241 0.78 NOS2 (0.33) ROCK2
SCHEMBL28787513 0.78 ROCK1 (0.37) ROCK2
SCHEMBL27972554 0.78 ROCK2 (0.41) ROCK2
SCHEMBL27545407 0.76 FFAR1 (0.38)
SCHEMBL28868753 0.73 LDHA (0.41) POLBROCK2
SCHEMBL27809130 0.72 ALDH1A1 (0.35)
SCHEMBL28832869 0.72 FDPS (0.38) ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105143201-B Benzyl amine derivative 卡尔维斯塔制药有限公司 2019-02-22 CN disclosed
CN-105452240-A Heterocyclic derivates KALVISTA PHARMACEUTICALS LTD 2016-03-30 CN disclosed
CN-105143201-A Benzylamine derivatives KALVISTA PHARMACEUTICALS LTD 2015-12-09 CN disclosed